JP6843114B2 - ムスカリン作動薬 - Google Patents

ムスカリン作動薬 Download PDF

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Publication number
JP6843114B2
JP6843114B2 JP2018504992A JP2018504992A JP6843114B2 JP 6843114 B2 JP6843114 B2 JP 6843114B2 JP 2018504992 A JP2018504992 A JP 2018504992A JP 2018504992 A JP2018504992 A JP 2018504992A JP 6843114 B2 JP6843114 B2 JP 6843114B2
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Japan
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group
formula
compound according
salt
hydrogen
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Japanese (ja)
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JP2018522033A5 (enExample
JP2018522033A (ja
Inventor
ブラウン，ジャイルズ・アルバート
キャンズフィールド，ジュリー
ピックワース，マーク
テハン，ベンジャミン・ジェラルド
テオボールド，バリー・ジョン
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Nxera Pharma UK Ltd
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Heptares Therapeutics Ltd
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Publication of JP2018522033A5 publication Critical patent/JP2018522033A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2018504992A 2015-08-03 2016-08-03 ムスカリン作動薬 Active JP6843114B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB1513743.3 2015-08-03
GBGB1513743.3A GB201513743D0 (en) 2015-08-03 2015-08-03 Muscarinic agonists
PCT/GB2016/052385 WO2017021729A1 (en) 2015-08-03 2016-08-03 Muscarinic agonists

Publications (3)

Publication Number Publication Date
JP2018522033A JP2018522033A (ja) 2018-08-09
JP2018522033A5 JP2018522033A5 (enExample) 2019-09-12
JP6843114B2 true JP6843114B2 (ja) 2021-03-17

Family

ID=54063149

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018504992A Active JP6843114B2 (ja) 2015-08-03 2016-08-03 ムスカリン作動薬

Country Status (10)

Country Link
US (3) US10738029B2 (enExample)
EP (1) EP3331529B1 (enExample)
JP (1) JP6843114B2 (enExample)
CN (1) CN108025004B (enExample)
AU (1) AU2016304387B2 (enExample)
CA (1) CA2994203C (enExample)
DK (1) DK3331529T3 (enExample)
ES (1) ES2894637T3 (enExample)
GB (1) GB201513743D0 (enExample)
WO (1) WO2017021729A1 (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
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GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds
KR102798432B1 (ko) 2019-10-09 2025-04-22 노파르티스 아게 M4 작용제로서의 5-옥사-2-아자스피로[3.4]옥탄 유도체
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Also Published As

Publication number Publication date
US11254656B2 (en) 2022-02-22
EP3331529B1 (en) 2021-09-29
CN108025004B (zh) 2021-07-09
CA2994203A1 (en) 2017-02-09
GB201513743D0 (en) 2015-09-16
US10738029B2 (en) 2020-08-11
CN108025004A (zh) 2018-05-11
US20200354339A1 (en) 2020-11-12
EP3331529A1 (en) 2018-06-13
US20230002354A1 (en) 2023-01-05
ES2894637T3 (es) 2022-02-15
AU2016304387A1 (en) 2018-02-22
US20180222885A1 (en) 2018-08-09
CA2994203C (en) 2023-11-28
JP2018522033A (ja) 2018-08-09
US12024499B2 (en) 2024-07-02
DK3331529T3 (da) 2021-10-18
WO2017021729A1 (en) 2017-02-09
AU2016304387B2 (en) 2020-10-22
HK1250138A1 (en) 2018-11-30

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