JP2020536870A5 - - Google Patents

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Publication number
JP2020536870A5
JP2020536870A5 JP2020519296A JP2020519296A JP2020536870A5 JP 2020536870 A5 JP2020536870 A5 JP 2020536870A5 JP 2020519296 A JP2020519296 A JP 2020519296A JP 2020519296 A JP2020519296 A JP 2020519296A JP 2020536870 A5 JP2020536870 A5 JP 2020536870A5
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JP
Japan
Prior art keywords
formula
compound
solvent
base
formamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2020519296A
Other languages
English (en)
Japanese (ja)
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JP2020536870A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2018/054661 external-priority patent/WO2019071162A2/en
Publication of JP2020536870A publication Critical patent/JP2020536870A/ja
Publication of JP2020536870A5 publication Critical patent/JP2020536870A5/ja
Withdrawn legal-status Critical Current

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JP2020519296A 2017-10-05 2018-10-05 アルファカルボキサミドピロリジン誘導体の調製方法 Withdrawn JP2020536870A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762568651P 2017-10-05 2017-10-05
US62/568,651 2017-10-05
PCT/US2018/054661 WO2019071162A2 (en) 2017-10-05 2018-10-05 PROCESS FOR THE PREPARATION OF PYRROLIDINE ALPHA-CARBOXAMIDE DERIVATIVES

Publications (2)

Publication Number Publication Date
JP2020536870A JP2020536870A (ja) 2020-12-17
JP2020536870A5 true JP2020536870A5 (https=) 2021-11-25

Family

ID=65995302

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020519296A Withdrawn JP2020536870A (ja) 2017-10-05 2018-10-05 アルファカルボキサミドピロリジン誘導体の調製方法

Country Status (12)

Country Link
US (2) US11192856B2 (https=)
EP (1) EP3691634A4 (https=)
JP (1) JP2020536870A (https=)
KR (1) KR20200061381A (https=)
CN (1) CN112153968A (https=)
AU (2) AU2018346763A1 (https=)
CA (1) CA3076823A1 (https=)
IL (1) IL273639B2 (https=)
MA (1) MA50630A (https=)
MX (1) MX2020003811A (https=)
SG (2) SG11202002706XA (https=)
WO (1) WO2019071162A2 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11192856B2 (en) 2017-10-05 2021-12-07 Biogen Inc. Process for preparing alpha-carboxamide pyrrolidine derivatives

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