MX2007012445A - Forma cristalina de maleato de asenapina. - Google Patents

Forma cristalina de maleato de asenapina.

Info

Publication number
MX2007012445A
MX2007012445A MX2007012445A MX2007012445A MX2007012445A MX 2007012445 A MX2007012445 A MX 2007012445A MX 2007012445 A MX2007012445 A MX 2007012445A MX 2007012445 A MX2007012445 A MX 2007012445A MX 2007012445 A MX2007012445 A MX 2007012445A
Authority
MX
Mexico
Prior art keywords
orthorhombic
dibenz
chloro
trans
methyl
Prior art date
Application number
MX2007012445A
Other languages
English (en)
Spanish (es)
Inventor
Gerhardus Johannes Heeres
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36617328&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2007012445(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Organon Nv filed Critical Organon Nv
Publication of MX2007012445A publication Critical patent/MX2007012445A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
MX2007012445A 2005-04-07 2006-04-06 Forma cristalina de maleato de asenapina. MX2007012445A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05102742 2005-04-07
EP05102969 2005-04-14
PCT/EP2006/061408 WO2006106135A1 (en) 2005-04-07 2006-04-06 Crystal form of asenapine maleate

Publications (1)

Publication Number Publication Date
MX2007012445A true MX2007012445A (es) 2007-11-07

Family

ID=36617328

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2007012445A MX2007012445A (es) 2005-04-07 2006-04-06 Forma cristalina de maleato de asenapina.

Country Status (31)

Country Link
EP (2) EP1710245B1 (zh)
JP (1) JP5058151B2 (zh)
KR (1) KR101422843B1 (zh)
AR (1) AR056306A1 (zh)
AT (2) ATE418556T1 (zh)
AU (1) AU2006231617B2 (zh)
BR (1) BRPI0609741A8 (zh)
CA (1) CA2603509C (zh)
CY (2) CY1106902T1 (zh)
DE (2) DE602006000080T2 (zh)
DK (2) DK1917267T3 (zh)
DO (1) DOP2006000082A (zh)
ES (2) ES2318742T3 (zh)
GT (1) GT200600135A (zh)
HN (1) HN2006014095A (zh)
HR (1) HRP20070429T3 (zh)
IL (1) IL186355A (zh)
MX (1) MX2007012445A (zh)
MY (1) MY137969A (zh)
NO (1) NO340520B1 (zh)
NZ (1) NZ562124A (zh)
PE (1) PE20061311A1 (zh)
PL (2) PL1710245T3 (zh)
PT (2) PT1917267E (zh)
RS (1) RS50532B (zh)
RU (1) RU2405786C2 (zh)
SI (2) SI1710245T1 (zh)
SV (1) SV2006002473A (zh)
TW (1) TWI364423B (zh)
UY (1) UY29459A1 (zh)
WO (1) WO2006106135A1 (zh)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2667668A1 (en) * 2006-10-06 2008-04-10 N.V. Organon Amorphous asenapine and processes for preparing same
AU2010264670A1 (en) * 2009-06-24 2012-01-19 Merck Sharp & Dohme B.V. Injectable formulations containing asenapine and method of treatment using same
AU2011268335A1 (en) 2010-06-18 2013-01-10 Dr. Reddy's Laboratories Ltd. Asenapine maleate
WO2012066565A2 (en) * 2010-11-16 2012-05-24 Cadila Healthcare Limited Asenapine maleate amorphous and crystalline form and process for preparation thereof
EP2468750A1 (en) 2010-12-13 2012-06-27 Chemo Ibérica, S.A. Polymorphic forms of asenapine maleate and processes for their preparation
WO2012123325A1 (en) 2011-03-11 2012-09-20 Medichem S.A. NEW CRYSTAL FORMS OF THE SALT OF TRANS-5-CHLORO-2-METHYL-2,3,3A,12b-TETRAHYDRO-1H-DIBENZO[2,3:6,7]OXEPINO[4,5-c]PYRROLE WITH MALEIC ACID
ITMI20110734A1 (it) * 2011-05-02 2012-11-03 Olon Spa Sali cristallini di asenapina
EP2524919A1 (en) 2011-05-17 2012-11-21 Sandoz AG Novel crystalline salts of Asenapine with organic Di-acids and Tri-acids
EP2524920A1 (en) 2011-05-17 2012-11-21 Sandoz AG Novel Crystalline Asenapine Hydrochloride Salt Forms
EP2524921A1 (en) 2011-05-17 2012-11-21 Sandoz AG Novel Crystalline Salts of Asenapine
WO2012156676A1 (en) 2011-05-18 2012-11-22 Laboratorios Lesvi S.L. Monoclinic crystalline form of asenapine maleate with a specific particle size distribution
US9505771B2 (en) * 2011-05-18 2016-11-29 Laboratories Lesvi S.L. Stable micronised monoclin form of asenapine maleate and its synthesis
WO2013041604A1 (en) 2011-09-21 2013-03-28 Sandoz Ag Crystal form of asenapine maleate
EP2572703A1 (en) 2011-09-21 2013-03-27 Hexal AG Compressed oral dosage form for asenapine maleate
CN104507472B (zh) * 2012-07-26 2016-10-05 久光制药株式会社 贴附剂
ITMI20121810A1 (it) 2012-10-24 2014-04-25 Chemo Iberica Sa Poliformi di maleato di asenapina e processo per la loro preparazione
WO2014090386A1 (en) 2012-12-11 2014-06-19 Alfred E. Tiefenbacher (Gmbh & Co. Kg) Orally disintegrating tablet containing asenapine
WO2014127786A1 (en) 2013-02-22 2014-08-28 Zentiva, K.S. Orally disintegrating pharmaceutical composition comprising asenapine
US10786520B2 (en) 2015-09-02 2020-09-29 Eloxx Pharmaceuticals Ltd. Aminoglycoside derivatives and uses thereof in treating genetic disorders
JP7236389B2 (ja) 2016-12-20 2023-03-09 エルテーエス ローマン テラピー-ジステーメ アーゲー アセナピンを含有する経皮治療システム
CN110087641B (zh) 2016-12-20 2024-03-12 罗曼治疗系统股份公司 含有阿塞那平和聚硅氧烷或聚异丁烯的透皮治疗系统
ES2881783T3 (es) 2017-06-26 2021-11-30 Lts Lohmann Therapie Systeme Ag Sistema terapéutico transdérmico que contiene asenapina y polímero de acrílico y silicona
KR20210022656A (ko) 2018-06-20 2021-03-03 에르테에스 로만 테라피-시스테메 아게 아세나핀을 함유하는 경피 치료 시스템

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7605526A (nl) * 1976-05-24 1977-11-28 Akzo Nv Nieuwe tetracyclische derivaten.
HU225051B1 (en) * 1994-03-02 2006-05-29 Organon Ireland Ltd Sublingual or buccal pharmaceutical compositions containing trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1h-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole
WO1999032108A1 (en) * 1997-12-19 1999-07-01 Akzo Nobel N.V. Org-5222 in the treatment of depression
TWI327915B (en) * 2003-06-12 2010-08-01 Organon Nv Pharmaceutical composition comprising antipsychotic agent and use of the antipsychotic agent for treating patients with overweight

Also Published As

Publication number Publication date
DE602006000080D1 (de) 2007-10-04
NO20075142L (no) 2007-11-05
ATE370954T1 (de) 2007-09-15
DE602006004463D1 (de) 2009-02-05
ES2318742T3 (es) 2009-05-01
PT1917267E (pt) 2009-02-04
DOP2006000082A (es) 2006-11-30
HRP20070429T3 (en) 2007-11-30
JP2008534656A (ja) 2008-08-28
UY29459A1 (es) 2006-11-30
EP1917267A1 (en) 2008-05-07
TWI364423B (en) 2012-05-21
DK1917267T3 (da) 2009-04-14
PT1710245E (pt) 2007-10-03
IL186355A0 (en) 2008-01-20
ATE418556T1 (de) 2009-01-15
EP1710245A1 (en) 2006-10-11
SI1710245T1 (sl) 2007-12-31
BRPI0609741A8 (pt) 2018-03-13
NO340520B1 (no) 2017-05-02
EP1917267B1 (en) 2008-12-24
CY1108742T1 (el) 2014-04-09
NZ562124A (en) 2010-07-30
WO2006106135A1 (en) 2006-10-12
JP5058151B2 (ja) 2012-10-24
CY1106902T1 (el) 2012-09-26
CA2603509A1 (en) 2006-10-12
AU2006231617A1 (en) 2006-10-12
RU2007141198A (ru) 2009-05-20
IL186355A (en) 2016-05-31
DK1710245T3 (da) 2007-12-03
KR20080005253A (ko) 2008-01-10
ES2293626T3 (es) 2008-03-16
RU2405786C2 (ru) 2010-12-10
KR101422843B1 (ko) 2014-07-24
DE602006000080T2 (de) 2008-05-15
BRPI0609741A2 (pt) 2010-04-27
AU2006231617B2 (en) 2010-06-03
AR056306A1 (es) 2007-10-03
HN2006014095A (es) 2010-08-19
SI1917267T1 (sl) 2009-04-30
SV2006002473A (es) 2009-11-24
MY137969A (en) 2009-04-30
CA2603509C (en) 2013-12-03
TW200722428A (en) 2007-06-16
RS50532B (sr) 2010-05-07
PL1917267T3 (pl) 2009-06-30
PL1710245T3 (pl) 2008-01-31
PE20061311A1 (es) 2007-02-09
GT200600135A (es) 2006-11-07
EP1710245B1 (en) 2007-08-22

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