JP6572497B2 - 修飾された治療剤、ステープル留めされたペプチド脂質複合体、及びそれらの組成物 - Google Patents

修飾された治療剤、ステープル留めされたペプチド脂質複合体、及びそれらの組成物 Download PDF

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JP6572497B2
JP6572497B2 JP2016541096A JP2016541096A JP6572497B2 JP 6572497 B2 JP6572497 B2 JP 6572497B2 JP 2016541096 A JP2016541096 A JP 2016541096A JP 2016541096 A JP2016541096 A JP 2016541096A JP 6572497 B2 JP6572497 B2 JP 6572497B2
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peptide
residues
amino acid
disease
lipids
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JP2017502024A (ja
JP2017502024A5 (enExample
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シェン,ウェイジュン
ヤン,ポンユ
ゾウ,フアフェイ
シュルツ,ピーター,ジー.
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Scripps Research Institute
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    • AHUMAN NECESSITIES
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    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
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    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/2278Vasoactive intestinal peptide [VIP]; Related peptides (e.g. Exendin)
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    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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JP2016541096A 2013-12-18 2014-12-17 修飾された治療剤、ステープル留めされたペプチド脂質複合体、及びそれらの組成物 Active JP6572497B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361917816P 2013-12-18 2013-12-18
US61/917,816 2013-12-18
PCT/US2014/070977 WO2015095406A1 (en) 2013-12-18 2014-12-17 Modified therapeutic agents, stapled peptide lipid conjugates, and compositions thereof

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JP2017502024A JP2017502024A (ja) 2017-01-19
JP2017502024A5 JP2017502024A5 (enExample) 2017-11-30
JP6572497B2 true JP6572497B2 (ja) 2019-09-11

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US (5) US10039809B2 (enExample)
EP (2) EP4212180A1 (enExample)
JP (1) JP6572497B2 (enExample)
KR (1) KR102455171B1 (enExample)
CN (1) CN106456589B (enExample)
AU (1) AU2014364589B2 (enExample)
CA (1) CA2933701C (enExample)
WO (1) WO2015095406A1 (enExample)

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