DE10237722A1 - Indol- oder Benzimidazolderivate zur Modulation der IKappaB-Kinase - Google Patents
Indol- oder Benzimidazolderivate zur Modulation der IKappaB-Kinase Download PDFInfo
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- DE10237722A1 DE10237722A1 DE10237722A DE10237722A DE10237722A1 DE 10237722 A1 DE10237722 A1 DE 10237722A1 DE 10237722 A DE10237722 A DE 10237722A DE 10237722 A DE10237722 A DE 10237722A DE 10237722 A1 DE10237722 A1 DE 10237722A1
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- 102000001284 I-kappa-B kinase Human genes 0.000 title claims abstract description 16
- 108060006678 I-kappa-B kinase Proteins 0.000 title claims abstract description 16
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- 229940054051 antipsychotic indole derivative Drugs 0.000 title description 8
- 229940058303 antinematodal benzimidazole derivative Drugs 0.000 title description 5
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
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Landscapes
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- General Chemical & Material Sciences (AREA)
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- Endocrinology (AREA)
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Priority Applications (52)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10237722A DE10237722A1 (de) | 2002-08-17 | 2002-08-17 | Indol- oder Benzimidazolderivate zur Modulation der IKappaB-Kinase |
| UAA200502387A UA78591C2 (en) | 2002-08-17 | 2003-05-08 | INDOLE OR BENZIMIDAZOLE DERIVATIVE AS SUBSTANCES MODULATING IkB KINASE |
| JO200387A JO2764B1 (en) | 2002-08-17 | 2003-07-23 | Indole derivatives or benzimidazole derivatives to modify the enzyme AKP kinase |
| EP03793685A EP1530568B1 (de) | 2002-08-17 | 2003-08-05 | INDOL-ODER BENZIMIDAZOLDERIVATE ZUR MODULATION DER IkB-KINASE |
| PE2003000772A PE20040893A1 (es) | 2002-08-17 | 2003-08-05 | DERIVADOS DE INDOL O DERIVADOS DE BENCIMIDAZOL PARA MODULAR IkB QUINASA |
| DK03793685.3T DK1530568T3 (da) | 2002-08-17 | 2003-08-05 | Indol- eller benzimidazolderivater til modulering af ikb-kinasen |
| PL03374229A PL374229A1 (en) | 2002-08-17 | 2003-08-05 | Indole or benzimidazole derivatives for modulating ik b kinase |
| AU2003263196A AU2003263196B2 (en) | 2002-08-17 | 2003-08-05 | Indole or benzimidazole derivatives for modulating IkappaB kinase |
| SI200332173T SI2233483T1 (sl) | 2002-08-17 | 2003-08-05 | Indolni ali benzimidazolni derivati za modulacijo IkapaB-kinaze in intermediati za njihovo pripravo |
| PT03793685T PT1530568E (pt) | 2002-08-17 | 2003-08-05 | DERIVADOS DE INDOLE OU DE BENZIMIDAZOLE PARA A MODULAÇÃO DA IkappaB CINASE |
| OA1200500047A OA12908A (en) | 2002-08-17 | 2003-08-05 | Indole or benzimidazole derivatives for modulatingIKB-kinase. |
| EP10163200A EP2233483B1 (de) | 2002-08-17 | 2003-08-05 | Indol- oder Benzimidazolderivate zur Modulation der IkB-Kinase und Zwischenprodukte zu deren Herstellung |
| ES03793685T ES2358795T3 (es) | 2002-08-17 | 2003-08-05 | Derivados de indol o derivados de bencimidazol para modular la ikb quinasa. |
| DE50313372T DE50313372D1 (de) | 2002-08-17 | 2003-08-05 | INDOL-ODER BENZIMIDAZOLDERIVATE ZUR MODULATION DER IkB-KINASE |
| CNB038195437A CN1314683C (zh) | 2002-08-17 | 2003-08-05 | 用于调节IkB激酶的吲哚或苯并咪唑衍生物 |
| SI200331971T SI1530568T1 (sl) | 2002-08-17 | 2003-08-05 | Indolni ali benzimidazolni derivati za modulacijo IkapaB-kinaze |
| BRPI0313562-4A BR0313562A (pt) | 2002-08-17 | 2003-08-05 | derivados de indol ou benzimidazol para a modulação da ikb-cinase |
| YU20050104A RS51902B (sr) | 2002-08-17 | 2003-08-05 | Derivati indola ili benzimidazola za modulaciju ikb-kinaze |
| JP2004533319A JP4504812B2 (ja) | 2002-08-17 | 2003-08-05 | ＩκＢキナーゼをモジュレートするためのインドール誘導体またはベンズイミダゾール誘導体 |
| DK10163200.8T DK2233483T3 (da) | 2002-08-17 | 2003-08-05 | Indol- eller benzimidazol-derivater til modulering af IKB-kinase og mellemprodukter til fremstilling deraf |
| NZ538296A NZ538296A (en) | 2002-08-17 | 2003-08-05 | Indole derivatives or benzimidazole derivatives for modulating IkB kinase |
| ES10163200T ES2387954T3 (es) | 2002-08-17 | 2003-08-05 | Derivados de indol o de bencimidazol para modular la IkB quinasa, y productos intermedios para su preparación |
| HRP20050042AA HRP20050042B1 (hr) | 2002-08-17 | 2003-08-05 | DERIVATI INDOLA ILI BENZIMIDAZOLA ZA MODULACIJU IkB KINAZE |
| MEP-606/08A MEP60608A (en) | 2002-08-17 | 2003-08-05 | INDOLE OR BENZIMIDAZOLE DERIVATIVES FOR MODULATING IkappaB KINASE |
| KR1020057002707A KR101162046B1 (ko) | 2002-08-17 | 2003-08-05 | ＩκＢ 키나제 조절용 인돌 또는 벤즈이미다졸 유도체 |
| HK05111392.6A HK1079509B (en) | 2002-08-17 | 2003-08-05 | INDOLE OR BENZIMIDAZOLE DERIVATIVES FOR MODULATING IκB KINASE |
| PT10163200T PT2233483E (pt) | 2002-08-17 | 2003-08-05 | Derivados de indole ou de benzimidazole para a modulação da iκb cinase e produtos intermédios para a sua preparação |
| RU2005107418/04A RU2318820C2 (ru) | 2002-08-17 | 2003-08-05 | ПРОИЗВОДНЫЕ ИНДОЛА ИЛИ БЕНЗИМИДАЗОЛА ДЛЯ МОДУЛЯЦИИ IkB-КИНАЗЫ |
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| AT03793685T ATE493402T1 (de) | 2002-08-17 | 2003-08-05 | Indol-oder benzimidazolderivate zur modulation der ikb-kinase |
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| AT10163200T ATE557018T1 (de) | 2002-08-17 | 2003-08-05 | Indol- oder benzimidazolderivate zur modulation der ikb-kinase und zwischenprodukte zu deren herstellung |
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| TW092122309A TWI290552B (en) | 2002-08-17 | 2003-08-14 | Indole derivatives or benzimidazole derivatives for modulating IkB kinase |
| UY27941A UY27941A1 (es) | 2002-08-17 | 2003-08-15 | Derivados de indol o derivados de bencimidazol para modular ikb quinasa |
| SV2003001599A SV2004001599A (es) | 2002-08-17 | 2003-08-15 | Derivados de indol o de bencimidazol para modula ikb quinasa |
| MYPI20033115A MY140074A (en) | 2002-08-17 | 2003-08-15 | INDOLE DERIVATIVES OR BENZIMIDAZOLE DERIVATIVES FOR MODULATING IkB KINASE |
| HN2003000249A HN2003000249A (es) | 2002-08-17 | 2003-08-15 | Derivados de indol o derivados de bencimidazol para modular ikb quinasa |
| US10/642,970 US7285560B2 (en) | 2002-08-17 | 2003-08-18 | Indole derivatives or benzimidazole derivatives for modulating IκB kinase |
| ZA200500322A ZA200500322B (en) | 2002-08-17 | 2005-01-13 | INdole of benzimidazole derivatives for modulating kB kinase |
| CR7668A CR7668A (es) | 2002-08-17 | 2005-01-28 | Derivados del indole o benzimidazole para modular ikappab kinasa |
| IL16678505A IL166785A0 (en) | 2002-08-17 | 2005-02-09 | Indole derivatives or benzimidazole derivatives for modulating ikappab kinase |
| MA28106A MA27382A1 (fr) | 2002-08-17 | 2005-02-15 | DERIVES D'INDOLE OU DE BENZIMIDAZOLE POUR MODULER L'IkB KINASE |
| CO05013335A CO5690586A2 (es) | 2002-08-17 | 2005-02-15 | Derivados de indol o derivados de bencimidazol para modular ixb quinasa |
| TNP2005000045A TNSN05045A1 (en) | 2002-08-17 | 2005-02-16 | Indole or benzimidazole derivatives for modulating ikappab kinase |
| EC2005005612A ECSP055612A (es) | 2002-08-17 | 2005-02-17 | Derivados de indol o derivados de bencimidazol para modular IkB quinasa |
| NO20051337A NO330981B1 (no) | 2002-08-17 | 2005-03-15 | Indol- eller benzimidazolderivater for modulering av IkB-kinase, fremgangsmate for fremstilling av disse, legemiddel og anvendelse av forbindelsene |
| US11/758,978 US8778955B2 (en) | 2002-08-17 | 2007-06-06 | Indole derivatives or benzimidazole derivatives for modulating IkB kinase |
| CY20111100246T CY1111692T1 (el) | 2002-08-17 | 2011-03-02 | ΠΑΡΑΓΩΓΑ ΙΝΔΟΛΗΣ Ή ΒΕΝΖΙΜΙΔΑΖΟΛΗΣ ΓΙΑ ΤΗ ΡΥΘΜΙΣΗ ΤΗΣ ΙκΒ ΚΙΝΑΣΗΣ |
| CY20121100658T CY1112991T1 (el) | 2002-08-17 | 2012-07-24 | ΠΑΡΑΓΩΓΑ ΙΝΔΟΛΗΣ Ή ΒΕΝΖΙΜΙΔΑΖΟΛΗΣ ΓΙΑ ΤΗ ΡΥΘΜΙΣΗ ΤΗΣ ΙκΒ ΚΙΝΑΣΗΣ ΚΑΙ ΕΝΔΙΑΜΕΣΑ ΠΡΟΪΟΝΤΑ ΓΙΑ ΤΗΝ ΠΑΡΑΣΚΕΥΗ ΤΟΥΣ |
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| DE10237722A DE10237722A1 (de) | 2002-08-17 | 2002-08-17 | Indol- oder Benzimidazolderivate zur Modulation der IKappaB-Kinase |
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