JPH0237354B2 - - Google Patents

Info

Publication number
JPH0237354B2
JPH0237354B2 JP56086312A JP8631281A JPH0237354B2 JP H0237354 B2 JPH0237354 B2 JP H0237354B2 JP 56086312 A JP56086312 A JP 56086312A JP 8631281 A JP8631281 A JP 8631281A JP H0237354 B2 JPH0237354 B2 JP H0237354B2
Authority
JP
Japan
Prior art keywords
chain
formula
general formula
aryl
oxazolidinones
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP56086312A
Other languages
English (en)
Japanese (ja)
Other versions
JPS5753473A (en
Inventor
Ansha Jannfuransowa
Buurujerii Gii
Dosuteru Fuiritsupu
Dozon Koretsuto
Gyare Patoritsuku
Rakuuru Aran
Rangurowa Mitsusheru
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8012423A external-priority patent/FR2458547B2/fr
Application filed by Delalande SA filed Critical Delalande SA
Publication of JPS5753473A publication Critical patent/JPS5753473A/ja
Publication of JPH0237354B2 publication Critical patent/JPH0237354B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/45—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by at least one doubly—bound oxygen atom, not being part of a —CHO group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP56086312A 1980-06-04 1981-06-04 Novel n-aryl-2-oxazolidinones, manufacture and drug containing them Granted JPS5753473A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8012423A FR2458547B2 (fr) 1978-06-09 1980-06-04 Nouvelles n-aryle azolones, leur procede de preparation et leur application en therapeutique

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013793A Division JPH03197470A (ja) 1980-06-04 1990-01-25 新規なｎ―アリール―２―オキサゾリジノン化合物

Publications (2)

Publication Number Publication Date
JPS5753473A JPS5753473A (en) 1982-03-30
JPH0237354B2 true JPH0237354B2 (enExample) 1990-08-23

Family

ID=9242708

Family Applications (2)

Application Number Title Priority Date Filing Date
JP56086312A Granted JPS5753473A (en) 1980-06-04 1981-06-04 Novel n-aryl-2-oxazolidinones, manufacture and drug containing them
JP2013793A Granted JPH03197470A (ja) 1980-06-04 1990-01-25 新規なｎ―アリール―２―オキサゾリジノン化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2013793A Granted JPH03197470A (ja) 1980-06-04 1990-01-25 新規なｎ―アリール―２―オキサゾリジノン化合物

Country Status (14)

Country Link
US (1) US4517197A (enExample)
JP (2) JPS5753473A (enExample)
AU (1) AU544542B2 (enExample)
BE (1) BE889091R (enExample)
CA (1) CA1171865A (enExample)
CH (1) CH650780A5 (enExample)
DE (1) DE3122291A1 (enExample)
ES (1) ES502546A0 (enExample)
GB (1) GB2076813B (enExample)
GR (1) GR75662B (enExample)
LU (1) LU83400A1 (enExample)
NL (1) NL8102715A (enExample)
SE (1) SE457259B (enExample)
ZA (1) ZA813567B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0498123A (ja) * 1990-08-16 1992-03-30 Hikoshima Seiren Kk 汚泥界面の検出方法及びその装置

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4348393A (en) * 1978-06-09 1982-09-07 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
FR2506769A2 (fr) * 1978-06-09 1982-12-03 Delalande Sa Para-((cyano-5 n pentyl-1) phenyl)-3 methoxymethyl-5 oxazolidinone-2, son procede de preparation et ses applications en therapeutique
FR2500450A1 (fr) * 1981-02-25 1982-08-27 Delalande Sa Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique
JPS58169602U (ja) * 1982-04-13 1983-11-12 出井　惣一 光飾機構に用いる携帯光源用電源構造
US4705799A (en) * 1983-06-07 1987-11-10 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents
CA1302422C (en) * 1986-09-03 1992-06-02 Margherita Strolin-Benedetti 5-aminoethyloxazolidin-2-one derivatives, process for the preparation thereofand their therapeutic use
US5032605A (en) * 1987-10-09 1991-07-16 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US5036092A (en) * 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US4985429A (en) * 1987-10-09 1991-01-15 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4965268A (en) * 1987-10-09 1990-10-23 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
FR2653017B1 (fr) * 1989-10-17 1995-05-05 Delalande Sa Derives d'aryl-3 oxazolidinone-2, leur procede de preparation et leur application en therapeutique.
US5235063A (en) * 1989-10-17 1993-08-10 Delalande S.A. Process of preparing by condensation certain
US5182296A (en) * 1989-10-26 1993-01-26 Tanabe Seiyaky Co., Ltd. Naphthyloxazolidone derivatives
FR2675504B1 (fr) * 1991-04-16 1995-01-27 Delalande Sa Derives d'aryl-3 oxazolidinone, leur procede de preparation et leur application en therapeutique.
JP2669579B2 (ja) * 1991-10-23 1997-10-29 エーザイ株式会社 オキサゾリドン誘導体
RU2117668C1 (ru) * 1991-10-23 1998-08-20 Эйсаи Ко., Лтд. Производное оксазолидона или его фармакологически приемлемые соли, фармацевтическая композиция, способ лечения
TW286317B (enExample) * 1993-12-13 1996-09-21 Hoffmann La Roche
FR2741072B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives d'oxazolidin-2-one, leur preparation et leur application en therapeutique
FR2741071B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives de 3-(benzofuran-5-yl)oxazolidin-2-one, leur preparation et leur application en therapeutique

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1180089A (en) * 1967-10-20 1970-02-04 Delalande Sa Acetylenic Derivatives of 2-Oxazolidinones and processes of preparation
GB1250538A (enExample) * 1969-03-18 1971-10-20
FR2356422A1 (fr) * 1976-03-01 1978-01-27 Delalande Sa Nouveaux hydroxymethyl-5 oxazolidinone-2, leur procede de preparation et leur application en therapeutique
LU80081A1 (fr) * 1977-08-26 1979-05-15 Delalande Sa Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique
US4348393A (en) * 1978-06-09 1982-09-07 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0498123A (ja) * 1990-08-16 1992-03-30 Hikoshima Seiren Kk 汚泥界面の検出方法及びその装置

Also Published As

Publication number Publication date
ZA813567B (en) 1982-06-30
GB2076813B (en) 1984-08-30
BE889091R (fr) 1981-12-04
AU7131981A (en) 1981-12-10
CA1171865A (en) 1984-07-31
NL8102715A (nl) 1982-01-04
ES8203356A1 (es) 1982-04-01
US4517197A (en) 1985-05-14
AU544542B2 (en) 1985-06-06
JPS5753473A (en) 1982-03-30
GB2076813A (en) 1981-12-09
JPH044311B2 (enExample) 1992-01-27
LU83400A1 (fr) 1983-04-06
GR75662B (enExample) 1984-08-02
SE457259B (sv) 1988-12-12
SE8103307L (sv) 1981-12-05
CH650780A5 (fr) 1985-08-15
ES502546A0 (es) 1982-04-01
JPH03197470A (ja) 1991-08-28
DE3122291A1 (de) 1982-05-13

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