MA24342A1 - Nouvelle modification du cristal de cdch, procede pour sa preparation et formules pharmaceutiques comprenant cette modification - Google Patents

Nouvelle modification du cristal de cdch, procede pour sa preparation et formules pharmaceutiques comprenant cette modification

Info

Publication number
MA24342A1
MA24342A1 MA24398A MA24398A MA24342A1 MA 24342 A1 MA24342 A1 MA 24342A1 MA 24398 A MA24398 A MA 24398A MA 24398 A MA24398 A MA 24398A MA 24342 A1 MA24342 A1 MA 24342A1
Authority
MA
Morocco
Prior art keywords
modification
cdch
crystal
preparation
novel
Prior art date
Application number
MA24398A
Other languages
English (en)
French (fr)
Inventor
Grunenberg Alfous
Bosche Apotheker Patrick
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7779831&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA24342(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of MA24342A1 publication Critical patent/MA24342A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA24398A 1995-12-12 1996-11-22 Nouvelle modification du cristal de cdch, procede pour sa preparation et formules pharmaceutiques comprenant cette modification MA24342A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19546249A DE19546249A1 (de) 1995-12-12 1995-12-12 Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen

Publications (1)

Publication Number Publication Date
MA24342A1 true MA24342A1 (fr) 1998-07-01

Family

ID=7779831

Family Applications (1)

Application Number Title Priority Date Filing Date
MA24398A MA24342A1 (fr) 1995-12-12 1996-11-22 Nouvelle modification du cristal de cdch, procede pour sa preparation et formules pharmaceutiques comprenant cette modification

Country Status (42)

Country Link
US (1) US5849752A (en:Method)
EP (1) EP0780390B1 (en:Method)
JP (1) JP4104687B2 (en:Method)
KR (1) KR100525146B1 (en:Method)
CN (1) CN1061348C (en:Method)
AR (1) AR005009A1 (en:Method)
AT (1) ATE221531T1 (en:Method)
AU (1) AU708006B2 (en:Method)
BG (1) BG62258B1 (en:Method)
BR (1) BR9605968A (en:Method)
CA (1) CA2192418C (en:Method)
CO (1) CO4480105A1 (en:Method)
CU (1) CU22774A3 (en:Method)
CZ (1) CZ288657B6 (en:Method)
DE (2) DE19546249A1 (en:Method)
DK (1) DK0780390T3 (en:Method)
EE (1) EE03474B1 (en:Method)
ES (1) ES2179910T3 (en:Method)
HR (1) HRP960558B1 (en:Method)
HU (1) HU226521B1 (en:Method)
ID (1) ID22625A (en:Method)
IL (1) IL119795A (en:Method)
IN (1) IN185805B (en:Method)
MA (1) MA24342A1 (en:Method)
MY (1) MY117492A (en:Method)
NL (1) NL300109I1 (en:Method)
NO (1) NO306725B1 (en:Method)
NZ (1) NZ299905A (en:Method)
PL (1) PL184885B1 (en:Method)
PT (1) PT780390E (en:Method)
RO (1) RO119782B1 (en:Method)
RU (1) RU2162468C2 (en:Method)
SA (1) SA96170492B1 (en:Method)
SG (1) SG47201A1 (en:Method)
SI (1) SI0780390T1 (en:Method)
SK (1) SK282805B6 (en:Method)
SV (1) SV1996000109A (en:Method)
TR (1) TR199600970A2 (en:Method)
TW (1) TW411340B (en:Method)
UA (1) UA35638C2 (en:Method)
YU (1) YU49485B (en:Method)
ZA (1) ZA9610405B (en:Method)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200000752T2 (tr) * 1997-09-25 2000-09-21 Bayer Aktiengesellschaft Etkin terkibin kontrollü salınımı için ilaç formülü.
DE19751948A1 (de) 1997-11-24 1999-05-27 Bayer Ag Verfahren zur Herstellung von 8-Methoxy-Chinoloncarbonsäuren
US6716830B2 (en) 1998-09-30 2004-04-06 Alcon, Inc. Ophthalmic antibiotic compositions containing moxifloxacin
US6395746B1 (en) 1998-09-30 2002-05-28 Alcon Manufacturing, Ltd. Methods of treating ophthalmic, otic and nasal infections and attendant inflammation
US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
US6610327B1 (en) * 1998-11-10 2003-08-26 Bayer Aktiengesellschaft Pharmaceutical moxifloxacin preparation
DE19854357A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854356A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation A von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo-/4.3.0/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854355A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation B von 8-Cyan-1-cyclopropyl-7-(1S, 6S-2,8-diazabicyclo-/4.3.O/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19908449A1 (de) * 1999-02-26 2000-08-31 Bayer Ag Kristallmodifikation C von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicylo-[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chino/incarbonsäure
WO2004039804A1 (en) * 2002-10-31 2004-05-13 Ranbaxy Laboratories Limited Amorphous moxifloxacin hydrochloride
EP1615645B2 (en) 2003-04-09 2013-08-21 Dr. Reddy's Laboratories Ltd. A crystalline form iii of anhydrous moxifloxacin hydrochloride and a process for the preparation thereof
WO2005012285A1 (en) * 2003-08-05 2005-02-10 Matrix Laboratories Ltd An improved process for the preparation of moxifloxacin hydrochloride
ITMI20032259A1 (it) 2003-11-20 2005-05-21 Chemi Spa Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
EP1685130B1 (en) * 2003-11-20 2008-12-10 CHEMI S.p.A. Polymorphs of 1-cyclopropyl-7-([s,s] - 2,8-diazadicyclo [4.3.0] non-8-yl) -6-fluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid hydrochloride and methods for the preparation thereof
US7491725B2 (en) 2004-02-06 2009-02-17 Bristol-Myers Squibb Company Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
DE102004015981A1 (de) * 2004-04-01 2005-10-20 Bayer Healthcare Ag Neue kirstalline Form von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE102004063347A1 (de) * 2004-12-23 2006-07-13 Stada Arzneimittel Ag Gebrauchsfertige Gemcitabinlösungen und Gemcitabinlösungskonzentrate
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
GB0612422D0 (en) * 2006-06-23 2006-08-02 Generics Uk Ltd Novel hydrate form
US20100204470A1 (en) 2006-06-27 2010-08-12 Sandoz Ag method for salt preparation
ES2303768B1 (es) * 2006-09-08 2009-06-05 Quimica Sintetica, S.A. Nueva forma cristalina de moxifloxacino clorhidrato.
KR20150048920A (ko) * 2006-11-13 2015-05-07 씨아이피엘에이 엘티디. 목시플록사신 염산염의 합성방법
EP1992626A1 (en) * 2007-05-10 2008-11-19 Sandoz AG Process for the preparation of moxifloxacin hydrochloride
EP2083010A1 (en) * 2008-01-08 2009-07-29 Chemo Ibérica, S.A. Polymorphic Forms of Moxifloxacin hydrochloride and processes for preparation thereof
EP2154137A1 (en) 2008-08-04 2010-02-17 Chemo Ibérica, S.A. Crystalline form of moxifloxacin base
BRPI0823092A2 (pt) 2008-10-09 2015-09-29 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi método de granulação úmida de moxifloxacin anídrico ou seus sais
EP2342204A1 (en) * 2008-11-06 2011-07-13 Hetero Research Foundation Novel polymorph of moxifloxacin hydrochloride
EA028676B1 (ru) 2008-12-08 2017-12-29 Рациофарм Гмбх Спрессованный моксифлоксацин
NZ596492A (en) 2009-05-15 2013-08-30 Redx Pharma Ltd Redox drug derivatives
WO2011121596A2 (en) * 2010-04-01 2011-10-06 Neuland Laboratories Ltd. Crystal modification of moxifloxacin hydrochloride
BRPI1106900A2 (pt) 2011-12-26 2013-11-05 Ems Sa Composição farmacêutica sólida compreendendo antibótico da familia das quinolonas e processo de sua obtenção
FR2992218B1 (fr) 2012-06-22 2015-01-23 Rivopharm Sa Composition pharmaceutique de chlorhydrate de moxifloxacine et procede de preparation
CN102924449B (zh) * 2012-10-30 2015-08-12 重庆福安药业集团庆余堂制药有限公司 盐酸莫西沙星h晶型及其制备方法和药物组合物
EP2928892B1 (en) 2012-12-04 2018-03-21 Mankind Pharma Ltd. An improved process for the preparation of moxifloxacin hydrochloride
RU2561037C2 (ru) * 2013-02-07 2015-08-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Антибактериальная фармацевтическая композиция и способ ее получения
KR102237887B1 (ko) 2013-03-15 2021-04-07 멜린타 서브시디어리 코프. 항생제를 사용하여 과체중 및 비만 환자에서 감염을 치료하는 방법

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
CN1019114B (zh) * 1986-03-31 1992-11-18 三共株式会社 喹啉-3-羟酸衍生物的制备方法
AU609974B2 (en) * 1988-05-18 1991-05-09 Warner-Lambert Company Improved process for the preparation of 5-amino-7- (substituted amino)-quinoline-3-carboxylic acids
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
RO108347B1 (ro) * 1989-10-30 1994-04-28 Bellon Labor Sa Roger DERIVATI DE BENZO-(b)-NAFTIRIDIN-1,8 SI PROCEDEU DE PREPARARE A ACESTORA
TW209865B (en:Method) 1992-01-10 1993-07-21 Bayer Ag
DE69331003T2 (de) * 1992-01-31 2002-06-20 Chugai Seiyaku K.K., Tokio/Tokyo Kristalle von derivaten von chinozon carbonsäure-hydraten
DE4234078A1 (de) 1992-10-09 1994-04-14 Bayer Ag Chinoloncarbonsäuren
NO301165B1 (no) * 1992-12-25 1997-09-22 Daiichi Seiyaku Co Bicykliske aminderivater og antibakterielle midler inneholdende disse
ZA946853B (en) * 1993-09-10 1995-04-24 Daiichi Seiyaku Co Crystals of antimicrobial compound.
EP0676199B1 (en) * 1994-04-07 1998-09-02 Pfizer Inc. Use of trovafloxacin or derivatives thereof for the manufacture of a medicament for the treatment of H. pylori infections

Also Published As

Publication number Publication date
EP0780390A1 (de) 1997-06-25
BG101043A (en) 1998-04-30
NZ299905A (en) 1998-09-24
NO965298L (no) 1997-06-13
CN1160052A (zh) 1997-09-24
ID22625A (id) 1999-12-02
ATE221531T1 (de) 2002-08-15
EP0780390B1 (de) 2002-07-31
IL119795A (en) 1998-12-27
TR199600970A2 (tr) 1997-06-21
ES2179910T3 (es) 2003-02-01
HRP960558B1 (en) 2002-04-30
CN1061348C (zh) 2001-01-31
AU708006B2 (en) 1999-07-29
RO119782B1 (ro) 2005-03-30
EE03474B1 (et) 2001-08-15
HU226521B1 (en) 2009-03-30
PT780390E (pt) 2002-11-29
IN185805B (en:Method) 2001-05-05
YU65096A (sh) 1998-12-23
JPH09169757A (ja) 1997-06-30
DE59609501D1 (de) 2002-09-05
HU9603428D0 (en) 1997-01-28
SK159196A3 (en) 1997-10-08
MY117492A (en) 2004-07-31
KR970042550A (ko) 1997-07-24
IL119795A0 (en) 1997-03-18
TW411340B (en) 2000-11-11
EE9600201A (et) 1997-06-16
CZ288657B6 (cs) 2001-08-15
SV1996000109A (es) 1997-10-23
RU2162468C2 (ru) 2001-01-27
PL184885B1 (pl) 2003-01-31
SI0780390T1 (en) 2002-10-31
MX9606325A (es) 1997-10-31
UA35638C2 (uk) 2001-04-16
DK0780390T3 (da) 2002-11-11
NO306725B1 (no) 1999-12-13
BR9605968A (pt) 1998-08-18
CA2192418A1 (en) 1997-06-13
ZA9610405B (en) 1997-06-23
NL300109I1 (nl) 2003-02-03
SG47201A1 (en) 1998-03-20
HUP9603428A2 (en) 1997-08-28
BG62258B1 (bg) 1999-06-30
SK282805B6 (sk) 2002-12-03
HUP9603428A3 (en) 1997-10-28
SA96170492B1 (ar) 2006-05-23
AU7421696A (en) 1997-06-19
CU22774A3 (es) 2002-07-24
CO4480105A1 (es) 1997-07-09
PL317415A1 (en) 1997-06-23
US5849752A (en) 1998-12-15
AR005009A1 (es) 1999-04-07
YU49485B (sh) 2006-08-17
CA2192418C (en) 2001-06-12
CZ364696A3 (en) 1997-07-16
KR100525146B1 (ko) 2006-01-27
HRP960558A2 (en) 1998-02-28
NO965298D0 (no) 1996-12-11
DE19546249A1 (de) 1997-06-19
JP4104687B2 (ja) 2008-06-18

Similar Documents

Publication Publication Date Title
MA24342A1 (fr) Nouvelle modification du cristal de cdch, procede pour sa preparation et formules pharmaceutiques comprenant cette modification
MA23942A1 (fr) Formulation nouvelle contenant de la paroxetine, et procede pour sa preparation
EP0888053A4 (en) METHOD FOR TREATING CANCER AND INFECTIOUS DISEASES AND COMPOSITIONS THAT CAN BE USED THEREFOR
FI942076L (fi) Sappihappojohdannaisia, menetelmä niiden valmistamiseksi ja näiden yhdisteiden käyttö lääkaaineina
FI942075A7 (fi) Sappihappojohdannaisten tetratsolijohdannaisia, menetelmä niiden valmistamiseksi ja näiden yhdisteiden käyttö lääkeaineina
FR2742148B1 (fr) Nouveaux derives du pyrazole-3-carboxamide, procede pour leur preparation et compositions pharmaceutiques les contenant
FI942077A7 (fi) Monomeerisiä sappihappojohdannaisia, menetelmä niiden valmistamiseksi ja näiden yhdisteiden käyttö lääkeaineina
RU97118673A (ru) Новые промежуточные продукты и способ получения производных камптотецина (срт-11) и родственных соединений
NO306614B1 (no) Derivater i vitamin D-serien modifisert ved 20-stilling, mellomprodukter anvendt ved fremstilling av disse, farmasöytiske preparater inneholdende derivatene og deres anvendelse ved fremstilling av legemidler
IS1665B (is) Nýjar króman og thíókróman afleiður
NO306400B1 (no) N-substituerte azabicykloheptan-derivater, anvendelse derav og farmasöytisk preparat
FR2627296B1 (fr) Appareil pour indiquer l'heure, du type analogique
FR2534139B1 (fr) Nouvelle forme galenique du sulpiride, son procede de preparation et medicament comprenant cette nouvelle forme
MA26522A1 (fr) Composition pharmaceutique pour le traitement du diabete sucre et d'etats associes.
EE9600109A (et) a-amino- ja tsüklopentaan-ß-aminohapet(-happeid) ja/või nende derivaate sisaldavad segud ja dipeptiidid, dipeptiidide valmistamismeetod ning nimetatud segusid ja/või dipeptiide sisaldavad ravimid
TNSN99124A1 (fr) Compositions pharmaceutiques mixtes pour le traitement de la faiblesse musculosquelettique et procede pour leur preparation.
FR2628421B1 (fr) Procede de preparation des derives de 1,4-dihydropyridine et nouveaux intermediaires utiles pour cette preparation
MA23953A1 (fr) Procede nouveau pour formuler des formes posologiques solides, et formes posologiques ainsi produites
BR9501921A (pt) Composto processo para sua preparação medicamento uso e método para inibir a atividade biológica do leucotrieno
ES2137665T3 (es) Nuevos derivados de piridina o piridazina, procedimientos para su preparacion, y medicamentos que contienen estos compuestos.
ATE170527T1 (de) Phosphonobernsteinsäurederivate und ihre verwendung als arzneimittel
FR2738740B1 (fr) Nouveau procede pour la deformation permanente des matieres keratiniques
NO962809D0 (no) Fremgangsmåte for fremstilling av N-substituerte 4-ketoprolinderivater
FR2661831B1 (fr) Formules pharmaceutiques pour le traitement des maladies vasculaires peripheriques.