JP2024529068A5 - - Google Patents

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Publication number
JP2024529068A5
JP2024529068A5 JP2024507166A JP2024507166A JP2024529068A5 JP 2024529068 A5 JP2024529068 A5 JP 2024529068A5 JP 2024507166 A JP2024507166 A JP 2024507166A JP 2024507166 A JP2024507166 A JP 2024507166A JP 2024529068 A5 JP2024529068 A5 JP 2024529068A5
Authority
JP
Japan
Prior art keywords
group
cancer
heterocyclyl
general formula
compound represented
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024507166A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024529068A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2022/111395 external-priority patent/WO2023016484A1/zh
Publication of JP2024529068A publication Critical patent/JP2024529068A/ja
Publication of JP2024529068A5 publication Critical patent/JP2024529068A5/ja
Pending legal-status Critical Current

Links

JP2024507166A 2021-08-10 2022-08-10 スルファミド誘導体、その調製方法及びその医薬的使用 Pending JP2024529068A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
CN202110913249 2021-08-10
CN202110913249.1 2021-08-10
CN202111142090.4 2021-09-28
CN202111142090 2021-09-28
CN202111500231 2021-12-09
CN202111500231.5 2021-12-09
PCT/CN2022/111395 WO2023016484A1 (zh) 2021-08-10 2022-08-10 磺酰胺衍生物、其制备方法及其在医药上的应用

Publications (2)

Publication Number Publication Date
JP2024529068A JP2024529068A (ja) 2024-08-01
JP2024529068A5 true JP2024529068A5 (https=) 2025-08-19

Family

ID=85200573

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024507166A Pending JP2024529068A (ja) 2021-08-10 2022-08-10 スルファミド誘導体、その調製方法及びその医薬的使用

Country Status (10)

Country Link
US (1) US20250145637A1 (https=)
EP (1) EP4385989A4 (https=)
JP (1) JP2024529068A (https=)
KR (1) KR20240046530A (https=)
CN (1) CN117597341A (https=)
AU (1) AU2022325367A1 (https=)
CA (1) CA3228411A1 (https=)
MX (1) MX2024001777A (https=)
TW (1) TW202321263A (https=)
WO (1) WO2023016484A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN118556053A (zh) 2021-11-16 2024-08-27 英矽智能科技知识产权有限公司 赖氨酸乙酰基转移酶6a(kat6a)抑制剂及其用途
WO2023114710A1 (en) * 2021-12-13 2023-06-22 Aurigene Oncology Limited Fused benzoisoxazolyl compounds as kat6a inhibitors
CN116621859A (zh) * 2022-02-18 2023-08-22 山东轩竹医药科技有限公司 三并环类kat6抑制剂
KR20250006833A (ko) 2022-03-28 2025-01-13 아이소스테릭스, 인코포레이티드 라이신 아세틸 전이효소의 myst 계열의 억제제
KR20250143814A (ko) * 2023-02-10 2025-10-02 지앙수 헨그루이 파마슈티컬스 컴퍼니 리미티드 설폰아미드 유도체 결정 형태 및 이의 제조 방법
WO2024189598A2 (en) 2023-03-16 2024-09-19 Olema Pharmaceuticals, Inc. Acylsulfonamide kat6a inhibitors
CN120981721A (zh) * 2023-03-30 2025-11-18 辉瑞大药厂 Kat6a作为用kat6a抑制剂治疗的预测性生物标志物和相关治疗方法
AU2024290895A1 (en) 2023-07-04 2026-01-29 Shanghai Qilu Pharmaceutical Research And Development Centre Ltd. Kat6 inhibitor
WO2025098417A1 (zh) * 2023-11-08 2025-05-15 再和医药科技(苏州)有限公司 磺酰胺类化合物及其应用
WO2025101942A1 (en) * 2023-11-10 2025-05-15 Prelude Therapeutics Incorporated Kat6 targeting compounds
AR134697A1 (es) * 2023-12-18 2026-03-04 Ideaya Biosciences Inc Compuestos químicos y sus usos

Family Cites Families (19)

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US5750542A (en) * 1993-09-28 1998-05-12 Pfizer Benzisoxazole and benzisothizole derivatives as cholinesterase inhibitors
HU225047B1 (en) * 1991-03-28 2006-05-29 Eisai Co Ltd Heterocyclic-piperidin-derivatives, pharmaceutical compositions containing them and process for their production
WO2002074746A1 (en) * 2001-03-16 2002-09-26 Yamanouchi Pharmaceutical Co., Ltd. Benzazepine derivatives
KR100965021B1 (ko) * 2002-02-22 2010-06-21 바이엘 파마슈티칼스 코포레이션 과다증식성 질환 치료에 유용한 벤조푸란 및 벤조티오펜유도체
AU2006281803B9 (en) * 2005-08-18 2013-05-30 Genmab A/S Therapy with CD4 binding peptides and radiation
CN105492430B (zh) * 2013-03-15 2017-10-10 基因泰克公司 取代的苯并噁唑及其使用方法
WO2015102929A1 (en) * 2013-12-30 2015-07-09 Novartis Ag Tricyclic sulfonamide derivatives
JP6568926B2 (ja) * 2014-03-20 2019-08-28 カペラ セラピューティクス,インコーポレーテッド 癌の治療のためのerbbチロシンキナーゼ阻害剤としてのベンゾイミダゾール誘導体
GB201510019D0 (en) 2015-06-09 2015-07-22 Cancer Therapeutics Crc Pty Ltd Compounds
WO2017218960A1 (en) 2016-06-17 2017-12-21 Fronthera U.S. Pharmaceuticals Llc Hemoglobin modifier compounds and uses thereof
GB201713962D0 (en) 2017-08-31 2017-10-18 Ctxt Pty Ltd Compounds
MX2020007131A (es) 2017-11-29 2021-01-08 Epizyme Inc Inhibidores de histona acetiltransferasa de la familia myst.
GB201810092D0 (en) 2018-06-20 2018-08-08 Ctxt Pty Ltd Compounds
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KR20210057767A (ko) * 2018-09-07 2021-05-21 치아타이 티안큉 파마수티컬 그룹 주식회사 Crbn단백질에 작용하는 삼환식 화합물
EA202092908A1 (ru) 2018-09-28 2021-05-14 Праксис Пресижн Медсинз, Инк. Модуляторы ионных каналов
CA3137472A1 (en) 2019-04-25 2020-10-29 Bayer Aktiengesellschaft Acyl sulfonamides for treating cancer
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US12545669B2 (en) 2019-06-19 2026-02-10 Pfizer Inc. Cycloalkyl and heterocycloalkyl benzisoxazole sulfonamide derivatives

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