ID22625A - Modifikasi kristal baru dari cdch, suatu proses untuk preparatnya dan formulasi farmasi terdiri dari modifikasi - Google Patents

Modifikasi kristal baru dari cdch, suatu proses untuk preparatnya dan formulasi farmasi terdiri dari modifikasi

Info

Publication number
ID22625A
ID22625A IDP963684A ID963684A ID22625A ID 22625 A ID22625 A ID 22625A ID P963684 A IDP963684 A ID P963684A ID 963684 A ID963684 A ID 963684A ID 22625 A ID22625 A ID 22625A
Authority
ID
Indonesia
Prior art keywords
modification
cdch
preparation
formulation containing
new crystals
Prior art date
Application number
IDP963684A
Other languages
English (en)
Inventor
Alfons Dr Grunenberg
Patrick Dr Bosche
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7779831&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ID22625(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of ID22625A publication Critical patent/ID22625A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
IDP963684A 1995-12-12 1996-12-10 Modifikasi kristal baru dari cdch, suatu proses untuk preparatnya dan formulasi farmasi terdiri dari modifikasi ID22625A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19546249A DE19546249A1 (de) 1995-12-12 1995-12-12 Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen

Publications (1)

Publication Number Publication Date
ID22625A true ID22625A (id) 1999-12-02

Family

ID=7779831

Family Applications (1)

Application Number Title Priority Date Filing Date
IDP963684A ID22625A (id) 1995-12-12 1996-12-10 Modifikasi kristal baru dari cdch, suatu proses untuk preparatnya dan formulasi farmasi terdiri dari modifikasi

Country Status (42)

Country Link
US (1) US5849752A (id)
EP (1) EP0780390B1 (id)
JP (1) JP4104687B2 (id)
KR (1) KR100525146B1 (id)
CN (1) CN1061348C (id)
AR (1) AR005009A1 (id)
AT (1) ATE221531T1 (id)
AU (1) AU708006B2 (id)
BG (1) BG62258B1 (id)
BR (1) BR9605968A (id)
CA (1) CA2192418C (id)
CO (1) CO4480105A1 (id)
CU (1) CU22774A3 (id)
CZ (1) CZ288657B6 (id)
DE (2) DE19546249A1 (id)
DK (1) DK0780390T3 (id)
EE (1) EE03474B1 (id)
ES (1) ES2179910T3 (id)
HR (1) HRP960558B1 (id)
HU (1) HU226521B1 (id)
ID (1) ID22625A (id)
IL (1) IL119795A (id)
IN (1) IN185805B (id)
MA (1) MA24342A1 (id)
MY (1) MY117492A (id)
NL (1) NL300109I1 (id)
NO (1) NO306725B1 (id)
NZ (1) NZ299905A (id)
PL (1) PL184885B1 (id)
PT (1) PT780390E (id)
RO (1) RO119782B1 (id)
RU (1) RU2162468C2 (id)
SA (1) SA96170492B1 (id)
SG (1) SG47201A1 (id)
SI (1) SI0780390T1 (id)
SK (1) SK282805B6 (id)
SV (1) SV1996000109A (id)
TR (1) TR199600970A2 (id)
TW (1) TW411340B (id)
UA (1) UA35638C2 (id)
YU (1) YU49485B (id)
ZA (1) ZA9610405B (id)

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JP2001517625A (ja) * 1997-09-25 2001-10-09 バイエル・アクチエンゲゼルシヤフト 活性成分放出制御薬物製剤
DE19751948A1 (de) 1997-11-24 1999-05-27 Bayer Ag Verfahren zur Herstellung von 8-Methoxy-Chinoloncarbonsäuren
US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
US6716830B2 (en) 1998-09-30 2004-04-06 Alcon, Inc. Ophthalmic antibiotic compositions containing moxifloxacin
US6395746B1 (en) 1998-09-30 2002-05-28 Alcon Manufacturing, Ltd. Methods of treating ophthalmic, otic and nasal infections and attendant inflammation
UA72483C2 (en) * 1998-11-10 2005-03-15 Moxifloxacin-containing pharmaceutical preparation and method for its manufacture
DE19854356A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation A von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo-/4.3.0/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854357A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854355A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation B von 8-Cyan-1-cyclopropyl-7-(1S, 6S-2,8-diazabicyclo-/4.3.O/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19908449A1 (de) * 1999-02-26 2000-08-31 Bayer Ag Kristallmodifikation C von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicylo-[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chino/incarbonsäure
WO2004039804A1 (en) * 2002-10-31 2004-05-13 Ranbaxy Laboratories Limited Amorphous moxifloxacin hydrochloride
EP1615645B2 (en) 2003-04-09 2013-08-21 Dr. Reddy's Laboratories Ltd. A crystalline form iii of anhydrous moxifloxacin hydrochloride and a process for the preparation thereof
EP1651630A1 (en) * 2003-08-05 2006-05-03 Matrix Laboratories Ltd An improved process for the preparation of moxifloxacin hydrochloride
WO2005054240A1 (en) * 2003-11-20 2005-06-16 Chemi Spa Polymorphs of 1-cyclopropyl-7-([s,s]-2,8-diazadicyclo[4.3.0]non-8-yl)-6-fluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid hydrochloride and methods for the preparation thereof
ITMI20032259A1 (it) 2003-11-20 2005-05-21 Chemi Spa Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
US7491725B2 (en) 2004-02-06 2009-02-17 Bristol-Myers Squibb Company Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
DE102004063347A1 (de) * 2004-12-23 2006-07-13 Stada Arzneimittel Ag Gebrauchsfertige Gemcitabinlösungen und Gemcitabinlösungskonzentrate
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
GB0612422D0 (en) * 2006-06-23 2006-08-02 Generics Uk Ltd Novel hydrate form
WO2008000418A2 (en) 2006-06-27 2008-01-03 Sandoz Ag New method for salt preparation
ES2303768B1 (es) * 2006-09-08 2009-06-05 Quimica Sintetica, S.A. Nueva forma cristalina de moxifloxacino clorhidrato.
IN2014MN02582A (id) * 2006-11-13 2015-09-11 Cipla Ltd
EP1992626A1 (en) * 2007-05-10 2008-11-19 Sandoz AG Process for the preparation of moxifloxacin hydrochloride
EP2083010A1 (en) * 2008-01-08 2009-07-29 Chemo Ibérica, S.A. Polymorphic Forms of Moxifloxacin hydrochloride and processes for preparation thereof
EP2154137A1 (en) 2008-08-04 2010-02-17 Chemo Ibérica, S.A. Crystalline form of moxifloxacin base
US8314122B2 (en) 2008-10-09 2012-11-20 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi Using of organic solvents in wet granulation of moxifloxacin
WO2010052726A1 (en) * 2008-11-06 2010-05-14 Hetero Research Foundation Novel polymorph of moxifloxacin hydrochloride
US20110293717A1 (en) 2008-12-08 2011-12-01 Ratiopharm Gmbh Compacted moxifloxacin
WO2010131054A1 (en) 2009-05-15 2010-11-18 Bradford Pharma Limited Redox drug derivatives
WO2011121596A2 (en) * 2010-04-01 2011-10-06 Neuland Laboratories Ltd. Crystal modification of moxifloxacin hydrochloride
BRPI1106900A2 (pt) 2011-12-26 2013-11-05 Ems Sa Composição farmacêutica sólida compreendendo antibótico da familia das quinolonas e processo de sua obtenção
FR2992218B1 (fr) 2012-06-22 2015-01-23 Rivopharm Sa Composition pharmaceutique de chlorhydrate de moxifloxacine et procede de preparation
CN102924449B (zh) * 2012-10-30 2015-08-12 重庆福安药业集团庆余堂制药有限公司 盐酸莫西沙星h晶型及其制备方法和药物组合物
EP2928892B1 (en) 2012-12-04 2018-03-21 Mankind Pharma Ltd. An improved process for the preparation of moxifloxacin hydrochloride
RU2561037C2 (ru) * 2013-02-07 2015-08-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Антибактериальная фармацевтическая композиция и способ ее получения

Family Cites Families (10)

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Publication number Priority date Publication date Assignee Title
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
EP0241206A3 (en) * 1986-03-31 1989-05-10 Sankyo Company Limited Quinoline-3-carboxylic acid derivatives, their preparation and use
AU609974B2 (en) * 1988-05-18 1991-05-09 Warner-Lambert Company Improved process for the preparation of 5-amino-7- (substituted amino)-quinoline-3-carboxylic acids
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
TW209865B (id) 1992-01-10 1993-07-21 Bayer Ag
EP0629621B1 (en) * 1992-01-31 2001-10-24 Chugai Seiyaku Kabushiki Kaisha Crystal of quinolonecarboxylic acid derivative hydrate
DE4234078A1 (de) * 1992-10-09 1994-04-14 Bayer Ag Chinoloncarbonsäuren
JP3268098B2 (ja) * 1992-12-25 2002-03-25 第一製薬株式会社 二環性環状アミン誘導体
ZA946853B (en) * 1993-09-10 1995-04-24 Daiichi Seiyaku Co Crystals of antimicrobial compound.
EP0676199B1 (en) * 1994-04-07 1998-09-02 Pfizer Inc. Use of trovafloxacin or derivatives thereof for the manufacture of a medicament for the treatment of H. pylori infections

Also Published As

Publication number Publication date
BG101043A (en) 1998-04-30
DE59609501D1 (de) 2002-09-05
CN1061348C (zh) 2001-01-31
HRP960558A2 (en) 1998-02-28
SA96170492B1 (ar) 2006-05-23
RU2162468C2 (ru) 2001-01-27
TR199600970A2 (tr) 1997-06-21
CN1160052A (zh) 1997-09-24
ES2179910T3 (es) 2003-02-01
NO965298D0 (no) 1996-12-11
DK0780390T3 (da) 2002-11-11
SV1996000109A (es) 1997-10-23
KR100525146B1 (ko) 2006-01-27
US5849752A (en) 1998-12-15
MX9606325A (es) 1997-10-31
YU65096A (sh) 1998-12-23
CA2192418C (en) 2001-06-12
EP0780390A1 (de) 1997-06-25
ZA9610405B (en) 1997-06-23
YU49485B (sh) 2006-08-17
EE9600201A (et) 1997-06-16
AU708006B2 (en) 1999-07-29
CZ364696A3 (en) 1997-07-16
NL300109I1 (nl) 2003-02-03
PL317415A1 (en) 1997-06-23
ATE221531T1 (de) 2002-08-15
NO965298L (no) 1997-06-13
CU22774A3 (es) 2002-07-24
BG62258B1 (bg) 1999-06-30
MA24342A1 (fr) 1998-07-01
BR9605968A (pt) 1998-08-18
AR005009A1 (es) 1999-04-07
MY117492A (en) 2004-07-31
IL119795A (en) 1998-12-27
HUP9603428A3 (en) 1997-10-28
IL119795A0 (en) 1997-03-18
HRP960558B1 (en) 2002-04-30
SI0780390T1 (en) 2002-10-31
SK282805B6 (sk) 2002-12-03
UA35638C2 (uk) 2001-04-16
NO306725B1 (no) 1999-12-13
PT780390E (pt) 2002-11-29
DE19546249A1 (de) 1997-06-19
NZ299905A (en) 1998-09-24
CZ288657B6 (cs) 2001-08-15
AU7421696A (en) 1997-06-19
EE03474B1 (et) 2001-08-15
JP4104687B2 (ja) 2008-06-18
JPH09169757A (ja) 1997-06-30
PL184885B1 (pl) 2003-01-31
SK159196A3 (en) 1997-10-08
KR970042550A (ko) 1997-07-24
HUP9603428A2 (en) 1997-08-28
TW411340B (en) 2000-11-11
SG47201A1 (en) 1998-03-20
EP0780390B1 (de) 2002-07-31
HU226521B1 (en) 2009-03-30
IN185805B (id) 2001-05-05
HU9603428D0 (en) 1997-01-28
CO4480105A1 (es) 1997-07-09
RO119782B1 (ro) 2005-03-30
CA2192418A1 (en) 1997-06-13

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