JP5406530B2 - 親水性ベヒクルに基づく二重制御された放出マトリクスシステム - Google Patents

親水性ベヒクルに基づく二重制御された放出マトリクスシステム Download PDF

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Publication number
JP5406530B2
JP5406530B2 JP2008538048A JP2008538048A JP5406530B2 JP 5406530 B2 JP5406530 B2 JP 5406530B2 JP 2008538048 A JP2008538048 A JP 2008538048A JP 2008538048 A JP2008538048 A JP 2008538048A JP 5406530 B2 JP5406530 B2 JP 5406530B2
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agent
matrix
hydrogel
hydrophilic vehicle
capsule
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JP2009513669A5 (https=
JP2009513669A (ja
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カルナカル スクル，
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バナー ファーマキャプス， インコーポレイテッド
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2008538048A 2005-10-26 2006-10-26 親水性ベヒクルに基づく二重制御された放出マトリクスシステム Expired - Fee Related JP5406530B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US73040605P 2005-10-26 2005-10-26
US60/730,406 2005-10-26
PCT/US2006/042177 WO2007050975A2 (en) 2005-10-26 2006-10-26 Hydrophilic vehicle-based dual controlled release matrix system as capsule fill

Related Child Applications (1)

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JP2013133677A Division JP2013216680A (ja) 2005-10-26 2013-06-26 親水性ベヒクルに基づく二重制御された放出マトリクスシステム

Publications (3)

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JP2009513669A JP2009513669A (ja) 2009-04-02
JP2009513669A5 JP2009513669A5 (https=) 2009-12-17
JP5406530B2 true JP5406530B2 (ja) 2014-02-05

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JP2008538048A Expired - Fee Related JP5406530B2 (ja) 2005-10-26 2006-10-26 親水性ベヒクルに基づく二重制御された放出マトリクスシステム
JP2013133677A Pending JP2013216680A (ja) 2005-10-26 2013-06-26 親水性ベヒクルに基づく二重制御された放出マトリクスシステム

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Country Link
US (1) US8333989B2 (https=)
EP (1) EP1959935A2 (https=)
JP (2) JP5406530B2 (https=)
CN (1) CN101360485B (https=)
CA (1) CA2627292C (https=)
WO (1) WO2007050975A2 (https=)

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Also Published As

Publication number Publication date
WO2007050975A3 (en) 2007-09-20
US8333989B2 (en) 2012-12-18
JP2013216680A (ja) 2013-10-24
CN101360485B (zh) 2013-04-17
US20070098783A1 (en) 2007-05-03
CN101360485A (zh) 2009-02-04
EP1959935A2 (en) 2008-08-27
JP2009513669A (ja) 2009-04-02
WO2007050975A2 (en) 2007-05-03
CA2627292C (en) 2012-04-17
CA2627292A1 (en) 2007-05-03

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