JP2020507566A5 - - Google Patents

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Publication number
JP2020507566A5
JP2020507566A5 JP2019542672A JP2019542672A JP2020507566A5 JP 2020507566 A5 JP2020507566 A5 JP 2020507566A5 JP 2019542672 A JP2019542672 A JP 2019542672A JP 2019542672 A JP2019542672 A JP 2019542672A JP 2020507566 A5 JP2020507566 A5 JP 2020507566A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
compound according
membered
cancer
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
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JP2019542672A
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English (en)
Japanese (ja)
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JP2020507566A (ja
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Priority claimed from PCT/US2018/017668 external-priority patent/WO2018148576A1/en
Publication of JP2020507566A publication Critical patent/JP2020507566A/ja
Publication of JP2020507566A5 publication Critical patent/JP2020507566A5/ja
Withdrawn legal-status Critical Current

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JP2019542672A 2017-02-10 2018-02-09 ベンゾチオフェンエストロゲン受容体モジュレーター Withdrawn JP2020507566A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201762457643P 2017-02-10 2017-02-10
US62/457,643 2017-02-10
US201762460358P 2017-02-17 2017-02-17
US62/460,358 2017-02-17
US201862614279P 2018-01-05 2018-01-05
US62/614,279 2018-01-05
PCT/US2018/017668 WO2018148576A1 (en) 2017-02-10 2018-02-09 Benzothiophene estrogen receptor modulators

Publications (2)

Publication Number Publication Date
JP2020507566A JP2020507566A (ja) 2020-03-12
JP2020507566A5 true JP2020507566A5 (https=) 2021-03-25

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ID=63106724

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JP2019542672A Withdrawn JP2020507566A (ja) 2017-02-10 2018-02-09 ベンゾチオフェンエストロゲン受容体モジュレーター

Country Status (10)

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US (3) US10208011B2 (https=)
EP (1) EP3580223A4 (https=)
JP (1) JP2020507566A (https=)
KR (1) KR20190117582A (https=)
CN (1) CN110461853A (https=)
AU (1) AU2018217809A1 (https=)
CA (1) CA3052810A1 (https=)
IL (1) IL268319A (https=)
TW (1) TW201835064A (https=)
WO (1) WO2018148576A1 (https=)

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CN112839646A (zh) * 2018-08-16 2021-05-25 G1治疗公司 用于治疗医学疾病的苯并噻吩雌激素受体调节剂
KR20220071223A (ko) 2019-09-30 2022-05-31 닛뽕 케미파 가부시키가이샤 아제판 유도체
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CN113816892A (zh) * 2021-08-27 2021-12-21 安徽鼎旺医药有限公司 一种醋酸巴多昔芬的合成方法
CN113801094A (zh) * 2021-10-29 2021-12-17 中国药科大学 一种2-羰基苯并噻吩类化合物及其制备方法和用途
TW202543650A (zh) 2024-03-08 2025-11-16 美商海爾達醫療運營公司 異雙官能化合物及其在治療疾病中之用途

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