JPS5973575A - プロピニルアミノイソオキサゾ−ル誘導体 - Google Patents

プロピニルアミノイソオキサゾ−ル誘導体

Info

Publication number
JPS5973575A
JPS5973575A JP57176762A JP17676282A JPS5973575A JP S5973575 A JPS5973575 A JP S5973575A JP 57176762 A JP57176762 A JP 57176762A JP 17676282 A JP17676282 A JP 17676282A JP S5973575 A JPS5973575 A JP S5973575A
Authority
JP
Japan
Prior art keywords
compound
alkyl
alkylene
hydrogen
propynyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP57176762A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0357900B2 (https=
Inventor
Tokuo Makikado
牧角　徳夫
Akira Murabayashi
村林　旭
Katsuya Tawara
俵　勝也
Yoshiya Watanabe
渡辺　吉八
Toshio Takahashi
俊夫 高橋
Takao Konishi
小西　喬郎
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shionogi and Co Ltd
Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd
Priority to JP57176762A priority Critical patent/JPS5973575A/ja
Priority to US06/530,883 priority patent/US4576956A/en
Priority to EP83201317A priority patent/EP0105548B1/en
Priority to DE8383201317T priority patent/DE3371513D1/de
Priority to ES525886A priority patent/ES525886A0/es
Priority to DK457483A priority patent/DK457483A/da
Priority to KR1019830004703A priority patent/KR880001047B1/ko
Priority to CA000438395A priority patent/CA1206154A/en
Priority to AU19904/83A priority patent/AU563285B2/en
Priority to GB08326637A priority patent/GB2128188B/en
Publication of JPS5973575A publication Critical patent/JPS5973575A/ja
Publication of JPH0357900B2 publication Critical patent/JPH0357900B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/14—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Oncology (AREA)
  • Environmental Sciences (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP57176762A 1982-10-05 1982-10-05 プロピニルアミノイソオキサゾ−ル誘導体 Granted JPS5973575A (ja)

Priority Applications (10)

Application Number Priority Date Filing Date Title
JP57176762A JPS5973575A (ja) 1982-10-05 1982-10-05 プロピニルアミノイソオキサゾ−ル誘導体
US06/530,883 US4576956A (en) 1982-10-05 1983-09-09 Iodo propargylaminoisoxazoles as fungicides
EP83201317A EP0105548B1 (en) 1982-10-05 1983-09-12 Propynylaminoisoxazole derivatives
DE8383201317T DE3371513D1 (de) 1982-10-05 1983-09-12 Propynylaminoisoxazole derivatives
ES525886A ES525886A0 (es) 1982-10-05 1983-09-23 Un procedimiento para preparar derivados de propinilaminoisoxazol
DK457483A DK457483A (da) 1982-10-05 1983-10-04 Antimikrobielle propynylaminoisoxazol derivater
KR1019830004703A KR880001047B1 (ko) 1982-10-05 1983-10-04 프로피닐아미노 이속사졸 유도체의 제조방법
CA000438395A CA1206154A (en) 1982-10-05 1983-10-05 Propynylaminoisoxazole derivatives
AU19904/83A AU563285B2 (en) 1982-10-05 1983-10-05 Propynylaminoisoxazole derivatives
GB08326637A GB2128188B (en) 1982-10-05 1983-10-05 Propynylaminoisoxazole derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP57176762A JPS5973575A (ja) 1982-10-05 1982-10-05 プロピニルアミノイソオキサゾ−ル誘導体

Publications (2)

Publication Number Publication Date
JPS5973575A true JPS5973575A (ja) 1984-04-25
JPH0357900B2 JPH0357900B2 (https=) 1991-09-03

Family

ID=16019362

Family Applications (1)

Application Number Title Priority Date Filing Date
JP57176762A Granted JPS5973575A (ja) 1982-10-05 1982-10-05 プロピニルアミノイソオキサゾ−ル誘導体

Country Status (10)

Country Link
US (1) US4576956A (https=)
EP (1) EP0105548B1 (https=)
JP (1) JPS5973575A (https=)
KR (1) KR880001047B1 (https=)
AU (1) AU563285B2 (https=)
CA (1) CA1206154A (https=)
DE (1) DE3371513D1 (https=)
DK (1) DK457483A (https=)
ES (1) ES525886A0 (https=)
GB (1) GB2128188B (https=)

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007052615A1 (ja) * 2005-10-31 2007-05-10 Eisai R & D Management Co., Ltd. ヘテロ環置換ピリジン誘導体およびそれらを含有する抗真菌剤
WO2008136279A1 (ja) * 2007-04-27 2008-11-13 Eisai R & D Management Co., Ltd. ヘテロ環置換ピリジン誘導体の塩またはその結晶
US7691882B2 (en) 2005-10-31 2010-04-06 Eisai R&D Management Co., Ltd. Heterocycles substituted pyridine derivatives and antifungal agent containing thereof
US7829585B2 (en) 2005-03-30 2010-11-09 Eisai R&D Management Co., Ltd. Antifungal agent containing pyridine derivative
US7932272B2 (en) 2003-09-30 2011-04-26 Eisai R&D Management Co., Ltd. Antifungal agent containing heterocyclic compound
US8183264B2 (en) 2006-09-21 2012-05-22 Eisai R&D Managment Co., Ltd. Pyridine derivative substituted by heteroaryl ring, and antifungal agent comprising the same
US8188119B2 (en) 2008-10-24 2012-05-29 Eisai R&D Management Co., Ltd Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same
US8507530B2 (en) 2007-04-27 2013-08-13 Eisai R&D Management Co., Ltd. Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same
US8513287B2 (en) 2007-12-27 2013-08-20 Eisai R&D Management Co., Ltd. Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60142987A (ja) * 1983-12-29 1985-07-29 Mochida Pharmaceut Co Ltd セフアロスポリン誘導体
DE3485860T2 (de) * 1983-12-29 1993-01-14 Mochida Pharm Co Ltd Cephalosporinverbindungen, verfahren zu ihrer herstellung und pharmazeutishe praeparate.
US4840945A (en) * 1985-04-01 1989-06-20 Mochida Pharmaceutical Co., Ltd. Cephalosporin derivatives
US4880798A (en) * 1986-11-25 1989-11-14 Mochida Pharmaceutical Co., Ltd. Cephalosporin derivatives
JPS63132893A (ja) * 1986-11-25 1988-06-04 Mochida Pharmaceut Co Ltd 新規セフアロスポリン誘導体、その製法およびそれらを有効成分とする抗菌剤
DE4328425A1 (de) * 1993-08-24 1995-03-02 Basf Ag Acylamino-substituierte Isoxazol- bzw. Isothiazolderivate, Verfahren zu deren Herstellung und ihre Verwendung
GB2368012A (en) * 2000-10-19 2002-04-24 Nicholas John Larkins Preparation for the relief of inflammatory disease
DE10256186A1 (de) * 2002-12-02 2004-06-09 Bayer Ag Cyclopenta(c)isoxazol-3-amine als Materialschutzmittel
GB2420302B (en) * 2003-09-30 2007-03-07 Advanced Micro Devices Inc A method and system for controlling the chemical mechanical polishing by using a sensor signal of a pad conditioner
US20050241110A1 (en) * 2004-04-09 2005-11-03 Bruce Baker Ergonomic handles, especially for garden tools
US20090227799A1 (en) * 2004-08-09 2009-09-10 Kazutaka Nakamoto Novel Antimalarial Agent Containing Heterocyclic Compound
CN101300250B (zh) * 2005-10-31 2012-09-05 卫材R&D管理有限公司 杂环取代吡啶衍生物及含有该衍生物的抗真菌剂

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH419716A (de) * 1963-03-29 1966-08-31 Geigy Ag J R Mittel zur Bekämpfung von pflanzenparasitären Nematoden und Verfahren zur Herstellung dieses Mittels
US3544582A (en) * 1965-04-06 1970-12-01 Hoffmann La Roche Process for preparing aminoisoxazoles
BE792338A (fr) * 1971-12-07 1973-06-06 Ciba Geigy Phenyl-formamidines et produits pesticides qui en contiennent
JPS5379862A (en) * 1976-12-24 1978-07-14 Dainippon Pharmaceut Co Ltd Iodepropargyl ethers
JPS5422365A (en) * 1977-07-20 1979-02-20 Sankyo Co Ltd Isoxazole derivative, and antiseptic and sntifugal agnets for wood meterials comprising the derivativs as active constituent
GB1590870A (en) * 1978-05-31 1981-06-10 Shionogi & Co N-(5-t-butyl-3-isoxazolyl) alkanamide derivatives having herbicidal activity
DE3167599D1 (en) * 1980-07-16 1985-01-17 Bayer Ag Use of 2-propargyloxy-benzazoles as synergists
JPS5815965A (ja) * 1981-07-23 1983-01-29 Nippon Tokushu Noyaku Seizo Kk ベンゾイソチアゾ−ル誘導体並びにその塩酸塩、その製法、及び農業用殺菌剤

Cited By (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7932272B2 (en) 2003-09-30 2011-04-26 Eisai R&D Management Co., Ltd. Antifungal agent containing heterocyclic compound
US7829585B2 (en) 2005-03-30 2010-11-09 Eisai R&D Management Co., Ltd. Antifungal agent containing pyridine derivative
US8158657B2 (en) 2005-10-31 2012-04-17 Eisai R&D Management Co., Ltd. Heterocycles substituted pyridine derivatives and antifungal agent containing thereof
US8841327B2 (en) 2005-10-31 2014-09-23 Eisai R&D Management Co., Ltd. Heterocycles substituted pyridine derivatives and antifungal agent containing thereof
US7691882B2 (en) 2005-10-31 2010-04-06 Eisai R&D Management Co., Ltd. Heterocycles substituted pyridine derivatives and antifungal agent containing thereof
WO2007052615A1 (ja) * 2005-10-31 2007-05-10 Eisai R & D Management Co., Ltd. ヘテロ環置換ピリジン誘導体およびそれらを含有する抗真菌剤
US8153662B2 (en) 2005-10-31 2012-04-10 Eisai R&D Management Co., Ltd. Heterocycles substituted pyridine derivatives and antifungal agent containing thereof
US8183264B2 (en) 2006-09-21 2012-05-22 Eisai R&D Managment Co., Ltd. Pyridine derivative substituted by heteroaryl ring, and antifungal agent comprising the same
JPWO2008136279A1 (ja) * 2007-04-27 2010-07-29 エーザイ・アール・アンド・ディー・マネジメント株式会社 ヘテロ環置換ピリジン誘導体の塩またはその結晶
US8058444B2 (en) 2007-04-27 2011-11-15 Eisai R&D Management Co., Ltd. Heterocycle-substituted pyridine derivative's salt or crystal thereof
US8507530B2 (en) 2007-04-27 2013-08-13 Eisai R&D Management Co., Ltd. Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same
WO2008136279A1 (ja) * 2007-04-27 2008-11-13 Eisai R & D Management Co., Ltd. ヘテロ環置換ピリジン誘導体の塩またはその結晶
US8513287B2 (en) 2007-12-27 2013-08-20 Eisai R&D Management Co., Ltd. Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same
US8188119B2 (en) 2008-10-24 2012-05-29 Eisai R&D Management Co., Ltd Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same

Also Published As

Publication number Publication date
CA1206154A (en) 1986-06-17
GB2128188B (en) 1986-05-08
KR840006341A (ko) 1984-11-29
DE3371513D1 (de) 1987-06-19
ES8503344A1 (es) 1985-02-16
DK457483A (da) 1984-04-06
EP0105548A1 (en) 1984-04-18
US4576956A (en) 1986-03-18
EP0105548B1 (en) 1987-05-13
AU1990483A (en) 1984-04-12
GB8326637D0 (en) 1983-11-09
DK457483D0 (da) 1983-10-04
AU563285B2 (en) 1987-07-02
ES525886A0 (es) 1985-02-16
JPH0357900B2 (https=) 1991-09-03
GB2128188A (en) 1984-04-26
KR880001047B1 (ko) 1988-06-18

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