KR101164694B1 - 피리딘 유도체의 제조 방법 - Google Patents

피리딘 유도체의 제조 방법 Download PDF

Info

Publication number
KR101164694B1
KR101164694B1 KR1020067012653A KR20067012653A KR101164694B1 KR 101164694 B1 KR101164694 B1 KR 101164694B1 KR 1020067012653 A KR1020067012653 A KR 1020067012653A KR 20067012653 A KR20067012653 A KR 20067012653A KR 101164694 B1 KR101164694 B1 KR 101164694B1
Authority
KR
South Korea
Prior art keywords
formula
alkyl
alkoxy
aryl
aryloxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
KR1020067012653A
Other languages
English (en)
Korean (ko)
Other versions
KR20060128896A (ko
Inventor
요아킴 게브하르트
노베르트 괴츠
하겐 야에디케
구이도 마이어
미카엘 라크
Original Assignee
다우 아그로사이언시즈 엘엘씨
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34923925&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR101164694(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 다우 아그로사이언시즈 엘엘씨 filed Critical 다우 아그로사이언시즈 엘엘씨
Publication of KR20060128896A publication Critical patent/KR20060128896A/ko
Application granted granted Critical
Publication of KR101164694B1 publication Critical patent/KR101164694B1/ko
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C07D213/71—Sulfur atoms to which a second hetero atom is attached
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Indole Compounds (AREA)
KR1020067012653A 2003-12-23 2004-12-22 피리딘 유도체의 제조 방법 Expired - Lifetime KR101164694B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US53161403P 2003-12-23 2003-12-23
EP03029730.3 2003-12-23
EP03029730 2003-12-23
US60/531,614 2003-12-23
PCT/EP2004/014590 WO2005063780A1 (en) 2003-12-23 2004-12-22 Process for the preparation of pyridine derivatives

Publications (2)

Publication Number Publication Date
KR20060128896A KR20060128896A (ko) 2006-12-14
KR101164694B1 true KR101164694B1 (ko) 2012-07-11

Family

ID=34923925

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020067012653A Expired - Lifetime KR101164694B1 (ko) 2003-12-23 2004-12-22 피리딘 유도체의 제조 방법

Country Status (16)

Country Link
US (1) US7687632B2 (enExample)
EP (1) EP1723156B1 (enExample)
JP (3) JP5160092B2 (enExample)
KR (1) KR101164694B1 (enExample)
CN (1) CN1898255B (enExample)
AR (1) AR046775A1 (enExample)
AU (1) AU2004309054B2 (enExample)
BR (1) BRPI0418047B8 (enExample)
CA (1) CA2550693C (enExample)
DK (1) DK1723156T3 (enExample)
ES (1) ES2528716T3 (enExample)
IL (1) IL176472A (enExample)
IN (2) IN2012DN02546A (enExample)
PL (1) PL1723156T3 (enExample)
WO (1) WO2005063780A1 (enExample)
ZA (1) ZA200605471B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7678920B2 (en) * 2004-04-08 2010-03-16 Dow Agrosciences Llc Insecticidal N-substituted sulfoximines
US7488828B2 (en) * 2004-06-25 2009-02-10 Dow Agrosciences Llc Process for the preparation of 4-trifluoromethyl-2(1H)-pyridinone
TW201309635A (zh) * 2006-02-10 2013-03-01 Dow Agrosciences Llc 殺蟲性之ｎ-取代（６-鹵烷基吡啶-３-基）烷基磺醯亞胺（二）
TWI381811B (zh) * 2006-06-23 2013-01-11 Dow Agrosciences Llc 用以防治可抵抗一般殺蟲劑之昆蟲的方法
MX2009002302A (es) * 2006-09-01 2009-03-13 Dow Agrosciences Llc Sulfoximinas de (2-sustituido-1,3-tiazol) alquilo n-sustituidas insecticidas.
TWI387585B (zh) * 2006-09-01 2013-03-01 Dow Agrosciences Llc 殺蟲性之ｎ-取代（雜芳基）烷基烴基硫亞胺
TWI395737B (zh) * 2006-11-08 2013-05-11 Dow Agrosciences Llc 作為殺蟲劑之雜芳基（取代的）烷基ｎ-取代的磺醯亞胺
US7709648B2 (en) * 2007-02-09 2010-05-04 Dow Agrosciences Llc Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines
AR066366A1 (es) * 2007-05-01 2009-08-12 Dow Agrosciences Llc Mezclas sinergicas plaguicidas
ATE523083T1 (de) * 2007-07-20 2011-09-15 Dow Agrosciences Llc Erhöhte pflanzenvitalität
ES2593116T3 (es) 2008-03-03 2016-12-05 Dow Agrosciences Llc Pesticidas
CN102875548A (zh) * 2011-07-14 2013-01-16 中国科学院大连化学物理研究所 一类基于肟的通过[2+2+2]环加成合成吡啶衍生物的方法
EP2607343A1 (en) 2011-12-22 2013-06-26 Solvay Sa Process for the manufacture of halogenated precursors of alkenones and of alkenones
WO2018099812A1 (en) * 2016-12-01 2018-06-07 Syngenta Participations Ag Pesticidally active heterocyclic derivatives with sulfur containing substituents
WO2020139734A1 (en) * 2018-12-27 2020-07-02 Dow Agrosciences Llc Preparation of sulfonamide herbicide process intermediates
JP7489390B2 (ja) * 2018-12-27 2024-05-23 コルテバ アグリサイエンス エルエルシー スルホンアミド除草剤プロセス中間生成物の調製
CN115286568B (zh) * 2022-08-24 2023-12-12 常州沃腾化工科技有限公司 一种2-羟基-4-三氟甲基吡啶的制备方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002030901A1 (en) 2000-10-10 2002-04-18 Boehringer Ingelheim Chemicals, Inc. Process for making 3-amino-2-chloro-4-methylpyridine

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE611728A (fr) * 1960-07-12 1962-06-19 American Cyanamid Co Perfectionnements aux compositions contenant des antibiotiques à base de tétracycline
US3993656A (en) * 1974-11-19 1976-11-23 Merck & Co., Inc. 1,8-Naphthyridine compounds
JPS5221196A (en) * 1975-08-12 1977-02-17 Fujio Hashimoto Device for removing red tide
JPS53127490A (en) * 1977-04-13 1978-11-07 Yamanouchi Pharmaceut Co Ltd Novel nitrogen-containing heterocyclic compound
JPS53121764A (en) * 1977-03-31 1978-10-24 Yamanouchi Pharmaceut Co Ltd Heterocyclic compounds and process for their preparation
JPS5384990A (en) * 1976-12-29 1978-07-26 Yamanouchi Pharmaceut Co Ltd Novel nitrogen-containing heterocyclic compound and its preparation
JPS55104266A (en) * 1979-02-02 1980-08-09 Yamanouchi Pharmaceut Co Ltd Novel pyridone derivative
JPS6210087A (ja) * 1985-07-03 1987-01-19 Shionogi & Co Ltd ４，７−ジヒドロチエノ〔２，３−ｂ〕ピリジン誘導体，その製造法および循環器系疾患治療剤
JPS6413065A (en) * 1987-07-06 1989-01-17 Mitsubishi Chem Ind Peptide derivative of beta-chloro-l-(z)- dehydroglutamic acid
DK177191D0 (da) * 1991-10-23 1991-10-23 Novo Nordisk As Heterocyclic compounds and their preparation and use
US5391745A (en) * 1992-07-23 1995-02-21 Sloan-Kettering Institute For Cancer Research Methods of preparation of camptothecin analogs
CZ297521B6 (cs) 1996-09-24 2007-01-03 Dow Agrosciences Llc N-([1,2,4]triazoloazinyl)benzensulfonamidové a pyridinsulfonamidové sloučeniny a jejich použití jako herbicidy
CN1312807A (zh) * 1998-06-19 2001-09-12 希龙公司 糖元合成酶激酶3的抑制剂
JP2004504300A (ja) * 2000-07-18 2004-02-12 ビーエーエスエフ　アクチェンゲゼルシャフト １−アリール−４−ハロアルキル−２−［１ｈ］ピリドン類
US7488828B2 (en) * 2004-06-25 2009-02-10 Dow Agrosciences Llc Process for the preparation of 4-trifluoromethyl-2(1H)-pyridinone

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002030901A1 (en) 2000-10-10 2002-04-18 Boehringer Ingelheim Chemicals, Inc. Process for making 3-amino-2-chloro-4-methylpyridine

Also Published As

Publication number Publication date
ZA200605471B (en) 2007-11-28
JP2007519625A (ja) 2007-07-19
US7687632B2 (en) 2010-03-30
AR046775A1 (es) 2005-12-21
ES2528716T3 (es) 2015-02-12
AU2004309054A1 (en) 2005-07-14
AU2004309054B2 (en) 2010-07-08
BRPI0418047B1 (pt) 2013-12-31
JP5160092B2 (ja) 2013-03-13
BRPI0418047B8 (pt) 2022-06-28
CA2550693A1 (en) 2005-07-14
JP2012214487A (ja) 2012-11-08
EP1723156B1 (en) 2015-01-21
EP1723156A1 (en) 2006-11-22
IL176472A0 (en) 2006-10-05
IL176472A (en) 2010-11-30
IN2012DN02545A (enExample) 2015-07-17
US20070249837A1 (en) 2007-10-25
JP2013047245A (ja) 2013-03-07
PL1723156T3 (pl) 2015-07-31
CA2550693C (en) 2013-07-30
IN2012DN02546A (enExample) 2015-08-28
CN1898255A (zh) 2007-01-17
CN1898255B (zh) 2010-06-09
WO2005063780A1 (en) 2005-07-14
BRPI0418047A (pt) 2007-04-17
KR20060128896A (ko) 2006-12-14
DK1723156T3 (en) 2015-04-27

Similar Documents

Publication Publication Date Title
KR101164694B1 (ko) 피리딘 유도체의 제조 방법
EP1071745B1 (en) Process for synthesizing cox-2 inhibitors
EP2368879B1 (en) 2,5-disubstituted pyridines for the preparation of 2-substituted 5-(1-alkylthio)-alkyl-pyridines
IE59324B1 (en) Preparation of substituted and disubstituted pyridine-2,3-dicarboxylate esters
WO2013090547A1 (en) Malonic acid di-salts and a method for preparing malonyl dihalides
JP5077969B2 (ja) ２−置換５−（１−アルキルチオ）アルキルピリジンの調製方法
KR20150093799A (ko) 4-아미노-5-플루오로-3-클로로-6-(치환된)피콜리네이트의제조 방법
IL290169B1 (en) Process and intermediates for the preparation of pyroxasulfone
US4824954A (en) Process for preparation of substituted pyridines
MXPA06007401A (es) Proceso para la preparacion de derivados de piridina
JPH04243875A (ja) ２−フェニル−６−（ピリミジン−２−イル）ピリジン化合物の製造方法、中間体化合物及び中間体化合物の製造方法
HK1031399B (en) Process for synthesizing cox-2 inhibitors
ZA200100474B (en) 3 substituted pyridine compounds and related synthesis.
HK1174028A (en) Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines
HK1136557B (en) Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines
HK1139402B (en) Process for the preparation of 2-substituted-5-(1-alkylthio) alkylpyridines

Legal Events

Date Code Title Description
PA0105 International application

Patent event date: 20060623

Patent event code: PA01051R01D

Comment text: International Patent Application

PG1501 Laying open of application
A201 Request for examination
PA0201 Request for examination

Patent event code: PA02012R01D

Patent event date: 20091221

Comment text: Request for Examination of Application

PE0902 Notice of grounds for rejection

Comment text: Notification of reason for refusal

Patent event date: 20110801

Patent event code: PE09021S01D

E701 Decision to grant or registration of patent right
PE0701 Decision of registration

Patent event code: PE07011S01D

Comment text: Decision to Grant Registration

Patent event date: 20120430

GRNT Written decision to grant
PR0701 Registration of establishment

Comment text: Registration of Establishment

Patent event date: 20120704

Patent event code: PR07011E01D

PR1002 Payment of registration fee

Payment date: 20120704

End annual number: 3

Start annual number: 1

PG1601 Publication of registration
J202 Request for trial for correction [limitation]
PJ0202 Trial for correction

Comment text: Request for Trial

Patent event date: 20130503

Patent event code: PJ02022R01D

Comment text: Registration of Establishment

Patent event date: 20120704

Patent event code: PJ02021E01I

Appeal kind category: Correction

Decision date: 20130613

Request date: 20130503

Appeal identifier: 2013105000045

J301 Trial decision

Free format text: TRIAL DECISION FOR CORRECTION REQUESTED 20130503

Effective date: 20130613

PJ1301 Trial decision

Patent event code: PJ13011S03D

Patent event date: 20130613

Comment text: Trial Decision on Correction (Patent, Utility Model)

Appeal kind category: Correction

Request date: 20130503

Decision date: 20130613

Appeal identifier: 2013105000045

PG1701 Publication of correction

Publication date: 20140107

FPAY Annual fee payment

Payment date: 20150619

Year of fee payment: 4

PR1001 Payment of annual fee

Payment date: 20150619

Start annual number: 4

End annual number: 4

FPAY Annual fee payment

Payment date: 20160616

Year of fee payment: 5

PR1001 Payment of annual fee

Payment date: 20160616

Start annual number: 5

End annual number: 5

FPAY Annual fee payment

Payment date: 20170616

Year of fee payment: 6

PR1001 Payment of annual fee

Payment date: 20170616

Start annual number: 6

End annual number: 6

PR1001 Payment of annual fee

Payment date: 20180615

Start annual number: 7

End annual number: 7

FPAY Annual fee payment

Payment date: 20190617

Year of fee payment: 8

PR1001 Payment of annual fee

Payment date: 20190617

Start annual number: 8

End annual number: 8

PR1001 Payment of annual fee

Payment date: 20200618

Start annual number: 9

End annual number: 9

PR1001 Payment of annual fee

Payment date: 20210617

Start annual number: 10

End annual number: 10

PR1001 Payment of annual fee

Payment date: 20220615

Start annual number: 11

End annual number: 11

PR1001 Payment of annual fee

Payment date: 20230703

Start annual number: 12

End annual number: 12

PR1001 Payment of annual fee

Payment date: 20240627

Start annual number: 13

End annual number: 13

PC1801 Expiration of term

Termination date: 20250622

Termination category: Expiration of duration