KR100869616B1 - 프롤린 유도체 및 그의 다이펩티딜 펩티다제-iv저해제로서의 용도 - Google Patents

프롤린 유도체 및 그의 다이펩티딜 펩티다제-iv저해제로서의 용도 Download PDF

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KR100869616B1
KR100869616B1 KR1020067023663A KR20067023663A KR100869616B1 KR 100869616 B1 KR100869616 B1 KR 100869616B1 KR 1020067023663 A KR1020067023663 A KR 1020067023663A KR 20067023663 A KR20067023663 A KR 20067023663A KR 100869616 B1 KR100869616 B1 KR 100869616B1
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pyrrolidin
methanone
compound
alkyl
compounds
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KR20070009699A (ko
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베르나드 휼린
데이비드 왈터 피오트로스키
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화이자 프로덕츠 인코포레이티드
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KR1020067023663A 2004-05-12 2005-04-29 프롤린 유도체 및 그의 다이펩티딜 펩티다제-iv저해제로서의 용도 Expired - Fee Related KR100869616B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US57030004P 2004-05-12 2004-05-12
US60/570,300 2004-05-12
US66430505P 2005-03-21 2005-03-21
US60/664,305 2005-03-21

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KR20070009699A KR20070009699A (ko) 2007-01-18
KR100869616B1 true KR100869616B1 (ko) 2008-11-21

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US (4) US7291618B2 (enExample)
EP (2) EP2116541B1 (enExample)
JP (1) JP4227660B2 (enExample)
KR (1) KR100869616B1 (enExample)
AP (1) AP2320A (enExample)
AR (1) AR049894A1 (enExample)
AT (1) ATE437870T1 (enExample)
AU (1) AU2005247684B2 (enExample)
BR (1) BRPI0510284A (enExample)
CA (1) CA2566108C (enExample)
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DK (1) DK1753748T3 (enExample)
EA (1) EA011086B9 (enExample)
EC (1) ECSP066985A (enExample)
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US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
PT1753748E (pt) 2004-05-12 2009-08-28 Pfizer Prod Inc Derivados de prolina e a sua utilização como inibidores de dipeptidil peptidase iv
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
WO2006071958A1 (en) 2004-12-29 2006-07-06 Millennium Pharmaceuticals, Inc. Compounds useful as chemokine receptor antagonists
US7880002B2 (en) 2004-12-29 2011-02-01 Millennium Pharmaceuticals, Inc. Substituted piperazinyl-pyrrolidine compounds useful as chemokine receptor antagonists
WO2006073167A1 (ja) * 2005-01-07 2006-07-13 Ono Pharmaceutical Co., Ltd. ピロリジン誘導体
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
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