JP2022527080A5 - - Google Patents

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Publication number
JP2022527080A5
JP2022527080A5 JP2021557368A JP2021557368A JP2022527080A5 JP 2022527080 A5 JP2022527080 A5 JP 2022527080A5 JP 2021557368 A JP2021557368 A JP 2021557368A JP 2021557368 A JP2021557368 A JP 2021557368A JP 2022527080 A5 JP2022527080 A5 JP 2022527080A5
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JP
Japan
Prior art keywords
methanone
imidazole
piperidine
phenyl
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021557368A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022527080A (ja
JP7454589B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/024969 external-priority patent/WO2020198478A1/en
Publication of JP2022527080A publication Critical patent/JP2022527080A/ja
Publication of JP2022527080A5 publication Critical patent/JP2022527080A5/ja
Application granted granted Critical
Publication of JP7454589B2 publication Critical patent/JP7454589B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021557368A 2019-03-28 2020-03-26 セロトニン5-ht2b阻害化合物 Active JP7454589B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962825051P 2019-03-28 2019-03-28
US62/825,051 2019-03-28
PCT/US2020/024969 WO2020198478A1 (en) 2019-03-28 2020-03-26 Serotonin 5-ht2b inhibitory compounds

Publications (3)

Publication Number Publication Date
JP2022527080A JP2022527080A (ja) 2022-05-30
JP2022527080A5 true JP2022527080A5 (https=) 2022-10-25
JP7454589B2 JP7454589B2 (ja) 2024-03-22

Family

ID=70775466

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021557368A Active JP7454589B2 (ja) 2019-03-28 2020-03-26 セロトニン5-ht2b阻害化合物

Country Status (13)

Country Link
US (2) US12240827B2 (https=)
EP (1) EP3947360B1 (https=)
JP (1) JP7454589B2 (https=)
CN (1) CN113631548B (https=)
AU (1) AU2020245614B2 (https=)
BR (1) BR112021019314A2 (https=)
CA (1) CA3134952C (https=)
DK (1) DK3947360T3 (https=)
ES (1) ES2991167T3 (https=)
FI (1) FI3947360T3 (https=)
PL (1) PL3947360T3 (https=)
PT (1) PT3947360T (https=)
WO (1) WO2020198478A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20240027076A (ko) * 2021-07-26 2024-02-29 조에티스 서비시즈 엘엘씨 세로토닌 5-ht2b 억제 화합물

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0515995D0 (en) 2005-08-03 2005-09-07 Sandoz Ag Organic compounds
WO2007097197A1 (ja) * 2006-02-20 2007-08-30 Astellas Pharma Inc. アミド誘導体またはその塩
TWI415845B (zh) 2006-10-03 2013-11-21 Arena Pharm Inc 用於治療與5-ht2a血清素受體相關聯病症之作為5-ht2a血清素受體之調節劑的吡唑衍生物
JP2012512877A (ja) * 2008-12-18 2012-06-07 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング セロトニン5−ht2b受容体阻害剤
US8697739B2 (en) 2010-07-29 2014-04-15 Novartis Ag Bicyclic acetyl-CoA carboxylase inhibitors and uses thereof

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