JP6148985B2 - ニトロカテコールの投与計画 - Google Patents

ニトロカテコールの投与計画 Download PDF

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Publication number
JP6148985B2
JP6148985B2 JP2013553014A JP2013553014A JP6148985B2 JP 6148985 B2 JP6148985 B2 JP 6148985B2 JP 2013553014 A JP2013553014 A JP 2013553014A JP 2013553014 A JP2013553014 A JP 2013553014A JP 6148985 B2 JP6148985 B2 JP 6148985B2
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administered
compound
pharmaceutical composition
formula
hour
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JP2014505096A (ja
JP2014505096A5 (enExample
Inventor
ダ シルヴァ、パトリシオ マヌエル ヴィエイラ アラウジョ ソアレス
ダ シルヴァ、パトリシオ マヌエル ヴィエイラ アラウジョ ソアレス
ルシア シルヴァ ペレイラ ヌネス、テレサ
ルシア シルヴァ ペレイラ ヌネス、テレサ
クリストファー ライト、リンドン
クリストファー ライト、リンドン
ヌノ リアル パルマ、ペドロ
ヌノ リアル パルマ、ペドロ
アレクサンダー リアマンス、デイヴィッド
アレクサンダー リアマンス、デイヴィッド
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ノヴィファーマ、エス．エー．
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00—Preparations for use in therapy

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
JP2013553014A 2011-02-11 2011-10-21 ニトロカテコールの投与計画 Active JP6148985B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161441988P 2011-02-11 2011-02-11
US61/441,988 2011-02-11
PCT/GB2011/052056 WO2012107708A1 (en) 2011-02-11 2011-10-21 Administration regime for nitrocatechols

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016220958A Division JP6389498B2 (ja) 2011-02-11 2016-11-11 ニトロカテコールの投与計画

Publications (3)

Publication Number Publication Date
JP2014505096A JP2014505096A (ja) 2014-02-27
JP2014505096A5 JP2014505096A5 (enExample) 2014-12-18
JP6148985B2 true JP6148985B2 (ja) 2017-06-14

Family

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Family Applications (4)

Application Number Title Priority Date Filing Date
JP2013553014A Active JP6148985B2 (ja) 2011-02-11 2011-10-21 ニトロカテコールの投与計画
JP2016220958A Active JP6389498B2 (ja) 2011-02-11 2016-11-11 ニトロカテコールの投与計画
JP2018153722A Active JP6568274B2 (ja) 2011-02-11 2018-08-17 ニトロカテコールの投与計画
JP2019142271A Active JP6843930B2 (ja) 2011-02-11 2019-08-01 ニトロカテコールの投与計画

Family Applications After (3)

Application Number Title Priority Date Filing Date
JP2016220958A Active JP6389498B2 (ja) 2011-02-11 2016-11-11 ニトロカテコールの投与計画
JP2018153722A Active JP6568274B2 (ja) 2011-02-11 2018-08-17 ニトロカテコールの投与計画
JP2019142271A Active JP6843930B2 (ja) 2011-02-11 2019-08-01 ニトロカテコールの投与計画

Country Status (18)

Country Link
US (4) US20140045900A1 (enExample)
EP (2) EP3831382A1 (enExample)
JP (4) JP6148985B2 (enExample)
AU (1) AU2011358842B2 (enExample)
BR (2) BR112013007380A2 (enExample)
CA (1) CA2826080C (enExample)
CY (1) CY1124022T1 (enExample)
DK (1) DK2672973T3 (enExample)
ES (1) ES2855162T3 (enExample)
HR (1) HRP20210474T1 (enExample)
HU (1) HUE054072T2 (enExample)
LT (1) LT2672973T (enExample)
PL (1) PL2672973T3 (enExample)
PT (1) PT2672973T (enExample)
RS (1) RS61643B1 (enExample)
RU (1) RU2639131C2 (enExample)
SI (1) SI2672973T1 (enExample)
WO (1) WO2012107708A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2017071619A (ja) * 2011-02-11 2017-04-13 ノヴィファーマ、エス．エー． ニトロカテコールの投与計画

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JP2020023540A (ja) * 2019-10-11 2020-02-13 ノヴィファーマ，エス．アー． パーキンソン病を遅延させるための医薬
JP7251026B2 (ja) 2019-11-14 2023-04-04 国立大学法人九州大学 ポリマー化合物およびコーティング組成物
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WO2022131944A1 (en) * 2020-12-17 2022-06-23 Bial-Portela & Ca., S.A. Treatment regimens for early idiopathic parkinson's disease

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