KR101567096B1 - 항균제로서의 트리시클릭 질소 함유 화합물 - Google Patents

항균제로서의 트리시클릭 질소 함유 화합물 Download PDF

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Publication number
KR101567096B1
KR101567096B1 KR1020097024090A KR20097024090A KR101567096B1 KR 101567096 B1 KR101567096 B1 KR 101567096B1 KR 1020097024090 A KR1020097024090 A KR 1020097024090A KR 20097024090 A KR20097024090 A KR 20097024090A KR 101567096 B1 KR101567096 B1 KR 101567096B1
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South Korea
Prior art keywords
dihydro
methyl
piperidinyl
amino
dione
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KR1020097024090A
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Korean (ko)
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KR20100017133A (ko
Inventor
데이비드 에반 데이비스
데이비드 토마스 데이비스
일라리아 지오다노
알란 죠셉 헤네시
네일 데이비드 피어슨
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글락소 그룹 리미티드
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39580226&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR101567096(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0707705A external-priority patent/GB0707705D0/en
Priority claimed from GB0720569A external-priority patent/GB0720569D0/en
Priority claimed from GB0805311A external-priority patent/GB0805311D0/en
Application filed by 글락소 그룹 리미티드 filed Critical 글락소 그룹 리미티드
Publication of KR20100017133A publication Critical patent/KR20100017133A/ko
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
KR1020097024090A 2007-04-20 2008-04-16 항균제로서의 트리시클릭 질소 함유 화합물 Active KR101567096B1 (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
GB0707705.0 2007-04-20
GB0707705A GB0707705D0 (en) 2007-04-20 2007-04-20 Compounds
GB0720569.3 2007-10-19
GB0720569A GB0720569D0 (en) 2007-10-19 2007-10-19 Compounds
GB0805311A GB0805311D0 (en) 2008-03-20 2008-03-20 Compounds
GB0805311.8 2008-03-20

Publications (2)

Publication Number Publication Date
KR20100017133A KR20100017133A (ko) 2010-02-16
KR101567096B1 true KR101567096B1 (ko) 2015-11-06

Family

ID=39580226

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020097024090A Active KR101567096B1 (ko) 2007-04-20 2008-04-16 항균제로서의 트리시클릭 질소 함유 화합물

Country Status (31)

Country Link
US (1) US8389524B2 (https=)
EP (1) EP2137196B1 (https=)
JP (1) JP5389013B2 (https=)
KR (1) KR101567096B1 (https=)
CN (1) CN101687887B (https=)
AR (1) AR066111A1 (https=)
AT (1) ATE483717T1 (https=)
AU (1) AU2008240764C1 (https=)
BR (1) BRPI0810064B8 (https=)
CA (1) CA2684659C (https=)
CL (1) CL2008001122A1 (https=)
CO (1) CO6251368A2 (https=)
CR (2) CR11123A (https=)
CY (1) CY1111248T1 (https=)
DE (1) DE602008002912D1 (https=)
DK (1) DK2137196T3 (https=)
DO (1) DOP2009000240A (https=)
EA (1) EA015821B1 (https=)
HR (1) HRP20100574T1 (https=)
IL (1) IL201204A0 (https=)
MA (1) MA31324B1 (https=)
MX (1) MX2009011317A (https=)
MY (1) MY149347A (https=)
NZ (1) NZ579877A (https=)
PE (1) PE20090274A1 (https=)
PL (1) PL2137196T3 (https=)
PT (1) PT2137196E (https=)
SI (1) SI2137196T1 (https=)
TW (1) TWI431006B (https=)
UY (1) UY31038A1 (https=)
WO (1) WO2008128942A1 (https=)

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CN103113291B (zh) * 2013-02-04 2015-03-04 浙江大学 一种3位烯基吡啶衍生物的合成方法
JP6453216B2 (ja) * 2013-07-23 2019-01-16 エーザイ・アール・アンド・ディー・マネジメント株式会社 ヘテロ縮合環化合物
JP6546654B2 (ja) 2014-08-22 2019-07-17 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ 淋菌感染を治療するための三環式含窒素化合物
MX385384B (es) * 2016-06-22 2025-03-18 Univ Vanderbilt Moduladores alostericos positivos del receptor muscarinico de acetilcolina m4
WO2018195098A1 (en) 2017-04-17 2018-10-25 Ohio State Innovation Foundation Type ii topoisomerase inhibitors and methods of making and using thereof
WO2020201833A1 (en) 2019-04-03 2020-10-08 Glaxomithkline Intellectual Property Development Limited Gepotidacin for use in the treatment of bacterial urinary tract infections
CN114173789A (zh) * 2019-07-05 2022-03-11 葛兰素史克知识产权发展有限公司 用于治疗由生殖支原体引起的感染的组合
ES3004932T3 (en) 2020-04-02 2025-03-13 Glaxosmithkline Ip Dev Ltd Regimen for treating a neisseria gonorrhoeae infection with gepotidacin
EP4143188A1 (en) * 2020-04-29 2023-03-08 GlaxoSmithKline Intellectual Property Development Limited Crystalline forms of gepotidacin
CN111494241B (zh) * 2020-06-01 2023-03-24 湖北洁世达环保科技有限公司 一种纸巾柔润保湿液
CA3210313A1 (en) * 2021-02-05 2022-08-11 Glaxosmithkline Intellectual Property Development Limited Oral solid dose formulations
US20250099535A1 (en) 2022-01-21 2025-03-27 Glaxosmithkline Intellectual Property Development Limited Gepotidacin and vancomycin for use in the treatment of an infection caused by staphylococcus saprophyticus
EP4316463A1 (en) 2022-08-02 2024-02-07 GlaxoSmithKline Intellectual Property Development Limited Novel formulation
CN119546302A (zh) 2022-09-26 2025-02-28 葛兰素史密斯克莱知识产权发展有限公司 用于治疗细菌性前列腺炎的吉泊达星
CN121537412B (zh) * 2026-01-16 2026-04-03 南京道尔医药研究院有限公司 一种吉泊达星甲磺酸盐的制备方法

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CR20150586A (es) 2016-04-04
ATE483717T1 (de) 2010-10-15
NZ579877A (en) 2011-09-30
EP2137196B1 (en) 2010-10-06
HRP20100574T1 (hr) 2010-12-31
CR11123A (es) 2010-03-08
TW200848420A (en) 2008-12-16
CA2684659A1 (en) 2008-10-30
EA200970987A1 (ru) 2010-04-30
US20100137282A1 (en) 2010-06-03
JP2010524884A (ja) 2010-07-22
IL201204A0 (en) 2010-05-17
CO6251368A2 (es) 2011-02-21
PL2137196T3 (pl) 2011-03-31
TWI431006B (zh) 2014-03-21
EP2137196A1 (en) 2009-12-30
DOP2009000240A (es) 2009-12-31
AR066111A1 (es) 2009-07-22
MX2009011317A (es) 2009-11-05
PT2137196E (pt) 2010-12-16
WO2008128942A1 (en) 2008-10-30
SI2137196T1 (sl) 2011-01-31
CY1111248T1 (el) 2015-06-11
AU2008240764A1 (en) 2008-10-30
DE602008002912D1 (de) 2010-11-18
JP5389013B2 (ja) 2014-01-15
CL2008001122A1 (es) 2008-10-24
MA31324B1 (fr) 2010-04-01
UY31038A1 (es) 2008-11-28
CN101687887B (zh) 2012-08-29
BRPI0810064B1 (pt) 2021-03-30
AU2008240764B2 (en) 2011-04-07
AU2008240764C1 (en) 2011-10-20
DK2137196T3 (da) 2011-01-10
PE20090274A1 (es) 2009-04-03
BRPI0810064A2 (pt) 2019-08-27
HK1138000A1 (en) 2010-08-13
MY149347A (en) 2013-08-30
BRPI0810064B8 (pt) 2021-05-25
KR20100017133A (ko) 2010-02-16
CA2684659C (en) 2015-11-24
US8389524B2 (en) 2013-03-05
EA015821B1 (ru) 2011-12-30
CN101687887A (zh) 2010-03-31

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