JP2021534095A5 - - Google Patents

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Publication number
JP2021534095A5
JP2021534095A5 JP2021506575A JP2021506575A JP2021534095A5 JP 2021534095 A5 JP2021534095 A5 JP 2021534095A5 JP 2021506575 A JP2021506575 A JP 2021506575A JP 2021506575 A JP2021506575 A JP 2021506575A JP 2021534095 A5 JP2021534095 A5 JP 2021534095A5
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JP
Japan
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unsubstituted
substituted
alkyl
halogen
pharmaceutically acceptable
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JP2021506575A
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English (en)
Japanese (ja)
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JP2021534095A (ja
JP7429988B2 (ja
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Priority claimed from EP18290093.6A external-priority patent/EP3608318A1/en
Priority claimed from EP18213635.8A external-priority patent/EP3670512A1/en
Application filed filed Critical
Priority claimed from PCT/EP2019/071370 external-priority patent/WO2020030761A1/en
Publication of JP2021534095A publication Critical patent/JP2021534095A/ja
Publication of JP2021534095A5 publication Critical patent/JP2021534095A5/ja
Application granted granted Critical
Publication of JP7429988B2 publication Critical patent/JP7429988B2/ja
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JP2021506575A 2018-08-09 2019-08-08 セリンベータ-ラクタマーゼのインヒビターとしてのジアザビシクロオクタノン Active JP7429988B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP18290093.6A EP3608318A1 (en) 2018-08-09 2018-08-09 Diaazabicyclooctanone derivatives as antibacterials
EP18290093.6 2018-08-09
EP18213635.8 2018-12-18
EP18213635.8A EP3670512A1 (en) 2018-12-18 2018-12-18 Diazabicyclooctanones as inhibitors of serine beta-lactamases
PCT/EP2019/071370 WO2020030761A1 (en) 2018-08-09 2019-08-08 Diazabicyclooctanones as inhibitors of serine beta-lactamases

Publications (3)

Publication Number Publication Date
JP2021534095A JP2021534095A (ja) 2021-12-09
JP2021534095A5 true JP2021534095A5 (enExample) 2022-08-18
JP7429988B2 JP7429988B2 (ja) 2024-02-09

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ID=67667824

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JP2021506575A Active JP7429988B2 (ja) 2018-08-09 2019-08-08 セリンベータ-ラクタマーゼのインヒビターとしてのジアザビシクロオクタノン

Country Status (24)

Country Link
US (1) US12378244B2 (enExample)
EP (2) EP4272831A3 (enExample)
JP (1) JP7429988B2 (enExample)
KR (1) KR102790878B1 (enExample)
CN (2) CN117384155A (enExample)
AU (1) AU2019318115B2 (enExample)
BR (1) BR112021002311A2 (enExample)
CA (1) CA3110111A1 (enExample)
DK (1) DK3833665T3 (enExample)
ES (1) ES2960952T3 (enExample)
FI (1) FI3833665T3 (enExample)
HR (1) HRP20231228T1 (enExample)
HU (1) HUE063324T2 (enExample)
IL (1) IL280770B2 (enExample)
LT (1) LT3833665T (enExample)
MX (1) MX2021001564A (enExample)
PL (1) PL3833665T3 (enExample)
RS (1) RS64679B1 (enExample)
SG (1) SG11202101255UA (enExample)
SI (1) SI3833665T1 (enExample)
SM (1) SMT202300354T1 (enExample)
TW (1) TWI764030B (enExample)
WO (1) WO2020030761A1 (enExample)
ZA (1) ZA202100906B (enExample)

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CN111943950B (zh) * 2020-09-10 2022-03-29 山东安信制药有限公司 一种瑞来巴坦的制备方法
US12410166B2 (en) 2021-05-07 2025-09-09 Ningxia Academy Of Agriculture And Forestry Sciences Sulfonylamidine substituted compounds and their use as beta-lactamase inhibitors
CN115448920B (zh) * 2022-10-14 2025-01-03 广州楷石医药有限公司 一种β-内酰胺酶抑制剂及其应用
GB202306833D0 (en) 2023-05-09 2023-06-21 Adjutec Pharma As Therapy
GB202306826D0 (en) 2023-05-09 2023-06-21 Adjutec Pharma As Therapy
CN117700415B (zh) * 2024-02-06 2024-04-30 成都四面体药物研究有限公司 含脲双环化合物、其用途、其制备的药物、其联合用药物及其复方制剂
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WO2026104587A1 (en) 2024-11-13 2026-05-21 Adjutec Pharma As Cyclic boronic acid esters useful as adjuvants in the treatment of bacterial infections

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