JP7129704B2 - ２－［３－［４－アミノ－３－（２－フルオロ－４－フェノキシ－フェニル）ピラゾロ［３，４－ｄ］ピリミジン－１－イル］ピペリジン－１－カルボニル］－４－メチル－４－［４－（オキセタン－３－イル）ピペラジン－１－イル］ペント－２－エネニトリルの放出調節製剤 - Google Patents

２－［３－［４－アミノ－３－（２－フルオロ－４－フェノキシ－フェニル）ピラゾロ［３，４－ｄ］ピリミジン－１－イル］ピペリジン－１－カルボニル］－４－メチル－４－［４－（オキセタン－３－イル）ピペラジン－１－イル］ペント－２－エネニトリルの放出調節製剤 Download PDF

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JP7129704B2
JP7129704B2 JP2018568426A JP2018568426A JP7129704B2 JP 7129704 B2 JP7129704 B2 JP 7129704B2 JP 2018568426 A JP2018568426 A JP 2018568426A JP 2018568426 A JP2018568426 A JP 2018568426A JP 7129704 B2 JP7129704 B2 JP 7129704B2
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ジェイ． フェルドース，アブ
アール． マゼジザデー，モハマド
リン，ウー
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プリンシピア バイオファーマ インコーポレイテッド
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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JP2018568426A 2016-06-29 2017-06-29 ２－［３－［４－アミノ－３－（２－フルオロ－４－フェノキシ－フェニル）ピラゾロ［３，４－ｄ］ピリミジン－１－イル］ピペリジン－１－カルボニル］－４－メチル－４－［４－（オキセタン－３－イル）ピペラジン－１－イル］ペント－２－エネニトリルの放出調節製剤 Active JP7129704B2 (ja)

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Application Number Priority Date Filing Date Title
US201662356345P 2016-06-29 2016-06-29
US62/356,345 2016-06-29
PCT/US2017/040075 WO2018005849A1 (en) 2016-06-29 2017-06-29 Modified release formulations of 2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile

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JP2019519581A JP2019519581A (ja) 2019-07-11
JP2019519581A5 JP2019519581A5 (enExample) 2020-08-13
JP7129704B2 true JP7129704B2 (ja) 2022-09-02

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US (3) US20190231784A1 (enExample)
EP (1) EP3478273A1 (enExample)
JP (1) JP7129704B2 (enExample)
KR (2) KR102391693B1 (enExample)
CN (2) CN109600989B (enExample)
AU (2) AU2017290354C1 (enExample)
CA (1) CA3028169C (enExample)
EA (1) EA201892836A1 (enExample)
IL (2) IL293621B2 (enExample)
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TW202214250A (zh) * 2020-08-10 2022-04-16 大陸商江蘇恆瑞醫藥股份有限公司 Ｂｔｋ抑制劑治療疾病的用途
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IL293621A (en) 2022-08-01
CN115054586B (zh) 2024-08-02
CA3028169A1 (en) 2018-01-04
IL293621B2 (en) 2023-09-01
US20240207275A1 (en) 2024-06-27
AU2017290354A1 (en) 2019-01-24
US20190231784A1 (en) 2019-08-01
EP3478273A1 (en) 2019-05-08
KR20190025947A (ko) 2019-03-12
IL263815A (en) 2019-01-31
IL293621B1 (en) 2023-05-01
JP2019519581A (ja) 2019-07-11
US12336999B2 (en) 2025-06-24
AU2017290354B8 (en) 2023-01-12
WO2018005849A1 (en) 2018-01-04
KR102391693B1 (ko) 2022-04-29
MX2022002952A (es) 2022-04-06

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