ATE441645T1 - Neue antibiotische derivate - Google Patents
Neue antibiotische derivateInfo
- Publication number
- ATE441645T1 ATE441645T1 AT06745019T AT06745019T ATE441645T1 AT E441645 T1 ATE441645 T1 AT E441645T1 AT 06745019 T AT06745019 T AT 06745019T AT 06745019 T AT06745019 T AT 06745019T AT E441645 T1 ATE441645 T1 AT E441645T1
- Authority
- AT
- Austria
- Prior art keywords
- alkyl
- antibiotic derivatives
- new antibiotic
- ncoch2
- nch2co
- Prior art date
Links
- 230000003115 biocidal effect Effects 0.000 title abstract 2
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 5
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 229910052731 fluorine Inorganic materials 0.000 abstract 1
- 239000011737 fluorine Substances 0.000 abstract 1
- 125000001072 heteroaryl group Chemical group 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Saccharide Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP2005005643 | 2005-05-25 | ||
| PCT/IB2006/051661 WO2006126171A2 (en) | 2005-05-25 | 2006-05-24 | New antibiotic derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE441645T1 true ATE441645T1 (de) | 2009-09-15 |
Family
ID=37075940
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT06745019T ATE441645T1 (de) | 2005-05-25 | 2006-05-24 | Neue antibiotische derivate |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7981886B2 (de) |
| EP (1) | EP1888574B1 (de) |
| JP (1) | JP2008542258A (de) |
| CN (1) | CN101180298B (de) |
| AT (1) | ATE441645T1 (de) |
| CA (1) | CA2608687A1 (de) |
| DE (1) | DE602006008932D1 (de) |
| ES (1) | ES2330670T3 (de) |
| WO (1) | WO2006126171A2 (de) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7165836B2 (en) | 2003-10-14 | 2007-01-23 | Hewlett-Packard Development Company, L.P. | Method of thermally sealing the overcoat of multilayer media |
| JP2008542258A (ja) | 2005-05-25 | 2008-11-27 | アクテリオン ファーマシューティカルズ リミテッド | 新規抗生物質誘導体 |
| ATE481406T1 (de) | 2006-04-06 | 2010-10-15 | Glaxo Group Ltd | Pyrrolochinoxalinonderivate als antibakterielle mittel |
| JP5389013B2 (ja) * | 2007-04-20 | 2014-01-15 | グラクソ グループ リミテッド | 抗菌剤としての三環式含窒素化合物 |
| JP5281647B2 (ja) * | 2008-09-08 | 2013-09-04 | 日本曹達株式会社 | 含窒素ヘテロ環化合物およびその塩並びに農園芸用殺菌剤 |
| EP2352734A1 (de) | 2008-10-17 | 2011-08-10 | Glaxo Group Limited | Als antibakterielle mittel verwendete tricyclische stickstoffverbindungen |
| AR076222A1 (es) * | 2009-04-09 | 2011-05-26 | Actelion Pharmaceuticals Ltd | Derivados 2-hidroxietil-1h-quinolin-ona y sus analogos azaisotericos con actividad antibacteriana y composiciones farmaceuticas que los contienen |
| FR2956941A1 (fr) | 2010-02-19 | 2011-09-02 | Ingenico Sa | Procede d'authentification biometrique, systeme d'authentification, programme et terminal correspondants. |
| AU2011218830B2 (en) | 2010-02-25 | 2014-07-24 | Merck Sharp & Dohme Corp. | Novel cyclic benzimidazole derivatives useful anti-diabetic agents |
| JP6546936B2 (ja) | 2014-05-28 | 2019-07-17 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | チアゾール誘導体を調製する方法 |
| EP3639824A1 (de) | 2014-08-22 | 2020-04-22 | GlaxoSmithKline Intellectual Property Development Limited | Tricyclische stickstoffhaltige verbindungen zur behandlung einer infektion mit neisseria gonorrhoea |
| CN114105971B (zh) * | 2021-09-30 | 2024-04-09 | 南京林业大学 | 6-(苯并1,3二氧五环基)-4苯基-6h-1,3-噻嗪-2-胺衍生物和应用 |
| EP4580618A2 (de) * | 2022-08-30 | 2025-07-09 | Pannex Therapeutics Inc. | Pannexin-1-modulatoren und verfahren zur behandlung von erkrankungen mit zusammenhang mit pannexin-1 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1992006086A1 (en) * | 1990-10-01 | 1992-04-16 | Janssen Pharmaceutica N.V. | Novel 4-piperidinylcarbonyl derivatives |
| DE19708846A1 (de) * | 1997-03-05 | 1998-09-17 | Gruenenthal Gmbh | Neue Benzoxazindionderivate, Verfahren zu ihrer Herstellung und ihre Verwendung |
| CA2581057A1 (en) * | 2004-10-05 | 2006-04-13 | Actelion Pharmaceuticals Ltd | New piperidine antibiotics |
| JP5314244B2 (ja) * | 2004-10-27 | 2013-10-16 | 富山化学工業株式会社 | 新規な含窒素複素環化合物およびその塩 |
| JP2008542258A (ja) | 2005-05-25 | 2008-11-27 | アクテリオン ファーマシューティカルズ リミテッド | 新規抗生物質誘導体 |
-
2006
- 2006-05-24 JP JP2008513003A patent/JP2008542258A/ja active Pending
- 2006-05-24 CN CN2006800180578A patent/CN101180298B/zh not_active Expired - Fee Related
- 2006-05-24 AT AT06745019T patent/ATE441645T1/de not_active IP Right Cessation
- 2006-05-24 US US11/915,179 patent/US7981886B2/en not_active Expired - Fee Related
- 2006-05-24 DE DE602006008932T patent/DE602006008932D1/de active Active
- 2006-05-24 CA CA002608687A patent/CA2608687A1/en not_active Abandoned
- 2006-05-24 WO PCT/IB2006/051661 patent/WO2006126171A2/en not_active Ceased
- 2006-05-24 EP EP06745019A patent/EP1888574B1/de not_active Not-in-force
- 2006-05-24 ES ES06745019T patent/ES2330670T3/es active Active
Also Published As
| Publication number | Publication date |
|---|---|
| CN101180298B (zh) | 2011-04-27 |
| US20080280888A1 (en) | 2008-11-13 |
| EP1888574B1 (de) | 2009-09-02 |
| US7981886B2 (en) | 2011-07-19 |
| CA2608687A1 (en) | 2006-11-30 |
| WO2006126171A2 (en) | 2006-11-30 |
| DE602006008932D1 (de) | 2009-10-15 |
| WO2006126171A3 (en) | 2007-02-08 |
| ES2330670T3 (es) | 2009-12-14 |
| JP2008542258A (ja) | 2008-11-27 |
| EP1888574A2 (de) | 2008-02-20 |
| CN101180298A (zh) | 2008-05-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |