BRPI0418047B8 - Processo para a preparação de derivados de piridina e composto intermediário - Google Patents
Processo para a preparação de derivados de piridina e composto intermediárioInfo
- Publication number
- BRPI0418047B8 BRPI0418047B8 BRPI0418047A BRPI0418047A BRPI0418047B8 BR PI0418047 B8 BRPI0418047 B8 BR PI0418047B8 BR PI0418047 A BRPI0418047 A BR PI0418047A BR PI0418047 A BRPI0418047 A BR PI0418047A BR PI0418047 B8 BRPI0418047 B8 BR PI0418047B8
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- pyridine derivatives
- intermediate compound
- formula
- reagent
- Prior art date
Links
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical class C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 title 1
- 239000003153 chemical reaction reagent Substances 0.000 abstract 2
- 150000001728 carbonyl compounds Chemical class 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- UMJSCPRVCHMLSP-UHFFFAOYSA-N pyridine Natural products COC1=CC=CN=C1 UMJSCPRVCHMLSP-UHFFFAOYSA-N 0.000 abstract 1
- 150000003222 pyridines Chemical class 0.000 abstract 1
- 238000007363 ring formation reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
- C07D213/71—Sulfur atoms to which a second hetero atom is attached
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
- C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
- C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Pyridine Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US53161403P | 2003-12-23 | 2003-12-23 | |
| EP03029730 | 2003-12-23 | ||
| EP2005063780 | 2005-07-14 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| BRPI0418047A BRPI0418047A (pt) | 2007-04-17 |
| BRPI0418047B1 BRPI0418047B1 (pt) | 2013-12-31 |
| BRPI0418047B8 true BRPI0418047B8 (pt) | 2022-06-28 |
Family
ID=34923925
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0418047A BRPI0418047B8 (pt) | 2003-12-23 | 2004-12-22 | Processo para a preparação de derivados de piridina e composto intermediário |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US7687632B2 (enExample) |
| EP (1) | EP1723156B1 (enExample) |
| JP (3) | JP5160092B2 (enExample) |
| KR (1) | KR101164694B1 (enExample) |
| CN (1) | CN1898255B (enExample) |
| AR (1) | AR046775A1 (enExample) |
| AU (1) | AU2004309054B2 (enExample) |
| BR (1) | BRPI0418047B8 (enExample) |
| CA (1) | CA2550693C (enExample) |
| DK (1) | DK1723156T3 (enExample) |
| ES (1) | ES2528716T3 (enExample) |
| IL (1) | IL176472A (enExample) |
| IN (2) | IN2012DN02546A (enExample) |
| PL (1) | PL1723156T3 (enExample) |
| WO (1) | WO2005063780A1 (enExample) |
| ZA (1) | ZA200605471B (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7678920B2 (en) * | 2004-04-08 | 2010-03-16 | Dow Agrosciences Llc | Insecticidal N-substituted sulfoximines |
| US7488828B2 (en) * | 2004-06-25 | 2009-02-10 | Dow Agrosciences Llc | Process for the preparation of 4-trifluoromethyl-2(1H)-pyridinone |
| TW201309635A (zh) | 2006-02-10 | 2013-03-01 | Dow Agrosciences Llc | 殺蟲性之ｎ-取代（６-鹵烷基吡啶-３-基）烷基磺醯亞胺（二） |
| TWI381811B (zh) * | 2006-06-23 | 2013-01-11 | Dow Agrosciences Llc | 用以防治可抵抗一般殺蟲劑之昆蟲的方法 |
| TWI387585B (zh) * | 2006-09-01 | 2013-03-01 | Dow Agrosciences Llc | 殺蟲性之ｎ-取代（雜芳基）烷基烴基硫亞胺 |
| WO2008027539A1 (en) * | 2006-09-01 | 2008-03-06 | Dow Agrosciences Llc | Insecticidal n-substituted (2- sudstituted-1,3-thiazol) alkyl sulfoximines |
| TWI395736B (zh) * | 2006-11-08 | 2013-05-11 | Dow Agrosciences Llc | 作為殺蟲劑之雜芳基（取代的）烷基ｎ-取代的磺醯亞胺（二） |
| US7709648B2 (en) * | 2007-02-09 | 2010-05-04 | Dow Agrosciences Llc | Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines |
| AR066366A1 (es) * | 2007-05-01 | 2009-08-12 | Dow Agrosciences Llc | Mezclas sinergicas plaguicidas |
| US20090023782A1 (en) * | 2007-07-20 | 2009-01-22 | Dow Agrosciences Llc | Increasing plant vigor |
| CN102015634B (zh) * | 2008-03-03 | 2014-02-12 | 陶氏益农公司 | 杀虫剂 |
| CN102875548A (zh) * | 2011-07-14 | 2013-01-16 | 中国科学院大连化学物理研究所 | 一类基于肟的通过[2+2+2]环加成合成吡啶衍生物的方法 |
| EP2607343A1 (en) | 2011-12-22 | 2013-06-26 | Solvay Sa | Process for the manufacture of halogenated precursors of alkenones and of alkenones |
| US10961248B2 (en) * | 2016-12-01 | 2021-03-30 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| US12077505B2 (en) | 2018-12-27 | 2024-09-03 | Corteva Agriscience Llc | Preparation of sulfonamide herbicide process intermediates |
| CN120172888A (zh) * | 2018-12-27 | 2025-06-20 | 科迪华农业科技有限责任公司 | 磺酰胺除草剂方法中间体的制备 |
| CN115286568B (zh) * | 2022-08-24 | 2023-12-12 | 常州沃腾化工科技有限公司 | 一种2-羟基-4-三氟甲基吡啶的制备方法 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE611728A (fr) * | 1960-07-12 | 1962-06-19 | American Cyanamid Co | Perfectionnements aux compositions contenant des antibiotiques à base de tétracycline |
| US3993656A (en) | 1974-11-19 | 1976-11-23 | Merck & Co., Inc. | 1,8-Naphthyridine compounds |
| JPS5221196A (en) * | 1975-08-12 | 1977-02-17 | Fujio Hashimoto | Device for removing red tide |
| JPS5384990A (en) * | 1976-12-29 | 1978-07-26 | Yamanouchi Pharmaceut Co Ltd | Novel nitrogen-containing heterocyclic compound and its preparation |
| JPS53121764A (en) * | 1977-03-31 | 1978-10-24 | Yamanouchi Pharmaceut Co Ltd | Heterocyclic compounds and process for their preparation |
| JPS53127490A (en) * | 1977-04-13 | 1978-11-07 | Yamanouchi Pharmaceut Co Ltd | Novel nitrogen-containing heterocyclic compound |
| JPS55104266A (en) * | 1979-02-02 | 1980-08-09 | Yamanouchi Pharmaceut Co Ltd | Novel pyridone derivative |
| JPS6210087A (ja) * | 1985-07-03 | 1987-01-19 | Shionogi & Co Ltd | ４，７−ジヒドロチエノ〔２，３−ｂ〕ピリジン誘導体，その製造法および循環器系疾患治療剤 |
| JPS6413065A (en) * | 1987-07-06 | 1989-01-17 | Mitsubishi Chem Ind | Peptide derivative of beta-chloro-l-(z)- dehydroglutamic acid |
| DK177191D0 (da) * | 1991-10-23 | 1991-10-23 | Novo Nordisk As | Heterocyclic compounds and their preparation and use |
| US5391745A (en) * | 1992-07-23 | 1995-02-21 | Sloan-Kettering Institute For Cancer Research | Methods of preparation of camptothecin analogs |
| PL190282B1 (pl) | 1996-09-24 | 2005-11-30 | Dow Agrosciences Llc | Związki N-([1,2,4]triazoloazynylo)benzeno-i pirydynosulfonamidowe, zawierające je kompozycje herbicydowe, pochodne chlorku pirydyno-3-sulfonylu i pochodne 2-amino[1.2.4]triazolo[1.5-c]pirymidyny |
| JP4533534B2 (ja) * | 1998-06-19 | 2010-09-01 | ノバルティス バクシンズ アンド ダイアグノスティックス，インコーポレーテッド | グリコーゲンシンターゼキナーゼ３のインヒビター |
| JP2004504300A (ja) * | 2000-07-18 | 2004-02-12 | ビーエーエスエフ アクチェンゲゼルシャフト | １−アリール−４−ハロアルキル−２−［１ｈ］ピリドン類 |
| US6399781B1 (en) | 2000-10-10 | 2002-06-04 | Boehringer Ingelheim Chemicals, Inc. | Process for making 3-amino-2-chloro-4-methylpyridine |
| US7488828B2 (en) * | 2004-06-25 | 2009-02-10 | Dow Agrosciences Llc | Process for the preparation of 4-trifluoromethyl-2(1H)-pyridinone |
-
2004
- 2004-12-11 ZA ZA200605471A patent/ZA200605471B/en unknown
- 2004-12-22 JP JP2006546051A patent/JP5160092B2/ja not_active Expired - Lifetime
- 2004-12-22 EP EP04804186.7A patent/EP1723156B1/en not_active Expired - Lifetime
- 2004-12-22 KR KR1020067012653A patent/KR101164694B1/ko not_active Expired - Lifetime
- 2004-12-22 PL PL04804186T patent/PL1723156T3/pl unknown
- 2004-12-22 WO PCT/EP2004/014590 patent/WO2005063780A1/en not_active Ceased
- 2004-12-22 AU AU2004309054A patent/AU2004309054B2/en not_active Expired
- 2004-12-22 IN IN2546DEN2012 patent/IN2012DN02546A/en unknown
- 2004-12-22 CN CN2004800388844A patent/CN1898255B/zh not_active Expired - Lifetime
- 2004-12-22 ES ES04804186.7T patent/ES2528716T3/es not_active Expired - Lifetime
- 2004-12-22 IN IN2545DEN2012 patent/IN2012DN02545A/en unknown
- 2004-12-22 DK DK04804186.7T patent/DK1723156T3/en active
- 2004-12-22 AR ARP040104854A patent/AR046775A1/es active IP Right Grant
- 2004-12-22 CA CA2550693A patent/CA2550693C/en not_active Expired - Lifetime
- 2004-12-22 US US10/584,354 patent/US7687632B2/en active Active
- 2004-12-22 BR BRPI0418047A patent/BRPI0418047B8/pt not_active IP Right Cessation
-
2006
- 2006-06-21 IL IL176472A patent/IL176472A/en active IP Right Grant
-
2012
- 2012-06-21 JP JP2012139429A patent/JP2012214487A/ja active Pending
- 2012-10-16 JP JP2012229144A patent/JP2013047245A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200605471B (en) | 2007-11-28 |
| AU2004309054A1 (en) | 2005-07-14 |
| BRPI0418047A (pt) | 2007-04-17 |
| KR20060128896A (ko) | 2006-12-14 |
| DK1723156T3 (en) | 2015-04-27 |
| AR046775A1 (es) | 2005-12-21 |
| PL1723156T3 (pl) | 2015-07-31 |
| CA2550693C (en) | 2013-07-30 |
| IL176472A (en) | 2010-11-30 |
| AU2004309054B2 (en) | 2010-07-08 |
| JP5160092B2 (ja) | 2013-03-13 |
| CN1898255B (zh) | 2010-06-09 |
| JP2007519625A (ja) | 2007-07-19 |
| CN1898255A (zh) | 2007-01-17 |
| IN2012DN02546A (enExample) | 2015-08-28 |
| EP1723156B1 (en) | 2015-01-21 |
| BRPI0418047B1 (pt) | 2013-12-31 |
| ES2528716T3 (es) | 2015-02-12 |
| IL176472A0 (en) | 2006-10-05 |
| US7687632B2 (en) | 2010-03-30 |
| KR101164694B1 (ko) | 2012-07-11 |
| CA2550693A1 (en) | 2005-07-14 |
| WO2005063780A1 (en) | 2005-07-14 |
| JP2012214487A (ja) | 2012-11-08 |
| JP2013047245A (ja) | 2013-03-07 |
| EP1723156A1 (en) | 2006-11-22 |
| IN2012DN02545A (enExample) | 2015-07-17 |
| US20070249837A1 (en) | 2007-10-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BRPI0418047B8 (pt) | Processo para a preparação de derivados de piridina e composto intermediário | |
| BRPI0417543A (pt) | quinolinas úteis no tratamento de doença cardiovascular | |
| BR0308979A (pt) | Derivados de indolilmaleimida | |
| CY1109055T1 (el) | 11-((4r,6r)-4,5,6-τριϋδροξυ-3-(r)-υδροξυ-εξυλοκαρβαμοϋλο)-ενδεκαϊνικο οξυ | |
| AR022469A1 (es) | Uso de acidos isoxazolcarboxilicos sustituidos y derivados y nuevas sustancias | |
| BRPI0207172B8 (pt) | pirido-pirimidinas 6-substituída, sua composição e seu uso, bem como seu intermediário | |
| BR0314688A (pt) | Novos derivados de piperidina para utilização no tratamento de estados de doença mediados pela quimiocina | |
| BR9904998B1 (pt) | derivados de hidroxamida do ácido 5-oxo-pirrolidina-2-carboxìlico e composição farmacêutica. | |
| PT911333E (pt) | Derivados de pirazolo¬4,3-d|pirimidina e composicoes farmaceuticas que os contenham | |
| BR0213380A (pt) | Derivados propiÈnicos alfa-oxissubstituìdos por beta-fenila: processo para sua preparação e seu uso na preparação de compostos farmaceuticamente importantes | |
| BR9917518A (pt) | Processos para a preparação de pestecidas 1-arilpirazóis e seus intermediários | |
| ECSP055910A (es) | Nuevos acidos carboxilicos y sus esteres, medicamentos que contienen estos compuestos y procedimientos para su preparacion | |
| BR0212968A (pt) | Composição farmacêutica, composto, e, método para tratar ou prevenir condições mediadas pelo ccr2, mcp-1 ou pela interação destes | |
| BR0211502A (pt) | Derivados de ácido acético de indano e seu uso como agentes farmacêuticos, intermediários, e método de preparação | |
| BRPI0410995A (pt) | derivados de n-alquinil-2-(arilóxi substituìdo)alquiltioamida como fungicidas | |
| DOP2001000205A (es) | Derivados de ciclopentil-glutaramida como inhibidores de endopeptidasa neutra | |
| CY1109740T1 (el) | Νεα μεθοδος συνθεσης παραγωγων της 1,3,4,5 -τετραϋδρο-2η- 3-βενζαζεπιν-2-ονης και εφαρμογη στη συνθεση της ιβαβραδινης και των αλατων προσθηκης της σε ενα φαρμακευτικως αποδεκτο οξυ | |
| BR0313846A (pt) | Derivados de dioxano-2-alquilcarbamatos, sua preparação e sua aplicação em terapêutica | |
| BR0210842A (pt) | Processo para a preparação de intermediários úteis na sìntese de derivados de estatina, especialmente derivados do ácido 7-amino 3,5-dihidróxi heptanóico, e intermediários dos mesmos | |
| BRPI0411738A (pt) | compostos orgánicos | |
| BRPI0406500A (pt) | processo farmacêutico e compostos preparados pelo mesmo | |
| BRPI0412862A (pt) | derivados da nicotinamida úteis como inibidores de pde4 | |
| BRPI0412910A (pt) | derivados de nicotinamida úteis como inibidores de pde4 | |
| MEP18708A (en) | Process for the production of beraprost and its salts | |
| BRPI0408389A (pt) | derivados de cromeno como agentes antiinflamatórios |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 22/12/2004, OBSERVADAS AS CONDICOES LEGAIS. |
|
| B25D | Requested change of name of applicant approved | ||
| B21A | Patent or certificate of addition expired [chapter 21.1 patent gazette] |
Free format text: PATENTE EXTINTA EM 22/12/2024 |