JP4881476B2 - ピリジルピペリジン・オレキシン受容体アンタゴニスト - Google Patents

ピリジルピペリジン・オレキシン受容体アンタゴニスト Download PDF

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JP4881476B2
JP4881476B2 JP2010509380A JP2010509380A JP4881476B2 JP 4881476 B2 JP4881476 B2 JP 4881476B2 JP 2010509380 A JP2010509380 A JP 2010509380A JP 2010509380 A JP2010509380 A JP 2010509380A JP 4881476 B2 JP4881476 B2 JP 4881476B2
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JP2010528011A (ja
JP2010528011A5 (enExample
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ブレスリン,マイケル,ジェイ
コールマン,ポール,ジェイ
コックス,クリストファー,ディー
シュライヤー,ジョン,ディー
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Merck and Co Inc
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Merck and Co Inc
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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
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    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
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JP2010509380A 2007-05-23 2008-05-22 ピリジルピペリジン・オレキシン受容体アンタゴニスト Expired - Fee Related JP4881476B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US93145807P 2007-05-23 2007-05-23
US60/931,458 2007-05-23
PCT/US2008/006563 WO2008147518A1 (en) 2007-05-23 2008-05-22 Pyridyl piperidine orexin receptor antagonists

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JP2011229710A Division JP5639564B2 (ja) 2007-05-23 2011-10-19 ピリジルピペリジン・オレキシン受容体アンタゴニスト

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JP2011520966A (ja) * 2008-05-22 2011-07-21 メルク・シャープ・エンド・ドーム・コーポレイション オレキシン受容体アンタゴニストの調製のための方法

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