JP2020529439A5 - - Google Patents

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Publication number
JP2020529439A5
JP2020529439A5 JP2020505898A JP2020505898A JP2020529439A5 JP 2020529439 A5 JP2020529439 A5 JP 2020529439A5 JP 2020505898 A JP2020505898 A JP 2020505898A JP 2020505898 A JP2020505898 A JP 2020505898A JP 2020529439 A5 JP2020529439 A5 JP 2020529439A5
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JP
Japan
Prior art keywords
dihydro
trifluoromethyl
oxadiazine
phenyl
groups
Prior art date
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Application number
JP2020505898A
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English (en)
Japanese (ja)
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JP7676141B2 (ja
JP2020529439A (ja
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Priority claimed from PCT/EP2018/071039 external-priority patent/WO2019025562A1/en
Publication of JP2020529439A publication Critical patent/JP2020529439A/ja
Publication of JP2020529439A5 publication Critical patent/JP2020529439A5/ja
Priority to JP2023097166A priority Critical patent/JP2023115065A/ja
Application granted granted Critical
Publication of JP7676141B2 publication Critical patent/JP7676141B2/ja
Active legal-status Critical Current
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JP2020505898A 2017-08-04 2018-08-02 ジヒドロオキサジアジノン Active JP7676141B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023097166A JP2023115065A (ja) 2017-08-04 2023-06-13 ジヒドロオキサジアジノン

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762541627P 2017-08-04 2017-08-04
US62/541,627 2017-08-04
PCT/EP2018/071039 WO2019025562A1 (en) 2017-08-04 2018-08-02 DIHYDROOXADIAZINONES

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023097166A Division JP2023115065A (ja) 2017-08-04 2023-06-13 ジヒドロオキサジアジノン

Publications (3)

Publication Number Publication Date
JP2020529439A JP2020529439A (ja) 2020-10-08
JP2020529439A5 true JP2020529439A5 (enExample) 2021-09-09
JP7676141B2 JP7676141B2 (ja) 2025-05-14

Family

ID=63207725

Family Applications (2)

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JP2020505898A Active JP7676141B2 (ja) 2017-08-04 2018-08-02 ジヒドロオキサジアジノン
JP2023097166A Pending JP2023115065A (ja) 2017-08-04 2023-06-13 ジヒドロオキサジアジノン

Family Applications After (1)

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JP2023097166A Pending JP2023115065A (ja) 2017-08-04 2023-06-13 ジヒドロオキサジアジノン

Country Status (26)

Country Link
US (3) US11427553B2 (enExample)
EP (1) EP3661517B1 (enExample)
JP (2) JP7676141B2 (enExample)
KR (1) KR20200036914A (enExample)
CN (1) CN111212647B (enExample)
AR (1) AR112402A1 (enExample)
AU (1) AU2018309356B2 (enExample)
BR (1) BR112020002351A2 (enExample)
CA (1) CA3071800A1 (enExample)
CL (1) CL2020000303A1 (enExample)
CO (1) CO2020001242A2 (enExample)
CR (1) CR20200057A (enExample)
CU (1) CU24608B1 (enExample)
EA (1) EA202090448A1 (enExample)
EC (1) ECSP20008441A (enExample)
IL (1) IL272098B2 (enExample)
JO (1) JOP20200024A1 (enExample)
MA (1) MA49750A (enExample)
MX (1) MX2020001404A (enExample)
PE (1) PE20200936A1 (enExample)
PH (1) PH12020500134A1 (enExample)
SG (1) SG11201913775UA (enExample)
TW (1) TWI791581B (enExample)
UA (1) UA125731C2 (enExample)
UY (1) UY37832A (enExample)
WO (1) WO2019025562A1 (enExample)

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JOP20200024A1 (ar) 2017-08-04 2020-02-02 Bayer Ag مركبات ثنائي هيدروكساديازينون
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TW202031677A (zh) 2018-11-01 2020-09-01 美商博得學院股份有限公司 Ｐｄｅ３調節劑反應性癌症之鑑定
WO2020157188A1 (en) * 2019-02-01 2020-08-06 Bayer Aktiengesellschaft Dihydrooxadiazinones for the treatment of hyperproliferative diseases
AU2020215088A1 (en) 2019-02-01 2021-07-22 Bayer Aktiengesellschaft 1,2,4-triazin-3(2H)-one compounds for the treatment of hyperproliferative diseases
CN117279644A (zh) 2021-03-03 2023-12-22 拜耳股份有限公司 用于治疗肉瘤的取代的3,6-二氢-2h-1,3,4-噁二嗪-2-酮
EP4289828A1 (en) 2022-06-10 2023-12-13 Bayer Aktiengesellschaft Method for the preparation of a 3,6-dihydro-2h-1,3,4-oxadiazin-2-one
EP4289829A1 (en) 2022-06-10 2023-12-13 Bayer Aktiengesellschaft Crystalline forms of (6s)-5-[4'-fluoro-2-(trifluoromethyl)biphenyl-4-yl]-6-methyl-3,6-dihydro- 2h-1,3,4-oxadiazin-2-one
CN120187704A (zh) * 2022-11-24 2025-06-20 盛睿泽华医药科技（苏州）有限公司 吡啶酮化合物及其制备方法和用途
CN117903077B (zh) * 2023-01-13 2024-09-03 上海超阳药业有限公司 二氢噁二嗪酮化合物及其应用
CN118420559B (zh) * 2023-04-27 2025-02-14 上海超阳药业有限公司 氘代噁二嗪酮化合物及其用途
CN118047833B (zh) * 2024-01-31 2025-03-14 海南大学 含二茂铁的取代氨基乙酰胺类化合物及其制备方法和应用

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KR101831772B1 (ko) * 2016-03-24 2018-03-06 아이디에스(주) 복합 광원 모듈을 가지는 카메라 접사용 기구 및 이를 이용한 지문 시편 촬영 방법
TWI808055B (zh) 2016-05-11 2023-07-11 美商滬亞生物國際有限公司 Hdac 抑制劑與 pd-1 抑制劑之組合治療
TWI794171B (zh) 2016-05-11 2023-03-01 美商滬亞生物國際有限公司 Ｈｄａｃ抑制劑與ｐｄ-ｌ１抑制劑之組合治療
JOP20200024A1 (ar) 2017-08-04 2020-02-02 Bayer Ag مركبات ثنائي هيدروكساديازينون
EP3661917B1 (en) 2017-08-04 2022-05-11 Bayer Aktiengesellschaft 6-((3-trifluoromethyl)phenyl)-4,5-dihydropyridazin-3(2h)-one derivatives as pde3a and pde3b inhibitors for treating cancer
TW202031677A (zh) 2018-11-01 2020-09-01 美商博得學院股份有限公司 Ｐｄｅ３調節劑反應性癌症之鑑定
AU2020215088A1 (en) 2019-02-01 2021-07-22 Bayer Aktiengesellschaft 1,2,4-triazin-3(2H)-one compounds for the treatment of hyperproliferative diseases

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