ES8203356A1 - Procedimiento para la preparacion de nuevas n-ariloxazolidi-nonas-2 - Google Patents
Procedimiento para la preparacion de nuevas n-ariloxazolidi-nonas-2Info
- Publication number
- ES8203356A1 ES8203356A1 ES502546A ES502546A ES8203356A1 ES 8203356 A1 ES8203356 A1 ES 8203356A1 ES 502546 A ES502546 A ES 502546A ES 502546 A ES502546 A ES 502546A ES 8203356 A1 ES8203356 A1 ES 8203356A1
- Authority
- ES
- Spain
- Prior art keywords
- oxazolidinones
- methoxymethyl
- pharmaceutical compositions
- substituted phenyl
- compositions containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- IJDJONDNDCLDOA-UHFFFAOYSA-N 5-(methoxymethyl)-3-phenyl-1,3-oxazolidin-2-one Chemical class O=C1OC(COC)CN1C1=CC=CC=C1 IJDJONDNDCLDOA-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/45—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by at least one doubly—bound oxygen atom, not being part of a —CHO group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Psychiatry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
PROCEDIMIENTO DE OBTENCION DE N-ARILOXAZOLIDINONAS-2. CONSISTE EN HIDROLIZAR EN MEDIO ACIDO EL COMPUESTO DE FORMULA GENERAL (I). SE OBTIENE EL COMPUESTO (II), EN QUE R REPRESENTA UN ENCADENAMIENTO (ACETIL-2) ETOLOXI; UN ENCADENAMIENTO (CIANO-5)N -PENTILO; EL NUCLEO P-CLOROFENILO O M-CIANOFENILO EL ENCAENAMIENTO (CICLOHEXIL-2) ETILINO O BIEN EL GRUPO (III).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8012423A FR2458547B2 (fr) | 1978-06-09 | 1980-06-04 | Nouvelles n-aryle azolones, leur procede de preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
ES502546A0 ES502546A0 (es) | 1982-04-01 |
ES8203356A1 true ES8203356A1 (es) | 1982-04-01 |
Family
ID=9242708
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES502546A Expired ES8203356A1 (es) | 1980-06-04 | 1981-05-27 | Procedimiento para la preparacion de nuevas n-ariloxazolidi-nonas-2 |
Country Status (14)
Country | Link |
---|---|
US (1) | US4517197A (es) |
JP (2) | JPS5753473A (es) |
AU (1) | AU544542B2 (es) |
BE (1) | BE889091R (es) |
CA (1) | CA1171865A (es) |
CH (1) | CH650780A5 (es) |
DE (1) | DE3122291A1 (es) |
ES (1) | ES8203356A1 (es) |
GB (1) | GB2076813B (es) |
GR (1) | GR75662B (es) |
LU (1) | LU83400A1 (es) |
NL (1) | NL8102715A (es) |
SE (1) | SE457259B (es) |
ZA (1) | ZA813567B (es) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4348393A (en) * | 1978-06-09 | 1982-09-07 | Delalande S.A. | N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones |
FR2506769A2 (fr) * | 1978-06-09 | 1982-12-03 | Delalande Sa | Para-((cyano-5 n pentyl-1) phenyl)-3 methoxymethyl-5 oxazolidinone-2, son procede de preparation et ses applications en therapeutique |
FR2500450A1 (fr) * | 1981-02-25 | 1982-08-27 | Delalande Sa | Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique |
JPS58169602U (ja) * | 1982-04-13 | 1983-11-12 | 出井 惣一 | 光飾機構に用いる携帯光源用電源構造 |
US4705799A (en) * | 1983-06-07 | 1987-11-10 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents |
AU7778087A (en) * | 1986-09-03 | 1988-04-14 | Delalande S.A. | 5-aminoethyloxazolidin-2-one derivatives |
US4985429A (en) * | 1987-10-09 | 1991-01-15 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
US5032605A (en) * | 1987-10-09 | 1991-07-16 | Du Pont Merck Pharmaceutical Company | Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents |
US4801600A (en) * | 1987-10-09 | 1989-01-31 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
US4965268A (en) * | 1987-10-09 | 1990-10-23 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents |
US5036092A (en) * | 1987-10-09 | 1991-07-30 | Du Pont Merck Pharmaceutical | Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents |
US5235063A (en) * | 1989-10-17 | 1993-08-10 | Delalande S.A. | Process of preparing by condensation certain |
FR2653017B1 (fr) * | 1989-10-17 | 1995-05-05 | Delalande Sa | Derives d'aryl-3 oxazolidinone-2, leur procede de preparation et leur application en therapeutique. |
US5182296A (en) * | 1989-10-26 | 1993-01-26 | Tanabe Seiyaky Co., Ltd. | Naphthyloxazolidone derivatives |
JPH0498123A (ja) * | 1990-08-16 | 1992-03-30 | Hikoshima Seiren Kk | 汚泥界面の検出方法及びその装置 |
FR2675504B1 (fr) * | 1991-04-16 | 1995-01-27 | Delalande Sa | Derives d'aryl-3 oxazolidinone, leur procede de preparation et leur application en therapeutique. |
JP2669579B2 (ja) * | 1991-10-23 | 1997-10-29 | エーザイ株式会社 | オキサゾリドン誘導体 |
TW286317B (es) * | 1993-12-13 | 1996-09-21 | Hoffmann La Roche | |
FR2741072B1 (fr) * | 1995-11-09 | 1997-12-12 | Synthelabo | Derives d'oxazolidin-2-one, leur preparation et leur application en therapeutique |
FR2741071B1 (fr) * | 1995-11-09 | 1997-12-12 | Synthelabo | Derives de 3-(benzofuran-5-yl)oxazolidin-2-one, leur preparation et leur application en therapeutique |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1180089A (en) * | 1967-10-20 | 1970-02-04 | Delalande Sa | Acetylenic Derivatives of 2-Oxazolidinones and processes of preparation |
GB1252101A (es) * | 1969-03-18 | 1971-11-03 | ||
FR2356422A1 (fr) * | 1976-03-01 | 1978-01-27 | Delalande Sa | Nouveaux hydroxymethyl-5 oxazolidinone-2, leur procede de preparation et leur application en therapeutique |
LU80081A1 (fr) * | 1977-08-26 | 1979-05-15 | Delalande Sa | Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique |
US4348393A (en) * | 1978-06-09 | 1982-09-07 | Delalande S.A. | N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones |
-
1981
- 1981-05-20 CA CA000377905A patent/CA1171865A/en not_active Expired
- 1981-05-21 GB GB8115597A patent/GB2076813B/en not_active Expired
- 1981-05-25 CH CH3393/81A patent/CH650780A5/fr not_active IP Right Cessation
- 1981-05-26 SE SE8103307A patent/SE457259B/sv not_active IP Right Cessation
- 1981-05-27 ES ES502546A patent/ES8203356A1/es not_active Expired
- 1981-05-27 ZA ZA00813567A patent/ZA813567B/xx unknown
- 1981-05-29 GR GR65106A patent/GR75662B/el unknown
- 1981-06-01 LU LU83400A patent/LU83400A1/fr unknown
- 1981-06-03 AU AU71319/81A patent/AU544542B2/en not_active Ceased
- 1981-06-04 NL NL8102715A patent/NL8102715A/nl not_active Application Discontinuation
- 1981-06-04 BE BE0/204995A patent/BE889091R/fr not_active IP Right Cessation
- 1981-06-04 DE DE19813122291 patent/DE3122291A1/de not_active Ceased
- 1981-06-04 JP JP56086312A patent/JPS5753473A/ja active Granted
-
1983
- 1983-07-29 US US06/518,320 patent/US4517197A/en not_active Expired - Fee Related
-
1990
- 1990-01-25 JP JP2013793A patent/JPH03197470A/ja active Granted
Also Published As
Publication number | Publication date |
---|---|
SE457259B (sv) | 1988-12-12 |
ZA813567B (en) | 1982-06-30 |
JPS5753473A (en) | 1982-03-30 |
AU544542B2 (en) | 1985-06-06 |
GB2076813B (en) | 1984-08-30 |
BE889091R (fr) | 1981-12-04 |
LU83400A1 (fr) | 1983-04-06 |
SE8103307L (sv) | 1981-12-05 |
ES502546A0 (es) | 1982-04-01 |
GB2076813A (en) | 1981-12-09 |
DE3122291A1 (de) | 1982-05-13 |
GR75662B (es) | 1984-08-02 |
CH650780A5 (fr) | 1985-08-15 |
NL8102715A (nl) | 1982-01-04 |
CA1171865A (en) | 1984-07-31 |
US4517197A (en) | 1985-05-14 |
JPH044311B2 (es) | 1992-01-27 |
JPH03197470A (ja) | 1991-08-28 |
AU7131981A (en) | 1981-12-10 |
JPH0237354B2 (es) | 1990-08-23 |
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