FI3947360T3 - Serotoniini 5-ht2b:tä estäviä yhdisteitä - Google Patents

Serotoniini 5-ht2b:tä estäviä yhdisteitä Download PDF

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Publication number
FI3947360T3
FI3947360T3 FIEP20726982.0T FI20726982T FI3947360T3 FI 3947360 T3 FI3947360 T3 FI 3947360T3 FI 20726982 T FI20726982 T FI 20726982T FI 3947360 T3 FI3947360 T3 FI 3947360T3
Authority
FI
Finland
Prior art keywords
methanone
imidazol
piperidin
methyl
biphenyl
Prior art date
Application number
FIEP20726982.0T
Other languages
English (en)
Finnish (fi)
Inventor
Richard Ewin
Govindan Subramanian
Jinxia Deng (Nancy)
Original Assignee
Zoetis Services Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zoetis Services Llc filed Critical Zoetis Services Llc
Application granted granted Critical
Publication of FI3947360T3 publication Critical patent/FI3947360T3/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FIEP20726982.0T 2019-03-28 2020-03-26 Serotoniini 5-ht2b:tä estäviä yhdisteitä FI3947360T3 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962825051P 2019-03-28 2019-03-28
PCT/US2020/024969 WO2020198478A1 (en) 2019-03-28 2020-03-26 Serotonin 5-ht2b inhibitory compounds

Publications (1)

Publication Number Publication Date
FI3947360T3 true FI3947360T3 (fi) 2024-10-07

Family

ID=70775466

Family Applications (1)

Application Number Title Priority Date Filing Date
FIEP20726982.0T FI3947360T3 (fi) 2019-03-28 2020-03-26 Serotoniini 5-ht2b:tä estäviä yhdisteitä

Country Status (13)

Country Link
US (2) US12240827B2 (https=)
EP (1) EP3947360B1 (https=)
JP (1) JP7454589B2 (https=)
CN (1) CN113631548B (https=)
AU (1) AU2020245614B2 (https=)
BR (1) BR112021019314A2 (https=)
CA (1) CA3134952C (https=)
DK (1) DK3947360T3 (https=)
ES (1) ES2991167T3 (https=)
FI (1) FI3947360T3 (https=)
PL (1) PL3947360T3 (https=)
PT (1) PT3947360T (https=)
WO (1) WO2020198478A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20240027076A (ko) * 2021-07-26 2024-02-29 조에티스 서비시즈 엘엘씨 세로토닌 5-ht2b 억제 화합물

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0515995D0 (en) 2005-08-03 2005-09-07 Sandoz Ag Organic compounds
WO2007097197A1 (ja) * 2006-02-20 2007-08-30 Astellas Pharma Inc. アミド誘導体またはその塩
TWI415845B (zh) 2006-10-03 2013-11-21 Arena Pharm Inc 用於治療與5-ht2a血清素受體相關聯病症之作為5-ht2a血清素受體之調節劑的吡唑衍生物
JP2012512877A (ja) * 2008-12-18 2012-06-07 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング セロトニン5−ht2b受容体阻害剤
US8697739B2 (en) 2010-07-29 2014-04-15 Novartis Ag Bicyclic acetyl-CoA carboxylase inhibitors and uses thereof

Also Published As

Publication number Publication date
US20220162183A1 (en) 2022-05-26
US12240827B2 (en) 2025-03-04
PL3947360T3 (pl) 2024-11-04
CA3134952A1 (en) 2020-10-01
EP3947360A1 (en) 2022-02-09
AU2020245614A1 (en) 2021-10-14
US20250179046A1 (en) 2025-06-05
JP2022527080A (ja) 2022-05-30
JP7454589B2 (ja) 2024-03-22
DK3947360T3 (da) 2024-08-26
WO2020198478A8 (en) 2021-09-16
ES2991167T3 (es) 2024-12-02
CA3134952C (en) 2023-08-08
BR112021019314A2 (pt) 2021-12-14
CN113631548A (zh) 2021-11-09
CN113631548B (zh) 2023-06-06
EP3947360B1 (en) 2024-08-07
WO2020198478A1 (en) 2020-10-01
AU2020245614B2 (en) 2023-01-19
PT3947360T (pt) 2024-09-20

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