JP2023507399A5 - - Google Patents
Info
- Publication number
- JP2023507399A5 JP2023507399A5 JP2022537301A JP2022537301A JP2023507399A5 JP 2023507399 A5 JP2023507399 A5 JP 2023507399A5 JP 2022537301 A JP2022537301 A JP 2022537301A JP 2022537301 A JP2022537301 A JP 2022537301A JP 2023507399 A5 JP2023507399 A5 JP 2023507399A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- process according
- dichlorophenyl
- acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962951691P | 2019-12-20 | 2019-12-20 | |
| US62/951,691 | 2019-12-20 | ||
| US202063120426P | 2020-12-02 | 2020-12-02 | |
| US63/120,426 | 2020-12-02 | ||
| PCT/IB2020/062040 WO2021124158A1 (en) | 2019-12-20 | 2020-12-16 | Efficient process for making 6-carboxy benzoxazole derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023507399A JP2023507399A (ja) | 2023-02-22 |
| JP2023507399A5 true JP2023507399A5 (https=) | 2023-12-12 |
Family
ID=73856234
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022537301A Pending JP2023507399A (ja) | 2019-12-20 | 2020-12-16 | ６－カルボキシベンゾオキサゾール誘導体を作製するための効率的なプロセス |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US12410145B2 (https=) |
| EP (1) | EP4077287B1 (https=) |
| JP (1) | JP2023507399A (https=) |
| KR (1) | KR20220114626A (https=) |
| CN (1) | CN115135639B (https=) |
| AU (1) | AU2020406455B2 (https=) |
| BR (1) | BR112022012097A2 (https=) |
| CA (1) | CA3165298A1 (https=) |
| ES (1) | ES3055912T3 (https=) |
| HR (1) | HRP20251570T1 (https=) |
| IL (1) | IL294115A (https=) |
| MX (1) | MX2022007787A (https=) |
| TW (1) | TWI771827B (https=) |
| WO (1) | WO2021124158A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4077287B1 (en) | 2019-12-20 | 2025-11-19 | Pfizer Ireland Pharmaceuticals Unlimited Company | Efficient process for making 6-carboxy benzoxazole derivatives |
| KR102657823B1 (ko) * | 2022-03-10 | 2024-04-16 | 고려대학교 산학협력단 | 타파미디스의 신규 합성법 |
| US11970468B1 (en) | 2023-10-23 | 2024-04-30 | King Faisal University | 2-(benzo[d]oxazol-2-yl)-N′-(3,5-dichlorobenzoyloxy)acetimidamide as an antimicrobial compound |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5222642A (en) | 1975-08-14 | 1977-02-21 | Kawasaki Heavy Ind Ltd | Power generation device by hot water |
| GB8703975D0 (en) | 1987-02-20 | 1987-03-25 | Wellcome Found | Pesticidal compounds |
| GB8809316D0 (en) * | 1987-05-11 | 1988-05-25 | Ici America Inc | Heterocyclic ketones |
| CA2800237C (en) * | 2002-12-19 | 2016-05-17 | The Scripps Research Institute | Compositions and methods for stabilizing transthyretin and inhibiting transthyretin misfolding |
| JP5419545B2 (ja) | 2009-05-25 | 2014-02-19 | 株式会社トクヤマ | オルトエステル化合物の製造方法 |
| US8168683B2 (en) | 2009-10-15 | 2012-05-01 | E. I. Du Pont De Nemours And Company | Fluorinated vinylidene cationic surfactant |
| TWI550071B (zh) * | 2011-03-25 | 2016-09-21 | 捷恩智股份有限公司 | 原酸酯化合物、液晶組成物及液晶顯示元件 |
| RU2586330C2 (ru) * | 2011-09-16 | 2016-06-10 | Пфайзер Инк. | Твердые формы ингибитора диссоциации транстиретина |
| US9499527B2 (en) * | 2012-05-10 | 2016-11-22 | Cellix Bio Private Limited | Compositions and methods for the treatment of familial amyloid polyneuropathy |
| PT4349406T (pt) * | 2014-09-08 | 2026-02-04 | Pfizer | Formas sólidas cristalinas de 6-carboxi-2-(3,5-diclorofenil)-benzoxazol para utilização como medicamento |
| CN107344927A (zh) * | 2016-05-05 | 2017-11-14 | 苏州晶云药物科技有限公司 | Tafamidis葡甲胺盐的晶型E及其制备方法和用途 |
| US10766893B2 (en) * | 2017-12-20 | 2020-09-08 | H. Lundbeck A/S | 1H-pyrazolo[4,3-b]pyridines as PDE1 inhibitors |
| EP4077287B1 (en) | 2019-12-20 | 2025-11-19 | Pfizer Ireland Pharmaceuticals Unlimited Company | Efficient process for making 6-carboxy benzoxazole derivatives |
-
2020
- 2020-12-16 EP EP20828342.4A patent/EP4077287B1/en active Active
- 2020-12-16 WO PCT/IB2020/062040 patent/WO2021124158A1/en not_active Ceased
- 2020-12-16 CA CA3165298A patent/CA3165298A1/en active Pending
- 2020-12-16 TW TW109144467A patent/TWI771827B/zh active
- 2020-12-16 CN CN202080096991.1A patent/CN115135639B/zh active Active
- 2020-12-16 JP JP2022537301A patent/JP2023507399A/ja active Pending
- 2020-12-16 BR BR112022012097A patent/BR112022012097A2/pt not_active Application Discontinuation
- 2020-12-16 MX MX2022007787A patent/MX2022007787A/es unknown
- 2020-12-16 HR HRP20251570TT patent/HRP20251570T1/hr unknown
- 2020-12-16 KR KR1020227024529A patent/KR20220114626A/ko not_active Withdrawn
- 2020-12-16 US US17/757,740 patent/US12410145B2/en active Active
- 2020-12-16 ES ES20828342T patent/ES3055912T3/es active Active
- 2020-12-16 IL IL294115A patent/IL294115A/en unknown
- 2020-12-16 AU AU2020406455A patent/AU2020406455B2/en active Active
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