LV12687B - Aterosklerozes arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas - Google Patents

Aterosklerozes arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas

Info

Publication number
LV12687B
LV12687B LV010058A LV010058A LV12687B LV 12687 B LV12687 B LV 12687B LV 010058 A LV010058 A LV 010058A LV 010058 A LV010058 A LV 010058A LV 12687 B LV12687 B LV 12687B
Authority
LV
Latvia
Prior art keywords
saturation
inhibitors
combinations
content
arteriosclerosis treatment
Prior art date
Application number
LV010058A
Other languages
English (en)
Latvian (lv)
Other versions
LV12687A (en
Inventor
Jeffrey Robl
Rex A Parker
Scott A Biller
Haris Jamil
Bruce L Jacobson
Krishna Kodukula
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22280975&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LV12687(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of LV12687A publication Critical patent/LV12687A/en
Publication of LV12687B publication Critical patent/LV12687B/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Electrical Discharge Machining, Electrochemical Machining, And Combined Machining (AREA)
LV010058A 1998-09-17 2001-04-12 Aterosklerozes arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas LV12687B (lv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10067798P 1998-09-17 1998-09-17
PCT/US1999/021069 WO2000015230A1 (en) 1998-09-17 1999-09-13 METHOD FOR TREATING ATHEROSCLEROSIS EMPLOYING AN aP2 INHIBITOR AND COMBINATION

Publications (2)

Publication Number Publication Date
LV12687A LV12687A (en) 2001-07-20
LV12687B true LV12687B (lv) 2001-10-20

Family

ID=22280975

Family Applications (2)

Application Number Title Priority Date Filing Date
LV010058A LV12687B (lv) 1998-09-17 2001-04-12 Aterosklerozes arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas
LV010057A LV12686B (lv) 1998-09-17 2001-04-12 Diabeta arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas

Family Applications After (1)

Application Number Title Priority Date Filing Date
LV010057A LV12686B (lv) 1998-09-17 2001-04-12 Diabeta arstesanas panemiens izmantojot ap2 inhibitoru un to saturosas kombinacijas

Country Status (30)

Country Link
US (1) US20020035064A1 (es)
EP (2) EP1113801A4 (es)
JP (2) JP2002524518A (es)
KR (2) KR20010075150A (es)
CN (2) CN1319012A (es)
AT (1) ATE406898T1 (es)
AU (2) AU754488B2 (es)
BG (2) BG105432A (es)
BR (2) BR9913833A (es)
CA (2) CA2344309A1 (es)
CO (2) CO5130025A1 (es)
CZ (2) CZ2001965A3 (es)
DE (1) DE69939481D1 (es)
EE (2) EE200100155A (es)
ES (1) ES2311306T3 (es)
GE (2) GEP20033045B (es)
HU (2) HUP0104240A2 (es)
ID (2) ID28450A (es)
IL (2) IL141785A0 (es)
LT (2) LT4870B (es)
LV (2) LV12687B (es)
NO (2) NO20011351L (es)
NZ (2) NZ510209A (es)
PE (2) PE20001047A1 (es)
PL (2) PL346660A1 (es)
SK (1) SK3202001A3 (es)
TR (2) TR200100774T2 (es)
UY (2) UY25714A1 (es)
WO (2) WO2000015229A1 (es)
ZA (2) ZA200207433B (es)

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JP6514282B2 (ja) * 2014-03-24 2019-05-15 花王株式会社 Ｇｉｐ上昇抑制剤の評価又は選択方法
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Also Published As

Publication number Publication date
BR9913831A (pt) 2001-05-29
HUP0104240A2 (hu) 2002-03-28
EE200100154A (et) 2002-12-16
CO5130025A1 (es) 2002-02-27
LT4870B (lt) 2001-12-27
BG105432A (en) 2001-12-29
GEP20033045B (en) 2003-08-25
NO20011352D0 (no) 2001-03-16
US20020035064A1 (en) 2002-03-21
LV12687A (en) 2001-07-20
AU754488B2 (en) 2002-11-14
SK3202001A3 (en) 2002-04-04
NZ510209A (en) 2003-07-25
LT2001023A (en) 2001-08-27
BG105431A (en) 2001-12-29
LV12686A (en) 2001-07-20
TR200100773T2 (tr) 2001-07-23
EE04356B1 (et) 2004-10-15
JP2002524517A (ja) 2002-08-06
NZ510207A (en) 2003-08-29
PE20001056A1 (es) 2000-12-24
BR9913833A (pt) 2001-05-29
WO2000015229A1 (en) 2000-03-23
CO5130026A1 (es) 2002-02-27
EP1121129A1 (en) 2001-08-08
EE200100155A (et) 2002-08-15
AU755563B2 (en) 2002-12-12
ZA200207433B (en) 2003-10-27
PE20001047A1 (es) 2000-12-24
ID27833A (id) 2001-04-26
CN1317970A (zh) 2001-10-17
CA2344300A1 (en) 2000-03-23
ES2311306T3 (es) 2009-02-01
CZ2001964A3 (cs) 2002-01-16
EP1113801A1 (en) 2001-07-11
EP1113801A4 (en) 2002-10-02
HUP0104108A2 (hu) 2002-03-28
CN1319012A (zh) 2001-10-24
UY25714A1 (es) 2001-08-27
UY25713A1 (es) 2001-08-27
LT2001022A (en) 2001-08-27
LT4871B (lt) 2001-12-27
LV12686B (lv) 2001-10-20
NO20011351D0 (no) 2001-03-16
AU6387799A (en) 2000-04-03
EP1121129B1 (en) 2008-09-03
PL346660A1 (en) 2002-02-25
IL141786A0 (en) 2002-03-10
ZA200207430B (en) 2003-09-16
CA2344309A1 (en) 2000-03-23
AU6143799A (en) 2000-04-03
ID28450A (id) 2001-05-24
GEP20033044B (en) 2003-08-25
IL141785A0 (en) 2002-03-10
KR20010079842A (ko) 2001-08-22
JP2002524518A (ja) 2002-08-06
TR200100774T2 (tr) 2001-12-21
EP1121129A4 (en) 2002-10-16
DE69939481D1 (de) 2008-10-16
WO2000015230A1 (en) 2000-03-23
KR20010075150A (ko) 2001-08-09
NO20011352L (no) 2001-05-11
CZ2001965A3 (cs) 2002-02-13
PL346661A1 (en) 2002-02-25
ATE406898T1 (de) 2008-09-15
NO20011351L (no) 2001-05-11

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