KR101162046B1 - ＩκＢ 키나제 조절용 인돌 또는 벤즈이미다졸 유도체 - Google Patents

ＩκＢ 키나제 조절용 인돌 또는 벤즈이미다졸 유도체 Download PDF

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KR101162046B1
KR101162046B1 KR1020057002707A KR20057002707A KR101162046B1 KR 101162046 B1 KR101162046 B1 KR 101162046B1 KR 1020057002707 A KR1020057002707 A KR 1020057002707A KR 20057002707 A KR20057002707 A KR 20057002707A KR 101162046 B1 KR101162046 B1 KR 101162046B1
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indole
ethyl
formula
compound
ylamino
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KR20050058338A (ko
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올라프 리트젤러
게르하르트 예네
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사노피-아벤티스 도이칠란트 게엠베하
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
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    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Health & Medical Sciences (AREA)
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  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
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  • Communicable Diseases (AREA)
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  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Molecular Biology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • AIDS & HIV (AREA)
KR1020057002707A 2002-08-17 2003-08-05 ＩκＢ 키나제 조절용 인돌 또는 벤즈이미다졸 유도체 Expired - Fee Related KR101162046B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10237722A DE10237722A1 (de) 2002-08-17 2002-08-17 Indol- oder Benzimidazolderivate zur Modulation der IKappaB-Kinase
DE10237722.7 2002-08-17
PCT/EP2003/008629 WO2004022553A1 (de) 2002-08-17 2003-08-05 INDOL-ODER BENZIMIDAZOLDERIVATE ZUR MODULATION DER IλB-KINASE

Publications (2)

Publication Number Publication Date
KR20050058338A KR20050058338A (ko) 2005-06-16
KR101162046B1 true KR101162046B1 (ko) 2012-07-04

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KR1020057002707A Expired - Fee Related KR101162046B1 (ko) 2002-08-17 2003-08-05 ＩκＢ 키나제 조절용 인돌 또는 벤즈이미다졸 유도체

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US (2) US7285560B2 (enExample)
EP (2) EP1530568B1 (enExample)
JP (1) JP4504812B2 (enExample)
KR (1) KR101162046B1 (enExample)
CN (1) CN1314683C (enExample)
AR (1) AR040975A1 (enExample)
AT (2) ATE493402T1 (enExample)
AU (1) AU2003263196B2 (enExample)
BR (1) BR0313562A (enExample)
CA (1) CA2498559C (enExample)
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DE (2) DE10237722A1 (enExample)
DK (2) DK2233483T3 (enExample)
EC (1) ECSP055612A (enExample)
ES (2) ES2387954T3 (enExample)
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