JP2023537501A5 - - Google Patents
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- Publication number
- JP2023537501A5 JP2023537501A5 JP2023507783A JP2023507783A JP2023537501A5 JP 2023537501 A5 JP2023537501 A5 JP 2023537501A5 JP 2023507783 A JP2023507783 A JP 2023507783A JP 2023507783 A JP2023507783 A JP 2023507783A JP 2023537501 A5 JP2023537501 A5 JP 2023537501A5
- Authority
- JP
- Japan
- Prior art keywords
- compound according
- group
- alkyl
- section
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2020/107437 | 2020-08-06 | ||
| CN2020107437 | 2020-08-06 | ||
| CNPCT/CN2021/073958 | 2021-01-27 | ||
| CN2021073958 | 2021-01-27 | ||
| PCT/CN2021/111193 WO2022028572A1 (en) | 2020-08-06 | 2021-08-06 | Heterocyclic glp-1 agonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023537501A JP2023537501A (ja) | 2023-09-01 |
| JP2023537501A5 true JP2023537501A5 (https=) | 2024-08-14 |
Family
ID=80117080
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023507783A Pending JP2023537501A (ja) | 2020-08-06 | 2021-08-06 | ヘテロ環ｇｌｐ－１アゴニスト |
Country Status (23)
| Country | Link |
|---|---|
| US (3) | US11897851B2 (https=) |
| EP (1) | EP4192831B1 (https=) |
| JP (1) | JP2023537501A (https=) |
| KR (1) | KR20230053620A (https=) |
| CN (1) | CN116323599A (https=) |
| AU (1) | AU2021323253A1 (https=) |
| CA (1) | CA3190163A1 (https=) |
| CL (2) | CL2023000374A1 (https=) |
| CO (1) | CO2023001263A2 (https=) |
| CR (1) | CR20230066A (https=) |
| DK (1) | DK4192831T3 (https=) |
| DO (1) | DOP2023000023A (https=) |
| FI (1) | FI4192831T3 (https=) |
| HR (1) | HRP20251653T1 (https=) |
| IL (1) | IL300155A (https=) |
| LT (1) | LT4192831T (https=) |
| MX (1) | MX2023001311A (https=) |
| PE (1) | PE20231181A1 (https=) |
| PL (1) | PL4192831T3 (https=) |
| PT (1) | PT4192831T (https=) |
| SI (1) | SI4192831T1 (https=) |
| TW (1) | TW202220973A (https=) |
| WO (1) | WO2022028572A1 (https=) |
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| JP2023537501A (ja) | 2020-08-06 | 2023-09-01 | ガシャーブラム・バイオ・インコーポレイテッド | ヘテロ環ｇｌｐ－１アゴニスト |
| EP4204415A4 (en) | 2020-08-28 | 2025-03-26 | Gasherbrum Bio, Inc. | HETEROCYCLIC GLP-1 AGONISTS |
| JP7772778B2 (ja) | 2021-03-24 | 2025-11-18 | 塩野義製薬株式会社 | 縮合環を有するｇｌｐ－１受容体作動薬を含有する医薬組成物 |
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| JP2025506474A (ja) * | 2022-02-09 | 2025-03-11 | ガシャーブラム・バイオ・インコーポレイテッド | ヘテロ環ｇｌｐ－１アゴニスト |
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| WO2022219495A1 (en) * | 2021-04-12 | 2022-10-20 | Novartis Ag | 2-((4-((s)-2-(4-chloro-2-fluorophenyl)-2-methylbenzo[d][1,3]dioxol-4-yl)piperidin-1-yl)methyl)-1-(((s)-oxetan-2-yl)methyl)-1h-imidazole derivatives as activators of the glp1 receptor for the treatment of obesity |
| CN117177970A (zh) * | 2021-04-30 | 2023-12-05 | 上海翰森生物医药科技有限公司 | 多环类衍生物调节剂、其制备方法和应用 |
| CN115594669B (zh) | 2021-07-09 | 2024-11-05 | 深圳信立泰药业股份有限公司 | 一种并环类衍生物及其制备方法和医药用途 |
| CN113480534B (zh) | 2021-07-23 | 2022-05-13 | 广州必贝特医药股份有限公司 | 苯并咪唑或氮杂苯并咪唑-6-羧酸类化合物及其应用 |
| EP4469444A4 (en) | 2022-01-24 | 2026-01-07 | Gasherbrum Bio Inc | GLP-1 HETEROCYCLIC AGONISTS |
| US20250177362A1 (en) | 2022-02-09 | 2025-06-05 | Gasherbrum Bio, Inc. | Heterocyclic glp-1 agonists |
| JP2025506474A (ja) | 2022-02-09 | 2025-03-11 | ガシャーブラム・バイオ・インコーポレイテッド | ヘテロ環ｇｌｐ－１アゴニスト |
| US20250206757A1 (en) | 2022-03-21 | 2025-06-26 | Gasherbrum Bio, Inc. | 5,8-dihydro-1,7-naphthyridine derivatives as glp-1 agonists for the treatment of diabetes |
| US20250250269A1 (en) | 2022-04-14 | 2025-08-07 | Gasherbrum Bio, Inc. | Heterocyclic glp-1 agonists |
| CN114716423A (zh) | 2022-05-20 | 2022-07-08 | 中国科学院上海药物研究所 | 5,6-二氢-1,2,4-三嗪类化合物及其作为glp-1受体激动剂的药学用途 |
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2021
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2025
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