JPS6041609A - 二元熱力学的活性を有する浸透装置 - Google Patents
二元熱力学的活性を有する浸透装置Info
- Publication number
- JPS6041609A JPS6041609A JP59024947A JP2494784A JPS6041609A JP S6041609 A JPS6041609 A JP S6041609A JP 59024947 A JP59024947 A JP 59024947A JP 2494784 A JP2494784 A JP 2494784A JP S6041609 A JPS6041609 A JP S6041609A
- Authority
- JP
- Japan
- Prior art keywords
- composition
- cellulose
- wall
- osmotic
- compartment
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
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- 150000003892 tartrate salts Chemical class 0.000 description 1
- RBTVSNLYYIMMKS-UHFFFAOYSA-N tert-butyl 3-aminoazetidine-1-carboxylate;hydrochloride Chemical compound Cl.CC(C)(C)OC(=O)N1CC(N)C1 RBTVSNLYYIMMKS-UHFFFAOYSA-N 0.000 description 1
- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
- 125000000383 tetramethylene group Chemical group [H]C([H])([*:1])C([H])([H])C([H])([H])C([H])([H])[*:2] 0.000 description 1
- 229960004605 timolol Drugs 0.000 description 1
- VZCYOOQTPOCHFL-UHFFFAOYSA-N trans-butenedioic acid Natural products OC(=O)C=CC(O)=O VZCYOOQTPOCHFL-UHFFFAOYSA-N 0.000 description 1
- 229910052723 transition metal Inorganic materials 0.000 description 1
- GFNANZIMVAIWHM-OBYCQNJPSA-N triamcinolone Chemical compound O=C1C=C[C@]2(C)[C@@]3(F)[C@@H](O)C[C@](C)([C@@]([C@H](O)C4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 GFNANZIMVAIWHM-OBYCQNJPSA-N 0.000 description 1
- 229960005294 triamcinolone Drugs 0.000 description 1
- PVNIQBQSYATKKL-UHFFFAOYSA-N tripalmitin Chemical compound CCCCCCCCCCCCCCCC(=O)OCC(OC(=O)CCCCCCCCCCCCCCC)COC(=O)CCCCCCCCCCCCCCC PVNIQBQSYATKKL-UHFFFAOYSA-N 0.000 description 1
- 150000004043 trisaccharides Chemical class 0.000 description 1
- RYFMWSXOAZQYPI-UHFFFAOYSA-K trisodium phosphate Chemical compound [Na+].[Na+].[Na+].[O-]P([O-])([O-])=O RYFMWSXOAZQYPI-UHFFFAOYSA-K 0.000 description 1
- 229910052721 tungsten Inorganic materials 0.000 description 1
- 229940045136 urea Drugs 0.000 description 1
- 210000001215 vagina Anatomy 0.000 description 1
- 229960002726 vincamine Drugs 0.000 description 1
- 229920002554 vinyl polymer Polymers 0.000 description 1
- 210000001835 viscera Anatomy 0.000 description 1
- 230000009278 visceral effect Effects 0.000 description 1
- 238000000196 viscometry Methods 0.000 description 1
- 230000001755 vocal effect Effects 0.000 description 1
- 229920003176 water-insoluble polymer Polymers 0.000 description 1
- 229920003169 water-soluble polymer Polymers 0.000 description 1
- NWONKYPBYAMBJT-UHFFFAOYSA-L zinc sulfate Chemical compound [Zn+2].[O-]S([O-])(=O)=O NWONKYPBYAMBJT-UHFFFAOYSA-L 0.000 description 1
- 229960001763 zinc sulfate Drugs 0.000 description 1
- 229910000368 zinc sulfate Inorganic materials 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Separation Using Semi-Permeable Membranes (AREA)
- External Artificial Organs (AREA)
- Infusion, Injection, And Reservoir Apparatuses (AREA)
- Medical Preparation Storing Or Oral Administration Devices (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49376083A | 1983-05-11 | 1983-05-11 | |
| US493760 | 1983-05-11 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS6041609A true JPS6041609A (ja) | 1985-03-05 |
| JPH0575725B2 JPH0575725B2 (OSRAM) | 1993-10-21 |
Family
ID=23961585
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP59024947A Granted JPS6041609A (ja) | 1983-05-11 | 1984-02-13 | 二元熱力学的活性を有する浸透装置 |
Country Status (20)
| Country | Link |
|---|---|
| JP (1) | JPS6041609A (OSRAM) |
| AT (1) | AT397180B (OSRAM) |
| AU (1) | AU566110B2 (OSRAM) |
| BE (1) | BE898819A (OSRAM) |
| CA (1) | CA1222950A (OSRAM) |
| CH (1) | CH669329A5 (OSRAM) |
| DE (1) | DE3417113A1 (OSRAM) |
| DK (1) | DK163910C (OSRAM) |
| ES (1) | ES8503503A1 (OSRAM) |
| FR (1) | FR2545721B1 (OSRAM) |
| GB (1) | GB2140687B (OSRAM) |
| IE (1) | IE56515B1 (OSRAM) |
| IL (1) | IL71727A (OSRAM) |
| IT (1) | IT1178911B (OSRAM) |
| MX (1) | MX163518B (OSRAM) |
| NL (1) | NL192250C (OSRAM) |
| NO (1) | NO170834C (OSRAM) |
| NZ (1) | NZ206600A (OSRAM) |
| SE (1) | SE455918B (OSRAM) |
| ZA (1) | ZA842422B (OSRAM) |
Cited By (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6153214A (ja) * | 1983-08-16 | 1986-03-17 | ザ ウエルカム フアウンデ−シヨン リミテツド | 調節された方法による有効成分の放出を可能にする医薬組成物 |
| JPS62185010A (ja) * | 1986-02-07 | 1987-08-13 | アルザ コ−ポレ−シヨン | 生体受容性を強化した薬物送達システム |
| JPH01113316A (ja) * | 1987-10-02 | 1989-05-02 | Alza Corp | 心臓血管系疾病処置用投薬形態 |
| JPH01242528A (ja) * | 1988-03-21 | 1989-09-27 | Alza Corp | 浸透性投薬形態 |
| JPH01313432A (ja) * | 1988-06-02 | 1989-12-18 | Alza Corp | ジルチアゼム投与用投薬形態 |
| JPH05504074A (ja) * | 1989-12-06 | 1993-07-01 | メドトロニック インコーポレーテッド | 比色定量分析による筋肉適合性検出 |
| JPH05506858A (ja) * | 1990-05-07 | 1993-10-07 | アルザ コーポレイション | 抗パーキンソン病剤供給用投与形態 |
| JP2007505894A (ja) * | 2003-09-19 | 2007-03-15 | サン・ファーマシューティカル・インダストリーズ・リミテッド | 経口薬送達システム |
| JP2008069177A (ja) * | 1993-05-27 | 2008-03-27 | Alza Corp | 抗鬱薬投薬形態 |
| JP2008525335A (ja) * | 2004-12-24 | 2008-07-17 | バイエル・ヘルスケア・アクチェンゲゼルシャフト | 経口投与できる固体の放出改変型医薬投与形 |
| JP2012528799A (ja) * | 2009-06-02 | 2012-11-15 | ダウ グローバル テクノロジーズ エルエルシー | 徐放製剤 |
| JP2015007144A (ja) * | 2014-10-17 | 2015-01-15 | ダウ グローバル テクノロジーズ エルエルシー | 徐放製剤 |
Families Citing this family (49)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4600773A (en) * | 1983-12-01 | 1986-07-15 | Eli Lilly And Company | Crystalline cephalexin hydrochloride monohydrate |
| US4624847A (en) * | 1985-04-22 | 1986-11-25 | Alza Corporation | Drug delivery device for programmed delivery of beneficial drug |
| US4704118A (en) * | 1985-08-16 | 1987-11-03 | Alza Corporation | Ruminant dispensing device with thermo-activated memory |
| ES8800043A1 (es) * | 1985-08-16 | 1987-10-16 | Alza Corp | Un dispositivo distribuidor para descargar una formulacion de agente beneficioso a un entorno de uso |
| US4963141A (en) * | 1985-08-16 | 1990-10-16 | Alza Corporation | Dispensing system for administering beneficial agent formulation to ruminants |
| US4716496A (en) * | 1986-05-09 | 1987-12-29 | Eaton Corporation | Panel-mounted control station housing |
| US4814181A (en) * | 1987-09-03 | 1989-03-21 | Alza Corporation | Dosage form comprising fast agent delivery followed by slow agent delivery |
| ES2037179T3 (es) * | 1987-11-25 | 1993-06-16 | American Cyanamid Company | Sistema de liberacion sostenida (controlada) para bloqueadores de canales de calcio de dihidropiridina. |
| US4855141A (en) * | 1988-03-25 | 1989-08-08 | Alza Corporation | Device comprising means for protecting and dispensing fluid sensitive medicament |
| IL91398A (en) * | 1988-08-30 | 1994-05-30 | Pfizer | Pharmaceutical delivery device comprising active substance surrounded by asymmetric membrane |
| US5612059A (en) * | 1988-08-30 | 1997-03-18 | Pfizer Inc. | Use of asymmetric membranes in delivery devices |
| GR1000270B (el) * | 1988-09-30 | 1992-05-12 | Alza Corp | Μορφη δοσολογιας για θεραπεια καρδιαγγειακων ασθενειων. |
| IL92966A (en) * | 1989-01-12 | 1995-07-31 | Pfizer | Dispensing devices powered by hydrogel |
| US5030452A (en) * | 1989-01-12 | 1991-07-09 | Pfizer Inc. | Dispensing devices powered by lyotropic liquid crystals |
| US5108756A (en) * | 1989-01-12 | 1992-04-28 | Pfizer Inc. | Dispensing devices powered by lyotropic liquid crystals |
| EP0408496A3 (en) * | 1989-07-12 | 1992-07-01 | Ciba-Geigy Ag | Solid dosage form for pharmaceutical substances |
| US5000962A (en) * | 1989-08-25 | 1991-03-19 | Schering Corporation | Long acting diltiazem formulation |
| US4992277A (en) * | 1989-08-25 | 1991-02-12 | Schering Corporation | Immediate release diltiazem formulation |
| US5081161A (en) * | 1990-06-15 | 1992-01-14 | E. I. Du Pont De Nemours And Company | Process for making shaped articles of a thermoplastic resin having a microcellular structure |
| NZ238867A (en) * | 1990-07-12 | 1993-08-26 | Alza Corp | Dosage form for delayed release comprising pharmaceutically active substance and a drug-release hindering means and a second composition which imbibes fluid, expands, and ejects the active substance from the device |
| DK0542926T3 (da) * | 1990-08-07 | 1995-05-15 | Pfizer | Brug af grænsefladepolymeriserede membraner i frigivelsesanordninger |
| US5166145A (en) * | 1990-09-10 | 1992-11-24 | Alza Corporation | Antiemetic therapy |
| ES2053339T3 (es) * | 1990-09-28 | 1994-07-16 | Pfizer | Dispositivo dispensador conteniendo un medio hidrofobo. |
| US5208037A (en) * | 1991-04-22 | 1993-05-04 | Alza Corporation | Dosage forms comprising polymers comprising different molecular weights |
| EP0612519B1 (en) * | 1993-02-23 | 2001-04-04 | Wolfgang Dr. Werner | Use of a calcium formulation in a medicament for therapeutic application to milk cows suffering from hypocalcaemia |
| US6287598B1 (en) * | 1993-05-28 | 2001-09-11 | Alza Corporation | Method for providing sustained antiepileptic therapy |
| HU213407B (en) * | 1993-12-09 | 1997-06-30 | Egyt Gyogyszervegyeszeti Gyar | Process for producing tablet with diffusive-osmotic release |
| US5460826A (en) * | 1994-06-27 | 1995-10-24 | Alza Corporation | Morphine therapy |
| US5948787A (en) | 1997-02-28 | 1999-09-07 | Alza Corporation | Compositions containing opiate analgesics |
| DE19962924A1 (de) | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
| BR0115382A (pt) * | 2000-10-30 | 2003-09-16 | Euro Celtique Sa | Formulações para liberação controlada de hidrocodona, método de produzir analgesia efetiva, processo de preparação de uma forma farmacêutica de um sólido oral de liberação controlada, liberação controlada da forma farmacêutica oral e uso da forma farmacêutica |
| US20110104214A1 (en) | 2004-04-15 | 2011-05-05 | Purdue Pharma L.P. | Once-a-day oxycodone formulations |
| DE10129725A1 (de) | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
| DE10300111A1 (de) | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
| US10213387B2 (en) | 2003-09-19 | 2019-02-26 | Sun Pharma Advanced Research Company Ltd. | Oral drug delivery system |
| US10226428B2 (en) | 2003-09-19 | 2019-03-12 | Sun Pharma Advanced Research Company Ltd. | Oral drug delivery system |
| DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
| EP1685841A1 (en) | 2005-01-31 | 2006-08-02 | Bayer Health Care Aktiengesellschaft | Prevention and treatment of thromboembolic disorders |
| DE102005031577A1 (de) | 2005-07-06 | 2007-01-11 | Bayer Healthcare Ag | Pharmazeutische Darreichungsformen enthaltend eine Wirkstoffkombination von Nifedipin und/oder Nisoldipin und einem Angiotensin-II Antagonisten |
| DE102005045518A1 (de) | 2005-09-23 | 2007-03-29 | Bayer Healthcare Ag | 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung |
| DE102005047561A1 (de) | 2005-10-04 | 2007-04-05 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung |
| PT1934208E (pt) | 2005-10-04 | 2011-06-01 | Bayer Schering Pharma Ag | Nova forma polimorfa de 5-cloro-n-({(5s)-2-oxo-3-[4-(3- oxo-4-morfolinil)-fenil]-1,3-oxazolidin-5-il}-metil)-2- tiofenocarboxamida |
| DE102008059206A1 (de) | 2008-11-27 | 2010-06-10 | Bayer Schering Pharma Aktiengesellschaft | Pharmazeutische Darreichungsform enthaltend Nifedipin oder Nisoldipin und einen Angiotensin-II Antagonisten und/oder ein Diuretikum |
| DE102011007272A1 (de) | 2011-04-13 | 2012-10-18 | Bayer Pharma Aktiengesellschaft | Verzweigte 3-Phenylpropionsäure-Derivate und ihre Verwendung |
| MX2014013320A (es) | 2012-05-07 | 2015-08-10 | Bayer Pharma AG | Procedimiento de fabricacion de una forma de dosificacion farmaceutica que comprende nifedipina y candesartan cilexetilo. |
| UY34856A (es) | 2012-07-03 | 2013-12-31 | Bayer Pharma AG | Formas de presentación farmacéuticas que contienen 5-cloro-n-({(5s)-2-oxo-3-[4-(3-oxo-4- morfolinil)-fenil]-1,3-oxazolidin-5-il}-metil)-2-tiofencarboxamida |
| US10905667B2 (en) | 2018-07-24 | 2021-02-02 | Bayer Pharma Aktiengesellschaft | Orally administrable modified-release pharmaceutical dosage form |
| JP2021531297A (ja) | 2018-07-24 | 2021-11-18 | バイエル・アクチエンゲゼルシヤフト | 経口投与可能であり、修飾された放出を有する薬学的投薬形態 |
| AU2019311234A1 (en) | 2018-07-24 | 2021-02-04 | Bayer Aktiengesellschaft | Pharmaceutical dosage form which can be administered orally and has modified release |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5793065A (en) * | 1980-11-25 | 1982-06-09 | Alza Corp | Permeation apparatus having hydrogel drive member |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL38538A (en) * | 1971-01-13 | 1974-09-10 | Alza Corp | Osmotic dispenser |
| US3977404A (en) * | 1975-09-08 | 1976-08-31 | Alza Corporation | Osmotic device having microporous reservoir |
| US4111202A (en) * | 1976-11-22 | 1978-09-05 | Alza Corporation | Osmotic system for the controlled and delivery of agent over time |
| US4160452A (en) * | 1977-04-07 | 1979-07-10 | Alza Corporation | Osmotic system having laminated wall comprising semipermeable lamina and microporous lamina |
| US4200098A (en) * | 1978-10-23 | 1980-04-29 | Alza Corporation | Osmotic system with distribution zone for dispensing beneficial agent |
| US4265874A (en) * | 1980-04-25 | 1981-05-05 | Alza Corporation | Method of delivering drug with aid of effervescent activity generated in environment of use |
| US4449983A (en) * | 1982-03-22 | 1984-05-22 | Alza Corporation | Simultaneous delivery of two drugs from unit delivery device |
-
1983
- 1983-12-16 NZ NZ206600A patent/NZ206600A/en unknown
- 1983-12-19 AU AU22511/83A patent/AU566110B2/en not_active Expired
- 1983-12-22 GB GB08334189A patent/GB2140687B/en not_active Expired
-
1984
- 1984-01-05 IE IE10/84A patent/IE56515B1/en not_active IP Right Cessation
- 1984-01-24 NO NO840248A patent/NO170834C/no not_active IP Right Cessation
- 1984-02-02 BE BE0/212326A patent/BE898819A/fr not_active IP Right Cessation
- 1984-02-13 JP JP59024947A patent/JPS6041609A/ja active Granted
- 1984-02-24 DK DK099784A patent/DK163910C/da not_active IP Right Cessation
- 1984-02-29 MX MX200502A patent/MX163518B/es unknown
- 1984-03-15 AT AT0088084A patent/AT397180B/de not_active IP Right Cessation
- 1984-03-23 IT IT8467283A patent/IT1178911B/it active
- 1984-03-30 ZA ZA842422A patent/ZA842422B/xx unknown
- 1984-04-05 FR FR8405362A patent/FR2545721B1/fr not_active Expired
- 1984-04-27 ES ES532018A patent/ES8503503A1/es not_active Expired
- 1984-05-02 IL IL71727A patent/IL71727A/xx not_active IP Right Cessation
- 1984-05-08 NL NL8401470A patent/NL192250C/nl not_active IP Right Cessation
- 1984-05-09 DE DE3417113A patent/DE3417113A1/de active Granted
- 1984-05-09 SE SE8402512A patent/SE455918B/sv not_active IP Right Cessation
- 1984-05-10 CH CH2309/84A patent/CH669329A5/de not_active IP Right Cessation
- 1984-05-10 CA CA000453998A patent/CA1222950A/en not_active Expired
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5793065A (en) * | 1980-11-25 | 1982-06-09 | Alza Corp | Permeation apparatus having hydrogel drive member |
Cited By (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6153214A (ja) * | 1983-08-16 | 1986-03-17 | ザ ウエルカム フアウンデ−シヨン リミテツド | 調節された方法による有効成分の放出を可能にする医薬組成物 |
| JPS62185010A (ja) * | 1986-02-07 | 1987-08-13 | アルザ コ−ポレ−シヨン | 生体受容性を強化した薬物送達システム |
| JPH01113316A (ja) * | 1987-10-02 | 1989-05-02 | Alza Corp | 心臓血管系疾病処置用投薬形態 |
| JPH01242528A (ja) * | 1988-03-21 | 1989-09-27 | Alza Corp | 浸透性投薬形態 |
| JPH01313432A (ja) * | 1988-06-02 | 1989-12-18 | Alza Corp | ジルチアゼム投与用投薬形態 |
| JPH05504074A (ja) * | 1989-12-06 | 1993-07-01 | メドトロニック インコーポレーテッド | 比色定量分析による筋肉適合性検出 |
| JPH05506858A (ja) * | 1990-05-07 | 1993-10-07 | アルザ コーポレイション | 抗パーキンソン病剤供給用投与形態 |
| JP2008069177A (ja) * | 1993-05-27 | 2008-03-27 | Alza Corp | 抗鬱薬投薬形態 |
| JP2010248259A (ja) * | 1993-05-27 | 2010-11-04 | Alza Corp | 抗鬱薬投薬形態 |
| JP2012031208A (ja) * | 1993-05-27 | 2012-02-16 | Alza Corp | 抗鬱薬投薬形態 |
| JP2007505894A (ja) * | 2003-09-19 | 2007-03-15 | サン・ファーマシューティカル・インダストリーズ・リミテッド | 経口薬送達システム |
| JP2008525335A (ja) * | 2004-12-24 | 2008-07-17 | バイエル・ヘルスケア・アクチェンゲゼルシャフト | 経口投与できる固体の放出改変型医薬投与形 |
| JP2012528799A (ja) * | 2009-06-02 | 2012-11-15 | ダウ グローバル テクノロジーズ エルエルシー | 徐放製剤 |
| JP2015007144A (ja) * | 2014-10-17 | 2015-01-15 | ダウ グローバル テクノロジーズ エルエルシー | 徐放製剤 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| LAPS | Cancellation because of no payment of annual fees |