KR100606323B1 - 1-치환된 5- 또는 3-히드록시피라졸의 제조 방법 - Google Patents

1-치환된 5- 또는 3-히드록시피라졸의 제조 방법 Download PDF

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Publication number
KR100606323B1
KR100606323B1 KR1020017006275A KR20017006275A KR100606323B1 KR 100606323 B1 KR100606323 B1 KR 100606323B1 KR 1020017006275 A KR1020017006275 A KR 1020017006275A KR 20017006275 A KR20017006275 A KR 20017006275A KR 100606323 B1 KR100606323 B1 KR 100606323B1
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South Korea
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formula
reaction
alkyl
methyl
substituted
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Korean (ko)
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KR20010080490A (ko
Inventor
볼커 마이발드
아드리안 스타인메쯔
미하엘 라크
노르버트 괴쯔
롤란트 괴쯔
요헴 헨켈만
하이케 베커
유안요제 아이스카바예토
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바스프 악티엔게젤샤프트
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020017006275A 1998-11-19 1999-11-06 1-치환된 5- 또는 3-히드록시피라졸의 제조 방법 Expired - Fee Related KR100606323B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19853502 1998-11-19
DE19853502.3 1998-11-19

Publications (2)

Publication Number Publication Date
KR20010080490A KR20010080490A (ko) 2001-08-22
KR100606323B1 true KR100606323B1 (ko) 2006-08-02

Family

ID=7888404

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020017006275A Expired - Fee Related KR100606323B1 (ko) 1998-11-19 1999-11-06 1-치환된 5- 또는 3-히드록시피라졸의 제조 방법

Country Status (27)

Country Link
US (1) US6392058B1 (https=)
EP (1) EP1131299B1 (https=)
JP (1) JP2002530381A (https=)
KR (1) KR100606323B1 (https=)
CN (1) CN1131218C (https=)
AR (1) AR021315A1 (https=)
AT (1) ATE250037T1 (https=)
AU (1) AU766546B2 (https=)
BG (1) BG65026B1 (https=)
BR (1) BR9915492A (https=)
CA (1) CA2351370C (https=)
CZ (1) CZ301828B6 (https=)
DE (1) DE59907053D1 (https=)
DK (1) DK1131299T3 (https=)
EA (1) EA003753B1 (https=)
ES (1) ES2207988T3 (https=)
HU (1) HU224721B1 (https=)
IL (1) IL143035A (https=)
NO (1) NO318052B1 (https=)
NZ (1) NZ511645A (https=)
PL (1) PL205283B1 (https=)
PT (1) PT1131299E (https=)
SK (1) SK286367B6 (https=)
TR (1) TR200101404T2 (https=)
UA (1) UA67815C2 (https=)
WO (1) WO2000031042A2 (https=)
ZA (1) ZA200104961B (https=)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA67815C2 (uk) 1998-11-19 2004-07-15 Басф Акцієнгезелльшафт Спосіб одержання 1-заміщених 5- або 3-гідроксипіразолів
CN101781201B (zh) * 2009-06-26 2013-07-31 上海海事大学 一种合成3-烷氧基丙烯酸酯的改进工艺
CN103698459A (zh) * 2013-12-30 2014-04-02 中美华世通生物医药科技（武汉）有限公司 一种药物中游离肼的检测方法
CN104059020B (zh) * 2014-06-27 2016-08-31 湖南海利常德农药化工有限公司 1-芳基-5-羟基吡唑的制备方法
WO2016184378A1 (zh) 2015-05-18 2016-11-24 沈阳中化农药化工研发有限公司 含嘧啶的取代吡唑类化合物及其制备方法和用途
CN108129305A (zh) * 2017-12-25 2018-06-08 凯莱英生命科学技术(天津)有限公司 E-烷氧基丙烯酸酯连续合成的方法
CN109320457A (zh) * 2018-10-12 2019-02-12 凯莱英医药化学（阜新）技术有限公司 羟基吡唑类化合物的制备方法及装置
CN112480008B (zh) * 2020-12-21 2022-10-11 浙江工业大学 一种1-甲基-5-羟基吡唑的合成方法
WO2024100791A1 (ja) 2022-11-09 2024-05-16 株式会社日本ファインケム １－アルキル－５－ヒドロキシピラゾールの製造方法

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JPS5714997A (en) 1980-06-30 1982-01-26 Matsushita Electric Works Ltd Signal processing circuit for ionization smoke sensor
JPS58140073A (ja) 1982-02-09 1983-08-19 Nissan Chem Ind Ltd １−メチル−５−ハイドロキシピラゾ−ルの製造法
JPS58174369A (ja) 1983-03-26 1983-10-13 Nissan Chem Ind Ltd １−メチル−５−ハイドロキシピラゾ−ル−４−カルボン酸低級アルキルエステルおよびその製造法
JPS6051175A (ja) 1983-08-30 1985-03-22 Nissan Chem Ind Ltd ピラゾ−ル誘導体および選択性除草剤
JPS61189271A (ja) * 1985-02-19 1986-08-22 Ube Ind Ltd １−メチル−５−ヒドロキシピラゾ−ルの製法
JPH0662577B2 (ja) 1985-04-03 1994-08-17 日産化学工業株式会社 １−メチル−５−ヒドロキシピラゾ−ルの製造法
JPS61257974A (ja) 1985-05-11 1986-11-15 Nissan Chem Ind Ltd ピラゾ−ル誘導体，その製造方法および選択性除草剤
US4744815A (en) 1985-05-11 1988-05-17 Nissan Chemical Industries, Ltd. 4-benzoyl-1-alkyl (alkenyl) - pyrazoles, composition containing them, herbicidal method of using them, and intermediate in their preparation
US4643757A (en) 1985-05-20 1987-02-17 Nissan Chemical Industries, Ltd. Herbicidal 4-benzoyl-1-methyl-5-hydroxypyrazoles
JPH0688977B2 (ja) 1985-05-23 1994-11-09 日産化学工業株式会社 １−メチル−５−ヒドロキシピラゾ−ルの製造法
JPH0730031B2 (ja) * 1986-04-02 1995-04-05 日産化学工業株式会社 ２―ピラゾリン―５―オン類の製造法
DE4230283A1 (de) * 1992-09-10 1994-03-17 Basf Ag Verfahren zur Herstellung von alpha, beta-ungesättigten beta-Oxycarbonsäurechloriden
US5607898A (en) 1993-08-02 1997-03-04 Idemitsu Kosan Company, Ltd. Pyrazole derivatives
JPH0735361B2 (ja) 1993-09-09 1995-04-19 日産化学工業株式会社 ヒドラゾン誘導体およびその製造方法
BR9508191A (pt) 1994-06-27 1997-08-12 Idemitsu Kosan Co Composição herbicida
EP0810226B1 (en) 1995-02-13 2003-05-02 Idemitsu Kosan Company Limited Pyrazole derivatives
JP4117386B2 (ja) 1995-02-24 2008-07-16 ビーエーエスエフ ソシエタス・ヨーロピア ピラゾリルベンゾイル誘導体
AR001805A1 (es) 1995-03-28 1997-12-10 Idemitsu Kosan Co Derivado de pirazol, acido carboxilico util como material de partida en la sintesis de dicho derivado y composicion herbicida que lo contiene
EP0819691A4 (en) 1995-04-05 1998-07-29 Idemitsu Kosan Co PYRAZOLE DERIVATIVES
BR9609502A (pt) 1995-06-29 1999-05-25 Du Pont Composto composição herbicida e método para controle do crescimento de vegetação indesejável
WO1997008164A1 (en) 1995-08-25 1997-03-06 E.I. Du Pont De Nemours And Company Bicyclic herbicides
EP0970956A4 (en) 1995-10-04 2000-01-12 Idemitsu Kosan Co PYRAZOLE DERIVATIVES
US5985799A (en) 1995-11-17 1999-11-16 E.I. Du Pont De Nemours And Company Tricyclic herbicidal heterocycles
WO1997023135A1 (fr) 1995-12-25 1997-07-03 Idemitsu Kosan Co., Ltd. Composition herbicide
US5631210A (en) 1996-06-14 1997-05-20 E. I. Du Pont De Nemours And Company Herbicidal thiophene ketones
JP3719318B2 (ja) * 1996-10-18 2005-11-24 宇部興産株式会社 １−エチル−５−ヒドロキシピラゾールの製法
US5808092A (en) 1996-10-18 1998-09-15 Ube Industries, Ltd. Process for preparing-1-ethyl-5-hydroxypyrazole
US5663365A (en) * 1996-10-29 1997-09-02 Japan Hydrazine Co., Ltd. Process for the preparation of pyrazolones
UA67815C2 (uk) 1998-11-19 2004-07-15 Басф Акцієнгезелльшафт Спосіб одержання 1-заміщених 5- або 3-гідроксипіразолів

Also Published As

Publication number Publication date
HUP0104504A3 (en) 2002-12-28
AR021315A1 (es) 2002-07-17
IL143035A0 (en) 2002-04-21
IL143035A (en) 2005-07-25
DE59907053D1 (de) 2003-10-23
WO2000031042A2 (de) 2000-06-02
CZ301828B6 (cs) 2010-07-07
CN1131218C (zh) 2003-12-17
EP1131299B1 (de) 2003-09-17
CZ20011713A3 (cs) 2002-01-16
ZA200104961B (en) 2002-06-18
JP2002530381A (ja) 2002-09-17
NO20012470D0 (no) 2001-05-18
WO2000031042A3 (de) 2000-10-26
EP1131299A2 (de) 2001-09-12
BG65026B1 (bg) 2006-12-29
AU1380900A (en) 2000-06-13
BG105538A (en) 2002-04-30
PL205283B1 (pl) 2010-03-31
EA003753B1 (ru) 2003-08-28
BR9915492A (pt) 2001-08-07
EA200100522A1 (ru) 2001-10-22
DK1131299T3 (da) 2004-02-02
CN1330639A (zh) 2002-01-09
NO20012470L (no) 2001-05-21
PT1131299E (pt) 2004-02-27
PL348751A1 (en) 2002-06-03
UA67815C2 (uk) 2004-07-15
HU224721B1 (en) 2006-01-30
KR20010080490A (ko) 2001-08-22
ES2207988T3 (es) 2004-06-01
NZ511645A (en) 2003-07-25
CA2351370A1 (en) 2000-06-02
SK286367B6 (sk) 2008-08-05
SK6792001A3 (en) 2001-11-06
AU766546B2 (en) 2003-10-16
ATE250037T1 (de) 2003-10-15
CA2351370C (en) 2008-03-11
TR200101404T2 (tr) 2002-01-21
NO318052B1 (no) 2005-01-24
US6392058B1 (en) 2002-05-21
HUP0104504A2 (hu) 2002-03-28

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