JP2025516005A5 - - Google Patents

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Publication number
JP2025516005A5
JP2025516005A5 JP2024563159A JP2024563159A JP2025516005A5 JP 2025516005 A5 JP2025516005 A5 JP 2025516005A5 JP 2024563159 A JP2024563159 A JP 2024563159A JP 2024563159 A JP2024563159 A JP 2024563159A JP 2025516005 A5 JP2025516005 A5 JP 2025516005A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
alkyl
isomer
acceptable salt
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024563159A
Other languages
English (en)
Japanese (ja)
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JP2025516005A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/019879 external-priority patent/WO2023211990A1/en
Publication of JP2025516005A publication Critical patent/JP2025516005A/ja
Publication of JP2025516005A5 publication Critical patent/JP2025516005A5/ja
Pending legal-status Critical Current

Links

JP2024563159A 2022-04-25 2023-04-25 疼痛の処置のためのnav1.8の二環式複素環アミド阻害剤 Pending JP2025516005A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN202211024240 2022-04-25
IN202211024240 2022-04-25
IN202311013223 2023-02-27
IN202311013223 2023-02-27
PCT/US2023/019879 WO2023211990A1 (en) 2022-04-25 2023-04-25 Bicyclic heterocyclic amide inhibitors of na v1.8 for the treatment of pain

Publications (2)

Publication Number Publication Date
JP2025516005A JP2025516005A (ja) 2025-05-23
JP2025516005A5 true JP2025516005A5 (enExample) 2026-03-17

Family

ID=86469337

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024563159A Pending JP2025516005A (ja) 2022-04-25 2023-04-25 疼痛の処置のためのnav1.8の二環式複素環アミド阻害剤

Country Status (16)

Country Link
EP (1) EP4514789A1 (enExample)
JP (1) JP2025516005A (enExample)
KR (1) KR20250006217A (enExample)
CN (1) CN119585247A (enExample)
AU (1) AU2023263309A1 (enExample)
CA (1) CA3256486A1 (enExample)
CL (1) CL2024003258A1 (enExample)
CO (1) CO2024015763A2 (enExample)
CR (1) CR20240512A (enExample)
DO (1) DOP2024000215A (enExample)
GE (1) GEAP202516637A (enExample)
IL (1) IL316433A (enExample)
JO (1) JOP20240238A1 (enExample)
MX (1) MX2024013065A (enExample)
PE (1) PE20251183A1 (enExample)
WO (1) WO2023211990A1 (enExample)

Families Citing this family (6)

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Publication number Priority date Publication date Assignee Title
CN117586180A (zh) 2022-08-12 2024-02-23 广州费米子科技有限责任公司 用作电压-门控钠通道抑制剂的化合物
AU2024393245A1 (en) 2023-12-07 2026-06-18 Vertex Pharmaceuticals Incorporated Dosing regimens and formulations of suzetrigine for use in the treatment of acute and chronic pain
TW202547515A (zh) * 2024-04-30 2025-12-16 大陸商江蘇恆瑞醫藥股份有限公司 芳香環類化合物、其製備方法及其在醫藥上的應用
WO2026001999A1 (zh) * 2024-06-25 2026-01-02 江苏恒瑞医药股份有限公司 芳香环类化合物、其制备方法及其在医药上的应用
WO2026021423A1 (zh) * 2024-07-23 2026-01-29 成都康弘药业集团股份有限公司 一种合成Nav1.8抑制剂的中间体,其制备方法和用途
WO2026030525A1 (en) 2024-07-31 2026-02-05 Vertex Pharmaceuticals Incorporated Zilvetrigine dosage forms and dosing regimens for treating pain

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