JPH0213645B2 - - Google Patents

Info

Publication number
JPH0213645B2
JPH0213645B2 JP58065160A JP6516083A JPH0213645B2 JP H0213645 B2 JPH0213645 B2 JP H0213645B2 JP 58065160 A JP58065160 A JP 58065160A JP 6516083 A JP6516083 A JP 6516083A JP H0213645 B2 JPH0213645 B2 JP H0213645B2
Authority
JP
Japan
Prior art keywords
acid
salt
mbp
value
biphosphonic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP58065160A
Other languages
English (en)
Japanese (ja)
Other versions
JPS58189193A (ja
Inventor
Rotsushiini Serujio
Sutaibaano Jorujo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ISUCHI JENCHIRI SpA
Original Assignee
ISUCHI JENCHIRI SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11171970&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JPH0213645(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by ISUCHI JENCHIRI SpA filed Critical ISUCHI JENCHIRI SpA
Publication of JPS58189193A publication Critical patent/JPS58189193A/ja
Publication of JPH0213645B2 publication Critical patent/JPH0213645B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3839—Polyphosphonic acids
    • C07F9/3873—Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3839—Polyphosphonic acids
    • C07F9/3856—Polyphosphonic acids containing halogen or nitro(so) substituents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP58065160A 1982-04-15 1983-04-13 薬理活性を有するバイホスホネートを有効成分とする医薬 Granted JPS58189193A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT20781A/82 1982-04-15
IT8220781A IT1201087B (it) 1982-04-15 1982-04-15 Bifosfonati farmacologicamente attivi,procedimento per la loro preparazione e relative composizioni farmaceutiche

Publications (2)

Publication Number Publication Date
JPS58189193A JPS58189193A (ja) 1983-11-04
JPH0213645B2 true JPH0213645B2 (OSRAM) 1990-04-04

Family

ID=11171970

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58065160A Granted JPS58189193A (ja) 1982-04-15 1983-04-13 薬理活性を有するバイホスホネートを有効成分とする医薬

Country Status (12)

Country Link
US (1) US4621077A (OSRAM)
JP (1) JPS58189193A (OSRAM)
BE (1) BE896453A (OSRAM)
CH (1) CH661437A5 (OSRAM)
FR (1) FR2525223B1 (OSRAM)
GB (1) GB2118042B (OSRAM)
HK (1) HK79390A (OSRAM)
IT (1) IT1201087B (OSRAM)
LU (2) LU84746A1 (OSRAM)
MX (1) MX9203428A (OSRAM)
NL (5) NL192562C (OSRAM)
SE (1) SE463239B (OSRAM)

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DE3623397A1 (de) * 1986-07-11 1988-01-14 Boehringer Mannheim Gmbh Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel
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US4621077A (en) 1986-11-04
NL970038I1 (nl) 1998-01-05
GB8308791D0 (en) 1983-05-11
BE896453A (fr) 1983-08-01
CH661437A5 (it) 1987-07-31
LU88714I2 (fr) 1996-08-23
SE8302130L (sv) 1983-10-16
MX9203428A (es) 1992-07-01
IT8220781A0 (it) 1982-04-15
SE463239B (sv) 1990-10-29
LU84746A1 (fr) 1983-11-17
SE8302130D0 (sv) 1983-04-15
IT1201087B (it) 1989-01-27
GB2118042A (en) 1983-10-26
GB2118042B (en) 1986-01-15
NL192562B (nl) 1997-06-02
NL980010I1 (nl) 1998-05-06
NL8301324A (nl) 1983-11-01
NL980004I1 (nl) 1998-04-01
NL980005I1 (nl) 1998-04-01
NL970038I2 (nl) 2000-11-01
JPS58189193A (ja) 1983-11-04
FR2525223A1 (fr) 1983-10-21
NL192562C (nl) 1997-10-03
HK79390A (en) 1990-10-12
FR2525223B1 (fr) 1986-04-25

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