JP2016523973A5 - - Google Patents
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- JP2016523973A5 JP2016523973A5 JP2016525463A JP2016525463A JP2016523973A5 JP 2016523973 A5 JP2016523973 A5 JP 2016523973A5 JP 2016525463 A JP2016525463 A JP 2016525463A JP 2016525463 A JP2016525463 A JP 2016525463A JP 2016523973 A5 JP2016523973 A5 JP 2016523973A5
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361844304P | 2013-07-09 | 2013-07-09 | |
| US61/844,304 | 2013-07-09 | ||
| US201361901808P | 2013-11-08 | 2013-11-08 | |
| US61/901,808 | 2013-11-08 | ||
| PCT/US2014/046022 WO2015006492A1 (en) | 2013-07-09 | 2014-07-09 | Kinase inhibitors for the treatment of disease |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2016523973A JP2016523973A (ja) | 2016-08-12 |
| JP2016523973A5 true JP2016523973A5 (enExample) | 2017-07-27 |
Family
ID=52280579
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016525463A Pending JP2016523973A (ja) | 2013-07-09 | 2014-07-09 | 疾患の処置のためのキナーゼ阻害物質 |
Country Status (6)
| Country | Link |
|---|---|
| US (3) | US9783504B2 (enExample) |
| EP (1) | EP3019491A4 (enExample) |
| JP (1) | JP2016523973A (enExample) |
| AU (1) | AU2014287209B2 (enExample) |
| CA (1) | CA2917667A1 (enExample) |
| WO (1) | WO2015006492A1 (enExample) |
Families Citing this family (74)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012088266A2 (en) | 2010-12-22 | 2012-06-28 | Incyte Corporation | Substituted imidazopyridazines and benzimidazoles as inhibitors of fgfr3 |
| GB201204384D0 (en) | 2012-03-13 | 2012-04-25 | Univ Dundee | Anti-flammatory agents |
| LT3495367T (lt) | 2012-06-13 | 2021-02-25 | Incyte Holdings Corporation | Pakeistieji tricikliniai junginiai, kaip fgfr inhibitoriai |
| WO2014026125A1 (en) | 2012-08-10 | 2014-02-13 | Incyte Corporation | Pyrazine derivatives as fgfr inhibitors |
| US9266892B2 (en) | 2012-12-19 | 2016-02-23 | Incyte Holdings Corporation | Fused pyrazoles as FGFR inhibitors |
| CA2907243C (en) | 2013-03-15 | 2021-12-28 | Celgene Avilomics Research, Inc. | Substituted dihydropyrimidopyrimidinone compounds and pharmaceutical compositions thereof use fgfr4 inhibitor |
| US9321786B2 (en) | 2013-03-15 | 2016-04-26 | Celgene Avilomics Research, Inc. | Heteroaryl compounds and uses thereof |
| JP6576325B2 (ja) | 2013-03-15 | 2019-09-18 | セルジーン シーエーアール エルエルシー | ヘテロアリール化合物およびそれらの使用 |
| LT2986610T (lt) | 2013-04-19 | 2018-04-10 | Incyte Holdings Corporation | Bicikliniai heterociklai, kaip fgfr inhibitoriai |
| AU2014287209B2 (en) * | 2013-07-09 | 2019-01-24 | Dana-Farber Cancer Institute, Inc. | Kinase inhibitors for the treatment of disease |
| SMT201800379T1 (it) | 2013-10-18 | 2018-09-13 | Eisai R&D Man Co Ltd | Inibitori di fgfr4 della pirimidina |
| BR112016008276B1 (pt) | 2013-10-25 | 2021-03-02 | Novartis Ag | derivados bicíclicos de piridila fundidos ao anel, seus usos e seu intermediário, e composição farmacêutica |
| CN105813635A (zh) | 2013-12-13 | 2016-07-27 | 诺华股份有限公司 | 药物剂型 |
| CN104860891B (zh) * | 2014-02-25 | 2017-06-30 | 上海海雁医药科技有限公司 | 芳氨基嘧啶类化合物及其应用以及由其制备的药物组合物和药用组合物 |
| DK3172213T3 (da) | 2014-07-21 | 2021-12-13 | Dana Farber Cancer Inst Inc | Makrocykliske kinasehæmmere og anvendelser deraf |
| US10287268B2 (en) | 2014-07-21 | 2019-05-14 | Dana-Farber Cancer Institute, Inc. | Imidazolyl kinase inhibitors and uses thereof |
| WO2016023014A2 (en) * | 2014-08-08 | 2016-02-11 | Dana-Farber Cancer Institute, Inc. | Uses of salt-inducible kinase (sik) inhibitors |
| WO2016054483A1 (en) | 2014-10-03 | 2016-04-07 | Novartis Ag | Use of ring-fused bicyclic pyridyl derivatives as fgfr4 inhibitors |
| US10851105B2 (en) | 2014-10-22 | 2020-12-01 | Incyte Corporation | Bicyclic heterocycles as FGFR4 inhibitors |
| EP4653015A3 (en) | 2015-01-26 | 2025-12-31 | Yale University | COMPOSITIONS AND METHODS OF USE OF TYROSINE KINASE INHIBITORS |
| CN105985342B (zh) * | 2015-02-06 | 2018-07-24 | 华东理工大学 | 作为egfr抑制剂的嘧啶并嘧啶二酮衍生物及其应用 |
| CN105884695B (zh) * | 2015-02-13 | 2019-02-26 | 山东轩竹医药科技有限公司 | 杂环衍生物类酪氨酸激酶抑制剂 |
| WO2016134294A1 (en) | 2015-02-20 | 2016-08-25 | Incyte Corporation | Bicyclic heterocycles as fgfr4 inhibitors |
| SG11201706287PA (en) * | 2015-02-20 | 2017-09-28 | Incyte Corp | Bicyclic heterocycles as fgfr inhibitors |
| MA41551A (fr) | 2015-02-20 | 2017-12-26 | Incyte Corp | Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4 |
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2014
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- 2014-07-09 EP EP14822373.8A patent/EP3019491A4/en not_active Withdrawn
- 2014-07-09 US US14/903,650 patent/US9783504B2/en active Active
- 2014-07-09 WO PCT/US2014/046022 patent/WO2015006492A1/en not_active Ceased
- 2014-07-09 JP JP2016525463A patent/JP2016523973A/ja active Pending
- 2014-07-09 CA CA2917667A patent/CA2917667A1/en not_active Abandoned
-
2017
- 2017-09-06 US US15/696,309 patent/US10316002B2/en not_active Expired - Fee Related
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2019
- 2019-05-06 US US16/403,793 patent/US10906878B2/en active Active
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