JP5160092B2 - ピリジン誘導体の調製方法 - Google Patents

ピリジン誘導体の調製方法 Download PDF

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Publication number
JP5160092B2
JP5160092B2 JP2006546051A JP2006546051A JP5160092B2 JP 5160092 B2 JP5160092 B2 JP 5160092B2 JP 2006546051 A JP2006546051 A JP 2006546051A JP 2006546051 A JP2006546051 A JP 2006546051A JP 5160092 B2 JP5160092 B2 JP 5160092B2
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JP
Japan
Prior art keywords
substituted
alkyl
branched
cyclic
aryl
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JP2006546051A
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English (en)
Japanese (ja)
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JP2007519625A (ja
JP2007519625A5 (enExample
Inventor
ゲバルドト，ヨアヒム
ゲーツ，ノーバート
ヤエディック，ハーゲン
マイヤー，グイド
ラック，ミハエル
Original Assignee
ダウ アグロサイエンシィズ エルエルシー
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Application filed by ダウ アグロサイエンシィズ エルエルシー filed Critical ダウ アグロサイエンシィズ エルエルシー
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Publication of JP2007519625A5 publication Critical patent/JP2007519625A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C07D213/71—Sulfur atoms to which a second hetero atom is attached
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Indole Compounds (AREA)
JP2006546051A 2003-12-23 2004-12-22 ピリジン誘導体の調製方法 Expired - Lifetime JP5160092B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US53161403P 2003-12-23 2003-12-23
EP03029730 2003-12-23
EP03029730.3 2003-12-23
US60/531,614 2003-12-23
PCT/EP2004/014590 WO2005063780A1 (en) 2003-12-23 2004-12-22 Process for the preparation of pyridine derivatives

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2012139429A Division JP2012214487A (ja) 2003-12-23 2012-06-21 ピリジン誘導体の調製方法
JP2012229144A Division JP2013047245A (ja) 2003-12-23 2012-10-16 ピリジン誘導体の調製方法

Publications (3)

Publication Number Publication Date
JP2007519625A JP2007519625A (ja) 2007-07-19
JP2007519625A5 JP2007519625A5 (enExample) 2012-12-06
JP5160092B2 true JP5160092B2 (ja) 2013-03-13

Family

ID=34923925

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2006546051A Expired - Lifetime JP5160092B2 (ja) 2003-12-23 2004-12-22 ピリジン誘導体の調製方法
JP2012139429A Pending JP2012214487A (ja) 2003-12-23 2012-06-21 ピリジン誘導体の調製方法
JP2012229144A Pending JP2013047245A (ja) 2003-12-23 2012-10-16 ピリジン誘導体の調製方法

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2012139429A Pending JP2012214487A (ja) 2003-12-23 2012-06-21 ピリジン誘導体の調製方法
JP2012229144A Pending JP2013047245A (ja) 2003-12-23 2012-10-16 ピリジン誘導体の調製方法

Country Status (16)

Country Link
US (1) US7687632B2 (enExample)
EP (1) EP1723156B1 (enExample)
JP (3) JP5160092B2 (enExample)
KR (1) KR101164694B1 (enExample)
CN (1) CN1898255B (enExample)
AR (1) AR046775A1 (enExample)
AU (1) AU2004309054B2 (enExample)
BR (1) BRPI0418047B8 (enExample)
CA (1) CA2550693C (enExample)
DK (1) DK1723156T3 (enExample)
ES (1) ES2528716T3 (enExample)
IL (1) IL176472A (enExample)
IN (2) IN2012DN02546A (enExample)
PL (1) PL1723156T3 (enExample)
WO (1) WO2005063780A1 (enExample)
ZA (1) ZA200605471B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2558647C (en) * 2004-04-08 2013-05-28 Dow Agrosciences Llc Insecticidal n-substituted sulfoximines
WO2006012320A1 (en) * 2004-06-25 2006-02-02 Dow Agrosciences Llc Process for the preparation of 4-trifluoromethyl-2(1h)-pyridinone
TWI398433B (zh) * 2006-02-10 2013-06-11 Dow Agrosciences Llc 殺蟲性之ｎ-取代（６-鹵烷基吡啶-３-基）烷基磺醯亞胺
TWI381811B (zh) * 2006-06-23 2013-01-11 Dow Agrosciences Llc 用以防治可抵抗一般殺蟲劑之昆蟲的方法
TWI387585B (zh) * 2006-09-01 2013-03-01 Dow Agrosciences Llc 殺蟲性之ｎ-取代（雜芳基）烷基烴基硫亞胺
EP2057135B1 (en) * 2006-09-01 2012-06-13 Dow AgroSciences LLC Insecticidal n-substituted (2- substituted-1,3-thiazol) alkyl sulfoximines
TWI395737B (zh) * 2006-11-08 2013-05-11 Dow Agrosciences Llc 作為殺蟲劑之雜芳基（取代的）烷基ｎ-取代的磺醯亞胺
US7709648B2 (en) * 2007-02-09 2010-05-04 Dow Agrosciences Llc Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines
AR066366A1 (es) * 2007-05-01 2009-08-12 Dow Agrosciences Llc Mezclas sinergicas plaguicidas
PL2166851T3 (pl) * 2007-07-20 2012-02-29 Dow Agrosciences Llc Zwiększanie żywotności roślin
JP5487123B2 (ja) * 2008-03-03 2014-05-07 ダウ アグロサイエンシィズ エルエルシー 農薬
CN102875548A (zh) * 2011-07-14 2013-01-16 中国科学院大连化学物理研究所 一类基于肟的通过[2+2+2]环加成合成吡啶衍生物的方法
EP2607343A1 (en) 2011-12-22 2013-06-26 Solvay Sa Process for the manufacture of halogenated precursors of alkenones and of alkenones
DK3548466T3 (da) * 2016-12-01 2022-04-19 Syngenta Participations Ag Fremgangsmåde til fremstilling af et mellemprodukt af pesticidaktive heterocykliske derivater med svovlindeholdende substituenter
JP7551622B2 (ja) * 2018-12-27 2024-09-17 コルテバ アグリサイエンス エルエルシー スルホンアミド除草剤プロセス中間生成物の調製
CN120172888A (zh) 2018-12-27 2025-06-20 科迪华农业科技有限责任公司 磺酰胺除草剂方法中间体的制备
CN115286568B (zh) * 2022-08-24 2023-12-12 常州沃腾化工科技有限公司 一种2-羟基-4-三氟甲基吡啶的制备方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE611728A (fr) * 1960-07-12 1962-06-19 American Cyanamid Co Perfectionnements aux compositions contenant des antibiotiques à base de tétracycline
US3993656A (en) 1974-11-19 1976-11-23 Merck & Co., Inc. 1,8-Naphthyridine compounds
JPS5221196A (en) * 1975-08-12 1977-02-17 Fujio Hashimoto Device for removing red tide
JPS53121764A (en) * 1977-03-31 1978-10-24 Yamanouchi Pharmaceut Co Ltd Heterocyclic compounds and process for their preparation
JPS5384990A (en) * 1976-12-29 1978-07-26 Yamanouchi Pharmaceut Co Ltd Novel nitrogen-containing heterocyclic compound and its preparation
JPS53127490A (en) * 1977-04-13 1978-11-07 Yamanouchi Pharmaceut Co Ltd Novel nitrogen-containing heterocyclic compound
JPS55104266A (en) * 1979-02-02 1980-08-09 Yamanouchi Pharmaceut Co Ltd Novel pyridone derivative
JPS6210087A (ja) * 1985-07-03 1987-01-19 Shionogi & Co Ltd ４，７−ジヒドロチエノ〔２，３−ｂ〕ピリジン誘導体，その製造法および循環器系疾患治療剤
JPS6413065A (en) * 1987-07-06 1989-01-17 Mitsubishi Chem Ind Peptide derivative of beta-chloro-l-(z)- dehydroglutamic acid
DK177191D0 (da) * 1991-10-23 1991-10-23 Novo Nordisk As Heterocyclic compounds and their preparation and use
US5391745A (en) * 1992-07-23 1995-02-21 Sloan-Kettering Institute For Cancer Research Methods of preparation of camptothecin analogs
CA2238316C (en) 1996-09-24 2007-01-30 Dow Agrosciences Llc N-([1,2,4]triazoloazinyl)benzenesulfonamide and pyridinesulfonamide compounds and their use as herbicides
ATE274510T1 (de) * 1998-06-19 2004-09-15 Chiron Corp Glycogen synthase kinase 3 inhibitoren
CA2416192A1 (en) * 2000-07-18 2003-01-15 Basf Aktiengesellschaft 1-aryl-4-alkyl halide-2(1h)-pyridones and their use as herbicides
US6399781B1 (en) * 2000-10-10 2002-06-04 Boehringer Ingelheim Chemicals, Inc. Process for making 3-amino-2-chloro-4-methylpyridine
WO2006012320A1 (en) * 2004-06-25 2006-02-02 Dow Agrosciences Llc Process for the preparation of 4-trifluoromethyl-2(1h)-pyridinone

Also Published As

Publication number Publication date
KR20060128896A (ko) 2006-12-14
ZA200605471B (en) 2007-11-28
EP1723156A1 (en) 2006-11-22
IL176472A (en) 2010-11-30
US7687632B2 (en) 2010-03-30
EP1723156B1 (en) 2015-01-21
WO2005063780A1 (en) 2005-07-14
AR046775A1 (es) 2005-12-21
BRPI0418047B1 (pt) 2013-12-31
IL176472A0 (en) 2006-10-05
DK1723156T3 (en) 2015-04-27
KR101164694B1 (ko) 2012-07-11
JP2013047245A (ja) 2013-03-07
US20070249837A1 (en) 2007-10-25
CA2550693A1 (en) 2005-07-14
AU2004309054B2 (en) 2010-07-08
CN1898255A (zh) 2007-01-17
JP2007519625A (ja) 2007-07-19
IN2012DN02546A (enExample) 2015-08-28
IN2012DN02545A (enExample) 2015-07-17
BRPI0418047A (pt) 2007-04-17
ES2528716T3 (es) 2015-02-12
AU2004309054A1 (en) 2005-07-14
JP2012214487A (ja) 2012-11-08
CA2550693C (en) 2013-07-30
BRPI0418047B8 (pt) 2022-06-28
CN1898255B (zh) 2010-06-09
PL1723156T3 (pl) 2015-07-31

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