JP2021511374A5 - - Google Patents

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Publication number
JP2021511374A5
JP2021511374A5 JP2020560532A JP2020560532A JP2021511374A5 JP 2021511374 A5 JP2021511374 A5 JP 2021511374A5 JP 2020560532 A JP2020560532 A JP 2020560532A JP 2020560532 A JP2020560532 A JP 2020560532A JP 2021511374 A5 JP2021511374 A5 JP 2021511374A5
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JP
Japan
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group
hydrocarbon
heterocyclic
stereoisomer
solvate
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JP2020560532A
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English (en)
Japanese (ja)
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JP7352297B2 (ja
JP2021511374A (ja
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Priority claimed from CN201810044308.4A external-priority patent/CN110041327B/zh
Priority claimed from CN201811517425.4A external-priority patent/CN111303147B/zh
Application filed filed Critical
Priority claimed from PCT/CN2019/071902 external-priority patent/WO2019141179A1/zh
Publication of JP2021511374A publication Critical patent/JP2021511374A/ja
Publication of JP2021511374A5 publication Critical patent/JP2021511374A5/ja
Application granted granted Critical
Publication of JP7352297B2 publication Critical patent/JP7352297B2/ja
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JP2020560532A 2018-01-17 2019-01-16 ピリドン誘導体と、その組成物、並びにそれらが抗ウイルス薬物としての応用 Active JP7352297B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CN201810044308.4 2018-01-17
CN201810044308.4A CN110041327B (zh) 2018-01-17 2018-01-17 吡啶酮衍生物、其组合物及作为抗流感病毒药物的应用
CN201811517425.4A CN111303147B (zh) 2018-12-12 2018-12-12 吡啶酮衍生物、其组合物及作为抗流感病毒药物的应用
CN201811517425.4 2018-12-12
PCT/CN2019/071902 WO2019141179A1 (zh) 2018-01-17 2019-01-16 吡啶酮衍生物、其组合物及作为抗流感病毒药物的应用

Publications (3)

Publication Number Publication Date
JP2021511374A JP2021511374A (ja) 2021-05-06
JP2021511374A5 true JP2021511374A5 (enExample) 2022-03-15
JP7352297B2 JP7352297B2 (ja) 2023-09-28

Family

ID=67301986

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020560532A Active JP7352297B2 (ja) 2018-01-17 2019-01-16 ピリドン誘導体と、その組成物、並びにそれらが抗ウイルス薬物としての応用

Country Status (11)

Country Link
US (1) US11247993B2 (enExample)
EP (1) EP3753936B1 (enExample)
JP (1) JP7352297B2 (enExample)
KR (1) KR102477187B1 (enExample)
CN (4) CN111848615B (enExample)
AU (1) AU2019210414B2 (enExample)
CA (1) CA3088926A1 (enExample)
PH (1) PH12020551264A1 (enExample)
SG (1) SG11202011447UA (enExample)
WO (1) WO2019141179A1 (enExample)
ZA (1) ZA202007143B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2881776T3 (es) 2016-03-08 2021-11-30 Novartis Ag Compuestos tricíclicos útiles para tratar las infecciones por ortomixovirus
JOP20170169A1 (ar) 2016-08-29 2019-01-30 Novartis Ag مركبات بيريدازين ثلاثية الحلقة مندمجة تفيد في علاج العدوى بفيروس أورثوميكسو
CN111386276B (zh) 2017-10-06 2023-06-23 盐野义制药株式会社 制备取代的多环吡啶酮衍生物的立体选择性方法
CN118878544A (zh) * 2018-02-28 2024-11-01 诺华股份有限公司 作为正粘病毒复制抑制剂用于治疗流感的化合物
CN112118891B (zh) * 2019-04-01 2023-10-31 尼坎医疗公司 作为流感病毒复制抑制剂的稠和多环吡啶酮化合物
CN111909174B (zh) * 2019-05-08 2022-01-21 江西彩石医药科技有限公司 吡啶酮衍生物的晶型及制备方法和应用
CN112574170A (zh) * 2019-09-29 2021-03-30 江西东邦药业有限公司 一种二苯并七元环衍生物及其制备方法和应用
WO2021129602A1 (zh) * 2019-12-23 2021-07-01 石家庄迪斯凯威医药科技有限公司 取代的多环化合物及其药物组合物和用途
CN113045589B (zh) * 2019-12-27 2024-08-23 广东东阳光药业股份有限公司 流感病毒复制抑制剂及其用途
CN112898346B (zh) * 2020-01-23 2023-11-10 南京知和医药科技有限公司 水溶性多环化合物及其药物组合物和用途
CN113116899B (zh) * 2020-03-06 2022-12-20 广东众生睿创生物科技有限公司 一种用于治疗流感的药物组合物及含有该药物组合物的制剂
CN111943879A (zh) * 2020-08-03 2020-11-17 南通大学 一种(3s,4r)3-氨基-4(甲氧基甲基)吡咯烷-1-甲酸叔丁酯及其合成方法
CN113583022B (zh) * 2020-08-11 2025-03-18 石家庄迪斯凯威医药科技有限公司 多环化合物及其药物组合物和用途
CN115385932A (zh) * 2021-05-22 2022-11-25 江西彩石医药科技有限公司 吡啶酮衍生物的中间体及其制备方法
KR20250078466A (ko) * 2022-10-08 2025-06-02 스자좡 디스커버리 메디슨 테크놀로지 컴퍼니 리미티드 인플루엔자 바이러스 억제 유도체 및 그 용도
CN117003771B (zh) * 2022-11-09 2024-02-02 石家庄迪斯凯威医药科技有限公司 一种抗流感病毒衍生物及其用途
CN116789556A (zh) * 2023-05-26 2023-09-22 康化(上海)新药研发有限公司 一种含环丙氧基乙胺的制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8927710B2 (en) 2009-06-15 2015-01-06 Shionogi & Co., Ltd. Substituted polycyclic carbamoylpyridone derivative
DK2620436T3 (en) 2010-09-24 2018-07-30 Shionogi & Co Substituted polycyclic carbamoylpyridone derivative prodrug
MX377396B (es) * 2013-09-12 2025-03-10 Janssen Biopharma Inc Compuestos de azapiridona y usos de los mismos.
SG11201708721XA (en) 2015-04-28 2017-11-29 Shionogi & Co Substituted polycyclic pyridone derivative and prodrug thereof
SG11201804348SA (en) * 2015-12-15 2018-06-28 Shionogi & Co Medicine for treating influenza characterized by comprising combination of cap-dependent endonuclease inhibitor with anti-influenza drug
JP6806413B2 (ja) * 2016-02-03 2021-01-06 塩野義製薬株式会社 多環性ピリドン誘導体およびそのプロドラッグ
KR20190018469A (ko) * 2016-08-10 2019-02-22 시오노기세야쿠 가부시키가이샤 치환된 다환성 피리돈 유도체 및 그의 프로드러그를 함유하는 의약 조성물
JOP20170169A1 (ar) 2016-08-29 2019-01-30 Novartis Ag مركبات بيريدازين ثلاثية الحلقة مندمجة تفيد في علاج العدوى بفيروس أورثوميكسو

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