JPS58128396A - ダウノルビシンおよびドキソルビシン同族体 - Google Patents

ダウノルビシンおよびドキソルビシン同族体

Info

Publication number
JPS58128396A
JPS58128396A JP58005974A JP597483A JPS58128396A JP S58128396 A JPS58128396 A JP S58128396A JP 58005974 A JP58005974 A JP 58005974A JP 597483 A JP597483 A JP 597483A JP S58128396 A JPS58128396 A JP S58128396A
Authority
JP
Japan
Prior art keywords
demethoxy
methyl
daunorubicin
compound according
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP58005974A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6328436B2 (fr
Inventor
セルジオ・ペンコ
ジユリア−ノ・フランキ
フエデリコ・アルカモ−ネ
アンナ・マリア・カサツザ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Carlo Erba SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Carlo Erba SpA filed Critical Carlo Erba SpA
Publication of JPS58128396A publication Critical patent/JPS58128396A/ja
Publication of JPS6328436B2 publication Critical patent/JPS6328436B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
JP58005974A 1982-01-26 1983-01-19 ダウノルビシンおよびドキソルビシン同族体 Granted JPS58128396A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8202080 1982-01-26
GB8202080 1982-01-26

Publications (2)

Publication Number Publication Date
JPS58128396A true JPS58128396A (ja) 1983-07-30
JPS6328436B2 JPS6328436B2 (fr) 1988-06-08

Family

ID=10527864

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58005974A Granted JPS58128396A (ja) 1982-01-26 1983-01-19 ダウノルビシンおよびドキソルビシン同族体

Country Status (28)

Country Link
JP (1) JPS58128396A (fr)
KR (1) KR900006214B1 (fr)
AT (1) AT378776B (fr)
AU (1) AU551700B2 (fr)
BE (1) BE895687A (fr)
CA (1) CA1197237A (fr)
CH (1) CH657622A5 (fr)
CS (1) CS235979B2 (fr)
DE (1) DE3301489A1 (fr)
DK (1) DK157322C (fr)
ES (1) ES8403140A1 (fr)
FI (1) FI74977C (fr)
FR (1) FR2520365B1 (fr)
GB (1) GB2116169B (fr)
GR (1) GR77890B (fr)
HU (1) HU192784B (fr)
IE (1) IE53750B1 (fr)
IL (1) IL67709A (fr)
IT (1) IT1210482B (fr)
NL (1) NL8300150A (fr)
NO (1) NO153456C (fr)
NZ (1) NZ203047A (fr)
PH (1) PH19130A (fr)
PT (1) PT76113A (fr)
SE (1) SE461591B (fr)
SU (1) SU1187724A3 (fr)
YU (1) YU43536B (fr)
ZA (1) ZA83450B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2182926B (en) * 1985-11-19 1989-10-04 Erba Farmitalia Nitro anthracyclines, process for their preparation and use thereof
GB8708927D0 (en) * 1987-04-14 1987-05-20 Erba Farmitalia Chiral synthesis of anthracyclines

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1509875A (en) * 1976-06-14 1978-05-04 Farmaceutici Italia Optically active anthracyclinones and anthracycline glycosides
GB1573037A (en) * 1977-05-05 1980-08-13 Farmaceutici Italia Anthracyclines
ATE4387T1 (de) * 1979-07-04 1983-08-15 Farmitalia Carlo Erba S.P.A. Anthracyclin-glycoside, verfahren zu ihrer herstellung und sie enthaltende therapeutische zusammensetzung.
DE3100968A1 (de) * 1980-01-16 1982-01-14 Farmitalia Carlo Erba S.p.A., 20159 Milano Anthracyclinderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
GB8301178D0 (en) 1983-02-16
CS235979B2 (en) 1985-05-15
ATA15683A (de) 1985-02-15
NL8300150A (nl) 1983-08-16
KR840003262A (ko) 1984-08-20
FI74977B (fi) 1987-12-31
IE53750B1 (en) 1989-02-01
FI830155L (fi) 1983-07-27
ZA83450B (en) 1983-10-26
DK157322B (da) 1989-12-11
DE3301489A1 (de) 1983-08-04
DK157322C (da) 1990-05-07
PT76113A (en) 1983-02-01
NO153456B (no) 1985-12-16
FR2520365A1 (fr) 1983-07-29
AU551700B2 (en) 1986-05-08
ES519255A0 (es) 1984-03-01
IE830144L (en) 1983-07-26
ES8403140A1 (es) 1984-03-01
NO830234L (no) 1983-07-27
KR900006214B1 (ko) 1990-08-25
SU1187724A3 (ru) 1985-10-23
CH657622A5 (it) 1986-09-15
SE8300324L (sv) 1983-07-27
IL67709A (en) 1986-03-31
FI74977C (fi) 1988-04-11
HU192784B (en) 1987-07-28
GB2116169A (en) 1983-09-21
FI830155A0 (fi) 1983-01-17
PH19130A (en) 1986-01-08
SE461591B (sv) 1990-03-05
DK27683D0 (da) 1983-01-25
BE895687A (fr) 1983-05-16
NO153456C (no) 1986-03-26
IL67709A0 (en) 1983-05-15
GR77890B (fr) 1984-09-25
GB2116169B (en) 1985-09-04
IT1210482B (it) 1989-09-14
YU43536B (en) 1989-08-31
NZ203047A (en) 1985-10-11
YU8983A (en) 1986-02-28
AU1052583A (en) 1983-08-04
CA1197237A (fr) 1985-11-26
AT378776B (de) 1985-09-25
JPS6328436B2 (fr) 1988-06-08
FR2520365B1 (fr) 1985-07-12
SE8300324D0 (sv) 1983-01-21
DK27683A (da) 1983-07-27
DE3301489C2 (fr) 1988-01-28
IT8319147A0 (it) 1983-01-18

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