JP2019529500A5 - - Google Patents

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JP2019529500A5
JP2019529500A5 JP2019517777A JP2019517777A JP2019529500A5 JP 2019529500 A5 JP2019529500 A5 JP 2019529500A5 JP 2019517777 A JP2019517777 A JP 2019517777A JP 2019517777 A JP2019517777 A JP 2019517777A JP 2019529500 A5 JP2019529500 A5 JP 2019529500A5
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cancer
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JP2019517777A
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JP2019529500A (ja
JP7184761B2 (ja
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Priority claimed from PCT/US2017/054694 external-priority patent/WO2018067424A1/en
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Priority to JP2022158467A priority Critical patent/JP2022173493A/ja
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JP2019517777A 2016-10-03 2017-10-02 アデノシン５’－ヌクレオチダーゼの阻害剤 Active JP7184761B2 (ja)

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Application Number Priority Date Filing Date Title
JP2022158467A JP2022173493A (ja) 2016-10-03 2022-09-30 アデノシン５’－ヌクレオチダーゼの阻害剤

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662403598P 2016-10-03 2016-10-03
US62/403,598 2016-10-03
PCT/US2017/054694 WO2018067424A1 (en) 2016-10-03 2017-10-02 Inhibitors of adenosine 5'-nucleotidase

Related Child Applications (1)

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JP2022158467A Division JP2022173493A (ja) 2016-10-03 2022-09-30 アデノシン５’－ヌクレオチダーゼの阻害剤

Publications (3)

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JP2019529500A JP2019529500A (ja) 2019-10-17
JP2019529500A5 true JP2019529500A5 (enExample) 2021-04-15
JP7184761B2 JP7184761B2 (ja) 2022-12-06

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JP2019517777A Active JP7184761B2 (ja) 2016-10-03 2017-10-02 アデノシン５’－ヌクレオチダーゼの阻害剤
JP2022158467A Withdrawn JP2022173493A (ja) 2016-10-03 2022-09-30 アデノシン５’－ヌクレオチダーゼの阻害剤

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JP2022158467A Withdrawn JP2022173493A (ja) 2016-10-03 2022-09-30 アデノシン５’－ヌクレオチダーゼの阻害剤

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US (3) US11058704B2 (enExample)
EP (1) EP3518934A4 (enExample)
JP (2) JP7184761B2 (enExample)
CN (1) CN110049767B (enExample)
TW (1) TWI781960B (enExample)
WO (1) WO2018067424A1 (enExample)

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CN112955444B (zh) * 2019-01-22 2023-12-12 江苏恒瑞医药股份有限公司 一种新型的小分子cd73抑制剂、其制备方法及其在医药上的应用
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IL292570B2 (en) * 2019-10-30 2024-04-01 Oric Pharmaceuticals Inc Cd73 inhibitors
IL295569B1 (en) 2020-03-19 2026-04-01 Arcus Biosciences Inc Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2ALPHA
US11820824B2 (en) 2020-06-02 2023-11-21 Arcus Biosciences, Inc. Antibodies to TIGIT
US20240226115A1 (en) 2021-05-21 2024-07-11 Arcus Biosciences, Inc. Axl inhibitor compounds
WO2022246177A1 (en) 2021-05-21 2022-11-24 Arcus Biosciences, Inc. Axl compounds
WO2023077046A1 (en) 2021-10-29 2023-05-04 Arcus Biosciences, Inc. Inhibitors of hif-2alpha and methods of use thereof
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WO2023215719A1 (en) 2022-05-02 2023-11-09 Arcus Biosciences, Inc. Anti-tigit antibodies and uses of the same
CN116768949B (zh) * 2022-07-12 2026-03-03 南京工业大学 一种基于3’-脱氧腺苷经化学修饰改性的具有抗癌效应的化合物
EP4554680A1 (en) 2022-07-15 2025-05-21 Arcus Biosciences, Inc. Inhibitors of hpk1 and methods of use thereof
WO2024020034A1 (en) 2022-07-20 2024-01-25 Arcus Biosciences, Inc. Cbl-b inhibitors and methods of use thereof
US20260115190A1 (en) 2022-09-14 2026-04-30 Arcus Biosciences, Inc. Dispersions of etrumadenant
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WO2024226872A2 (en) * 2023-04-26 2024-10-31 Lakewood Amedex, Inc. Substituted bicyclic heterocycle compounds, compositions, and uses thereof
US20240425497A1 (en) 2023-05-05 2024-12-26 Arcus Biosciences, Inc. Cbl-b Inhibitors and Methods of Use Thereof
WO2024243502A1 (en) 2023-05-25 2024-11-28 Arcus Biosciences, Inc. Cbl-b inhibitors and methods of use thereof
WO2025054339A1 (en) 2023-09-08 2025-03-13 Arcus Biosciences, Inc. Triazolopyridine compounds as inhibitors of kit
WO2025072330A1 (en) 2023-09-26 2025-04-03 Arcus Biosciences, Inc. Kit inhibitor compounds and methods of use thereof
US20260116868A1 (en) 2023-10-06 2026-04-30 Arcus Biosciences, Inc. Cbl-b inhibitors and methods of use thereof
TW202523302A (zh) 2023-11-02 2025-06-16 美商阿克思生物科學有限公司 噻唑化合物及其使用方法
WO2025113498A1 (zh) * 2023-12-01 2025-06-05 无锡和誉生物医药科技有限公司 一种cd73抑制剂碱式盐及其制备方法和应用
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