KR100187328B1 - 15-데옥시스퍼구알린 동족체, 그의 제조방법 및 치료학적 용도 - Google Patents

15-데옥시스퍼구알린 동족체, 그의 제조방법 및 치료학적 용도 Download PDF

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KR100187328B1
KR100187328B1 KR1019930025761A KR930025761A KR100187328B1 KR 100187328 B1 KR100187328 B1 KR 100187328B1 KR 1019930025761 A KR1019930025761 A KR 1019930025761A KR 930025761 A KR930025761 A KR 930025761A KR 100187328 B1 KR100187328 B1 KR 100187328B1
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South Korea
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group
formula
compound
iii
och
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KR1019930025761A
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KR940014435A (ko
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빠뜨리쓰르노
뤽르브르똥
필립데르빠스
소뜨쌍레뜨
페트릭뒤따르뜨르
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프랑소와 피까르
푸르니에엥뒤스트리에에쌍뜨
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/04—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
    • C07C279/12—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton being further substituted by nitrogen atoms not being part of nitro or nitroso groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/20—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylguanidines
    • C07C279/24—Y being a hetero atom

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Steroid Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Soil Conditioners And Soil-Stabilizing Materials (AREA)
  • Curing Cements, Concrete, And Artificial Stone (AREA)
KR1019930025761A 1992-12-02 1993-11-30 15-데옥시스퍼구알린 동족체, 그의 제조방법 및 치료학적 용도 Expired - Fee Related KR100187328B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9214517 1992-12-02
FR9214517A FR2698628B1 (fr) 1992-12-02 1992-12-02 Analogues de 15-déoxyspergualine, leur procédé de préparation et leur utilisation en thérapeutique.

Publications (2)

Publication Number Publication Date
KR940014435A KR940014435A (ko) 1994-07-18
KR100187328B1 true KR100187328B1 (ko) 1999-05-15

Family

ID=9436147

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019930025761A Expired - Fee Related KR100187328B1 (ko) 1992-12-02 1993-11-30 15-데옥시스퍼구알린 동족체, 그의 제조방법 및 치료학적 용도

Country Status (24)

Country Link
US (1) US5476870A (enExample)
EP (1) EP0600762B1 (enExample)
JP (1) JP2945261B2 (enExample)
KR (1) KR100187328B1 (enExample)
CN (1) CN1045431C (enExample)
AT (1) ATE140215T1 (enExample)
AU (1) AU664124B2 (enExample)
CA (1) CA2110437C (enExample)
CZ (1) CZ284958B6 (enExample)
DE (1) DE69303583T2 (enExample)
DK (1) DK0600762T3 (enExample)
ES (1) ES2092263T3 (enExample)
FI (1) FI112211B (enExample)
FR (1) FR2698628B1 (enExample)
GR (1) GR3021269T3 (enExample)
HK (1) HK1000467A1 (enExample)
HU (1) HU218908B (enExample)
NO (1) NO180483C (enExample)
NZ (1) NZ250330A (enExample)
RU (1) RU2114823C1 (enExample)
SK (1) SK280286B6 (enExample)
TW (1) TW311132B (enExample)
UA (1) UA39920C2 (enExample)
ZA (1) ZA938821B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20160109293A (ko) 2015-03-10 2016-09-21 하경훈 마늘꼭지 절단기의 절단장치

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69600780T2 (de) * 1995-02-10 1999-05-27 Fournier Industrie Et Sante, Paris 15-deoxyspergualin-analoge verbindungen, ihre verwendung als therapeutika und verfahren zu ihrer herstellung
FR2734263B1 (fr) * 1995-05-17 1997-06-20 Fournier Ind & Sante Analogues de la 15-deoxyspergualine, leur procede de preparation et leur utilisation en therapeutique
JP3090960B2 (ja) * 1996-12-20 2000-09-25 エス カー ヴエー トローストベルク アクチエンゲゼルシヤフト クレアチン―ピルベート及びその製造方法
DE19728436A1 (de) * 1997-07-03 1999-01-07 Niels Franke Niedrigdosierte 15-Desoxyspergualin-Präparate
ES2170042T3 (es) * 1998-08-28 2004-10-01 Gryphon Therapeutics, Inc. Procedimiento para la preparacion de cadenas de poliamida de longitud precisa y sus conjugados con proteinas.
DE19923961A1 (de) * 1999-05-25 2000-11-30 Euro Nippon Kayaku Gmbh Verwendung von 15-Deoxyspergualin zur Behandlung von hyperreaktiven entzündlichen Erkrankungen und Autoimmunerkrankungen
US8017804B2 (en) 2004-05-05 2011-09-13 Silence Therapeutics Ag Lipids, lipid complexes and use thereof
DK1830888T3 (en) 2004-12-27 2015-10-19 Silence Therapeutics Gmbh LIPID COMPLEX COATED WITH PEG AND APPLICATION THEREOF
EP2269980A4 (de) 2008-12-24 2011-05-18 Vertex Closed Joint Stock Company Creatinamide, verfahren zu ihrer herstellung und wirkstoff zur ausführung einer neuroprotektiven aktion
RU2428414C2 (ru) 2009-11-03 2011-09-10 Закрытое Акционерное Общество "Вертекс" Способ получения амидов креатина
FR2963238B1 (fr) * 2010-07-29 2012-12-28 Fournier Lab Sa Derives de 15-desoxyspergualine pour le traitement et/ou la prevention des maladies inflammatoires oculaires
EP2598131A1 (fr) * 2010-07-29 2013-06-05 Laboratoires Fournier S.A. Composes pour le traitement/la prevention des maladies inflammatoires oculaires
FR3050455B1 (fr) * 2016-04-26 2019-06-14 Temisis Derives amides des acides polycafeoylquiniques, procede de preparation et utilisations

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5942356A (ja) * 1982-09-02 1984-03-08 Microbial Chem Res Found スパガリン関連化合物およびその製造法
ES2039213T3 (es) * 1986-04-04 1993-09-16 Microbial Chemistry Research Foundation Procedimiento para producir nuevos compuestos relacionados con espergualina.
US5061787A (en) * 1988-06-24 1991-10-29 Nippon Kayaku Kabushiki Kaisha Novel spergualin-related compounds and compositions

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20160109293A (ko) 2015-03-10 2016-09-21 하경훈 마늘꼭지 절단기의 절단장치

Also Published As

Publication number Publication date
HU218908B (hu) 2000-12-28
TW311132B (enExample) 1997-07-21
FI935318A0 (fi) 1993-11-29
DE69303583T2 (de) 1996-11-21
CZ262293A3 (en) 1994-06-15
JPH06293728A (ja) 1994-10-21
CA2110437A1 (en) 1994-06-03
HU9303406D0 (en) 1994-03-28
DE69303583D1 (de) 1996-08-14
RU2114823C1 (ru) 1998-07-10
HUT65782A (en) 1994-07-28
FR2698628B1 (fr) 1995-02-17
GR3021269T3 (en) 1997-01-31
DK0600762T3 (da) 1996-11-11
AU664124B2 (en) 1995-11-02
UA39920C2 (uk) 2001-07-16
SK280286B6 (sk) 1999-11-08
CN1045431C (zh) 1999-10-06
CZ284958B6 (cs) 1999-04-14
ATE140215T1 (de) 1996-07-15
CN1095709A (zh) 1994-11-30
FI935318L (fi) 1994-06-03
NO180483C (no) 1997-04-30
US5476870A (en) 1995-12-19
FR2698628A1 (fr) 1994-06-03
NO934338L (no) 1994-06-03
NO180483B (no) 1997-01-20
ZA938821B (en) 1994-06-30
FI112211B (fi) 2003-11-14
HK1000467A1 (en) 1998-03-27
ES2092263T3 (es) 1996-11-16
JP2945261B2 (ja) 1999-09-06
CA2110437C (en) 1999-04-13
NZ250330A (en) 1995-06-27
SK135793A3 (en) 1994-06-08
EP0600762B1 (fr) 1996-07-10
EP0600762A1 (fr) 1994-06-08
NO934338D0 (no) 1993-11-30
AU5188393A (en) 1994-06-16
KR940014435A (ko) 1994-07-18

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