JP5160092B2 - ピリジン誘導体の調製方法 - Google Patents

ピリジン誘導体の調製方法 Download PDF

Info

Publication number
JP5160092B2
JP5160092B2 JP2006546051A JP2006546051A JP5160092B2 JP 5160092 B2 JP5160092 B2 JP 5160092B2 JP 2006546051 A JP2006546051 A JP 2006546051A JP 2006546051 A JP2006546051 A JP 2006546051A JP 5160092 B2 JP5160092 B2 JP 5160092B2
Authority
JP
Japan
Prior art keywords
substituted
alkyl
branched
cyclic
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP2006546051A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007519625A5 (enExample
JP2007519625A (ja
Inventor
ゲバルドト,ヨアヒム
ゲーツ,ノーバート
ヤエディック,ハーゲン
マイヤー,グイド
ラック,ミハエル
Original Assignee
ダウ アグロサイエンシィズ エルエルシー
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34923925&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JP5160092(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by ダウ アグロサイエンシィズ エルエルシー filed Critical ダウ アグロサイエンシィズ エルエルシー
Publication of JP2007519625A publication Critical patent/JP2007519625A/ja
Publication of JP2007519625A5 publication Critical patent/JP2007519625A5/ja
Application granted granted Critical
Publication of JP5160092B2 publication Critical patent/JP5160092B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C07D213/71—Sulfur atoms to which a second hetero atom is attached
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Indole Compounds (AREA)
JP2006546051A 2003-12-23 2004-12-22 ピリジン誘導体の調製方法 Expired - Lifetime JP5160092B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US53161403P 2003-12-23 2003-12-23
US60/531,614 2003-12-23
EP03029730.3 2003-12-23
EP03029730 2003-12-23
PCT/EP2004/014590 WO2005063780A1 (en) 2003-12-23 2004-12-22 Process for the preparation of pyridine derivatives

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2012139429A Division JP2012214487A (ja) 2003-12-23 2012-06-21 ピリジン誘導体の調製方法
JP2012229144A Division JP2013047245A (ja) 2003-12-23 2012-10-16 ピリジン誘導体の調製方法

Publications (3)

Publication Number Publication Date
JP2007519625A JP2007519625A (ja) 2007-07-19
JP2007519625A5 JP2007519625A5 (enExample) 2012-12-06
JP5160092B2 true JP5160092B2 (ja) 2013-03-13

Family

ID=34923925

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2006546051A Expired - Lifetime JP5160092B2 (ja) 2003-12-23 2004-12-22 ピリジン誘導体の調製方法
JP2012139429A Pending JP2012214487A (ja) 2003-12-23 2012-06-21 ピリジン誘導体の調製方法
JP2012229144A Pending JP2013047245A (ja) 2003-12-23 2012-10-16 ピリジン誘導体の調製方法

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2012139429A Pending JP2012214487A (ja) 2003-12-23 2012-06-21 ピリジン誘導体の調製方法
JP2012229144A Pending JP2013047245A (ja) 2003-12-23 2012-10-16 ピリジン誘導体の調製方法

Country Status (16)

Country Link
US (1) US7687632B2 (enExample)
EP (1) EP1723156B1 (enExample)
JP (3) JP5160092B2 (enExample)
KR (1) KR101164694B1 (enExample)
CN (1) CN1898255B (enExample)
AR (1) AR046775A1 (enExample)
AU (1) AU2004309054B2 (enExample)
BR (1) BRPI0418047B8 (enExample)
CA (1) CA2550693C (enExample)
DK (1) DK1723156T3 (enExample)
ES (1) ES2528716T3 (enExample)
IL (1) IL176472A (enExample)
IN (2) IN2012DN02545A (enExample)
PL (1) PL1723156T3 (enExample)
WO (1) WO2005063780A1 (enExample)
ZA (1) ZA200605471B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101648906B (zh) * 2004-04-08 2012-07-11 美国陶氏益农公司 杀虫用n-取代亚磺酰亚胺
US7488828B2 (en) * 2004-06-25 2009-02-10 Dow Agrosciences Llc Process for the preparation of 4-trifluoromethyl-2(1H)-pyridinone
TW201309635A (zh) 2006-02-10 2013-03-01 Dow Agrosciences Llc 殺蟲性之n-取代(6-鹵烷基吡啶-3-基)烷基磺醯亞胺(二)
TWI381811B (zh) * 2006-06-23 2013-01-11 Dow Agrosciences Llc 用以防治可抵抗一般殺蟲劑之昆蟲的方法
TWI387585B (zh) * 2006-09-01 2013-03-01 Dow Agrosciences Llc 殺蟲性之n-取代(雜芳基)烷基烴基硫亞胺
US7863303B2 (en) * 2006-09-01 2011-01-04 Dow Agrosciences Llc Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines
TWI395736B (zh) * 2006-11-08 2013-05-11 Dow Agrosciences Llc 作為殺蟲劑之雜芳基(取代的)烷基n-取代的磺醯亞胺(二)
US7709648B2 (en) * 2007-02-09 2010-05-04 Dow Agrosciences Llc Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines
AR066366A1 (es) * 2007-05-01 2009-08-12 Dow Agrosciences Llc Mezclas sinergicas plaguicidas
US20090023782A1 (en) * 2007-07-20 2009-01-22 Dow Agrosciences Llc Increasing plant vigor
KR20100127255A (ko) * 2008-03-03 2010-12-03 다우 아그로사이언시즈 엘엘씨 살충제
CN102875548A (zh) * 2011-07-14 2013-01-16 中国科学院大连化学物理研究所 一类基于肟的通过[2+2+2]环加成合成吡啶衍生物的方法
EP2607343A1 (en) 2011-12-22 2013-06-26 Solvay Sa Process for the manufacture of halogenated precursors of alkenones and of alkenones
CN117624038A (zh) * 2016-12-01 2024-03-01 先正达参股股份有限公司 具有含硫取代基的杀有害生物活性杂环衍生物
US12077505B2 (en) 2018-12-27 2024-09-03 Corteva Agriscience Llc Preparation of sulfonamide herbicide process intermediates
CN113227052B (zh) * 2018-12-27 2025-05-06 科迪华农业科技有限责任公司 磺酰胺除草剂方法中间体的制备
CN115286568B (zh) * 2022-08-24 2023-12-12 常州沃腾化工科技有限公司 一种2-羟基-4-三氟甲基吡啶的制备方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE611728A (fr) * 1960-07-12 1962-06-19 American Cyanamid Co Perfectionnements aux compositions contenant des antibiotiques à base de tétracycline
US3993656A (en) 1974-11-19 1976-11-23 Merck & Co., Inc. 1,8-Naphthyridine compounds
JPS5221196A (en) * 1975-08-12 1977-02-17 Fujio Hashimoto Device for removing red tide
JPS5384990A (en) * 1976-12-29 1978-07-26 Yamanouchi Pharmaceut Co Ltd Novel nitrogen-containing heterocyclic compound and its preparation
JPS53121764A (en) * 1977-03-31 1978-10-24 Yamanouchi Pharmaceut Co Ltd Heterocyclic compounds and process for their preparation
JPS53127490A (en) * 1977-04-13 1978-11-07 Yamanouchi Pharmaceut Co Ltd Novel nitrogen-containing heterocyclic compound
JPS55104266A (en) * 1979-02-02 1980-08-09 Yamanouchi Pharmaceut Co Ltd Novel pyridone derivative
JPS6210087A (ja) * 1985-07-03 1987-01-19 Shionogi & Co Ltd 4,7−ジヒドロチエノ〔2,3−b〕ピリジン誘導体,その製造法および循環器系疾患治療剤
JPS6413065A (en) * 1987-07-06 1989-01-17 Mitsubishi Chem Ind Peptide derivative of beta-chloro-l-(z)- dehydroglutamic acid
DK177191D0 (da) * 1991-10-23 1991-10-23 Novo Nordisk As Heterocyclic compounds and their preparation and use
US5391745A (en) * 1992-07-23 1995-02-21 Sloan-Kettering Institute For Cancer Research Methods of preparation of camptothecin analogs
CN1159297C (zh) 1996-09-24 2004-07-28 道农业科学公司 N-([1,2,4]三唑并吖嗪基)苯磺酰胺和吡啶磺酰胺化合物和它们作为除草剂的用途
DE69919707T2 (de) * 1998-06-19 2005-09-01 Chiron Corp., Emeryville Glycogen synthase kinase 3 inhibitoren
EP1301483A1 (de) * 2000-07-18 2003-04-16 Basf Aktiengesellschaft 1-aryl-4-halogenalkyl-2-(1h)-pyridone und ihre verwendung als herbizide
US6399781B1 (en) 2000-10-10 2002-06-04 Boehringer Ingelheim Chemicals, Inc. Process for making 3-amino-2-chloro-4-methylpyridine
US7488828B2 (en) * 2004-06-25 2009-02-10 Dow Agrosciences Llc Process for the preparation of 4-trifluoromethyl-2(1H)-pyridinone

Also Published As

Publication number Publication date
IL176472A (en) 2010-11-30
CN1898255B (zh) 2010-06-09
IN2012DN02546A (enExample) 2015-08-28
PL1723156T3 (pl) 2015-07-31
KR101164694B1 (ko) 2012-07-11
BRPI0418047B8 (pt) 2022-06-28
EP1723156B1 (en) 2015-01-21
IL176472A0 (en) 2006-10-05
BRPI0418047B1 (pt) 2013-12-31
AR046775A1 (es) 2005-12-21
JP2013047245A (ja) 2013-03-07
IN2012DN02545A (enExample) 2015-07-17
JP2012214487A (ja) 2012-11-08
CN1898255A (zh) 2007-01-17
US20070249837A1 (en) 2007-10-25
KR20060128896A (ko) 2006-12-14
CA2550693C (en) 2013-07-30
AU2004309054B2 (en) 2010-07-08
BRPI0418047A (pt) 2007-04-17
JP2007519625A (ja) 2007-07-19
US7687632B2 (en) 2010-03-30
ES2528716T3 (es) 2015-02-12
DK1723156T3 (en) 2015-04-27
EP1723156A1 (en) 2006-11-22
WO2005063780A1 (en) 2005-07-14
CA2550693A1 (en) 2005-07-14
AU2004309054A1 (en) 2005-07-14
ZA200605471B (en) 2007-11-28

Similar Documents

Publication Publication Date Title
JP2013047245A (ja) ピリジン誘導体の調製方法
EP1071745B1 (en) Process for synthesizing cox-2 inhibitors
JP4157325B2 (ja) Cox−2のインヒビターとして有用なジアリールピリジンの製造方法
KR20130105936A (ko) 2-치환된-5-(1-알킬티오)알킬피리딘의 제조 방법
JP5077969B2 (ja) 2−置換5−(1−アルキルチオ)アルキルピリジンの調製方法
PL190265B1 (pl) Sposób wytwarzania związków 2-arylo-3-arylopirydynowych
KR20150093799A (ko) 4-아미노-5-플루오로-3-클로로-6-(치환된)피콜리네이트의제조 방법
KR100411410B1 (ko) 2-(치환된벤조일)-1,3싸이클로헥산디온의제조방법
JP2583062B2 (ja) 複素環化合物の製造法
JPH0742303B2 (ja) ホスホン酸のふっ素含有誘導体の製造法
MXPA06007401A (es) Proceso para la preparacion de derivados de piridina
JPH04243875A (ja) 2−フェニル−6−(ピリミジン−2−イル)ピリジン化合物の製造方法、中間体化合物及び中間体化合物の製造方法
EP2797897B1 (en) 2,6-dihalo-5-alkoxy-4-substituted-pyrimidines, pyrimidine- carbaldehydes, and methods of formation and use
JP4316299B2 (ja) 鎖状乳酸オリゴマー誘導体およびその製造方法
JP2005126340A (ja) 置換ピリドン類の製造法、その原料化合物及びその製造方法
Goehring A CONVENIENT PREPARATION OF 9 H-FLUORENE-9-ACETIC ACID
JP2005068036A (ja) 置換ピリドン類の製造方法、その原料化合物およびその製造方法
JP2861157B2 (ja) 置換基を有するニコチン酸誘導体及びその製造方法
JPS5951534B2 (ja) 2−アミノ−3−ヒドロキシピリジン誘導体の製造法
JPS6231696B2 (enExample)
HK1023771B (en) Process for making 2-aryl-3-aryl-5-halo pyridines useful as cox-2 inhibitors
JPS5940814B2 (ja) α−クロロカルボン酸類
JPH0434551B2 (enExample)
HK1174028A (en) Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines

Legal Events

Date Code Title Description
A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20071219

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20110621

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20110920

A602 Written permission of extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A602

Effective date: 20110928

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20111021

A602 Written permission of extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A602

Effective date: 20111028

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20111118

A02 Decision of refusal

Free format text: JAPANESE INTERMEDIATE CODE: A02

Effective date: 20120221

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20120621

A911 Transfer to examiner for re-examination before appeal (zenchi)

Free format text: JAPANESE INTERMEDIATE CODE: A911

Effective date: 20120702

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20120724

A524 Written submission of copy of amendment under article 19 pct

Free format text: JAPANESE INTERMEDIATE CODE: A524

Effective date: 20121016

TRDD Decision of grant or rejection written
A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

Effective date: 20121113

A61 First payment of annual fees (during grant procedure)

Free format text: JAPANESE INTERMEDIATE CODE: A61

Effective date: 20121212

R150 Certificate of patent or registration of utility model

Free format text: JAPANESE INTERMEDIATE CODE: R150

Ref document number: 5160092

Country of ref document: JP

Free format text: JAPANESE INTERMEDIATE CODE: R150

FPAY Renewal fee payment (event date is renewal date of database)

Free format text: PAYMENT UNTIL: 20151221

Year of fee payment: 3

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

S533 Written request for registration of change of name

Free format text: JAPANESE INTERMEDIATE CODE: R313533

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R350 Written notification of registration of transfer

Free format text: JAPANESE INTERMEDIATE CODE: R350

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

R250 Receipt of annual fees

Free format text: JAPANESE INTERMEDIATE CODE: R250

EXPY Cancellation because of completion of term