JP2019137703A5 - - Google Patents

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Publication number
JP2019137703A5
JP2019137703A5 JP2019104562A JP2019104562A JP2019137703A5 JP 2019137703 A5 JP2019137703 A5 JP 2019137703A5 JP 2019104562 A JP2019104562 A JP 2019104562A JP 2019104562 A JP2019104562 A JP 2019104562A JP 2019137703 A5 JP2019137703 A5 JP 2019137703A5
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JP
Japan
Prior art keywords
tablet
iron oxide
titanium dioxide
light stabilizer
red
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JP2019104562A
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English (en)
Japanese (ja)
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JP6861758B2 (ja
JP2019137703A (ja
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Publication of JP2019137703A publication Critical patent/JP2019137703A/ja
Publication of JP2019137703A5 publication Critical patent/JP2019137703A5/ja
Priority to JP2021057424A priority Critical patent/JP2021100971A/ja
Application granted granted Critical
Publication of JP6861758B2 publication Critical patent/JP6861758B2/ja
Priority to JP2023049709A priority patent/JP2023068197A/ja
Active legal-status Critical Current
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JP2019104562A 2013-06-06 2019-06-04 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤 Active JP6861758B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2021057424A JP2021100971A (ja) 2013-06-06 2021-03-30 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤
JP2023049709A JP2023068197A (ja) 2013-06-06 2023-03-27 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361831909P 2013-06-06 2013-06-06
US61/831,909 2013-06-06

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2016517984A Division JP6604941B2 (ja) 2013-06-06 2014-06-05 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2021057424A Division JP2021100971A (ja) 2013-06-06 2021-03-30 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤

Publications (3)

Publication Number Publication Date
JP2019137703A JP2019137703A (ja) 2019-08-22
JP2019137703A5 true JP2019137703A5 (enExample) 2019-11-14
JP6861758B2 JP6861758B2 (ja) 2021-04-21

Family

ID=51063834

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2016517984A Active JP6604941B2 (ja) 2013-06-06 2014-06-05 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤
JP2019104562A Active JP6861758B2 (ja) 2013-06-06 2019-06-04 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤
JP2021057424A Withdrawn JP2021100971A (ja) 2013-06-06 2021-03-30 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤
JP2023049709A Pending JP2023068197A (ja) 2013-06-06 2023-03-27 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2016517984A Active JP6604941B2 (ja) 2013-06-06 2014-06-05 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2021057424A Withdrawn JP2021100971A (ja) 2013-06-06 2021-03-30 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤
JP2023049709A Pending JP2023068197A (ja) 2013-06-06 2023-03-27 Hifプロリルヒドロキシラーゼ阻害剤の医薬製剤

Country Status (24)

Country Link
US (3) US20160120859A1 (enExample)
EP (2) EP3708154A1 (enExample)
JP (4) JP6604941B2 (enExample)
KR (3) KR20220164069A (enExample)
CN (5) CN111728951A (enExample)
AU (1) AU2014274890B2 (enExample)
CA (1) CA2914049C (enExample)
CY (1) CY1122951T1 (enExample)
DK (1) DK3003284T3 (enExample)
ES (1) ES2786924T3 (enExample)
HR (1) HRP20200615T1 (enExample)
HU (1) HUE049623T2 (enExample)
IL (3) IL296484B2 (enExample)
LT (1) LT3003284T (enExample)
ME (1) ME03777B (enExample)
MX (3) MX2015016536A (enExample)
PL (1) PL3003284T3 (enExample)
PT (1) PT3003284T (enExample)
RS (1) RS60464B1 (enExample)
SG (1) SG11201509764RA (enExample)
SI (1) SI3003284T1 (enExample)
SM (1) SMT202000190T1 (enExample)
WO (1) WO2014197660A1 (enExample)
ZA (1) ZA201508712B (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100932169B1 (ko) 2003-06-06 2009-12-16 피브로겐, 인크. 질소-함유 헤테로아릴 화합물 및 내인성 적혈구생성소의증가에서의 그들의 사용
CN102272117B (zh) 2008-11-14 2015-06-17 菲布罗根有限公司 作为hif羟化酶抑制剂的苯并噻喃衍生物
US9115085B2 (en) 2012-07-16 2015-08-25 Fibrogen, Inc. Crystalline forms of a prolyl hydroxylase inhibitor
US8883823B2 (en) 2012-07-16 2014-11-11 Fibrogen, Inc. Crystalline forms of a prolyl hydroxylase inhibitor
US9340511B2 (en) 2012-07-16 2016-05-17 Fibrogen, Inc. Process for making isoquinoline compounds
IL296484B2 (en) 2013-06-06 2025-03-01 Fibrogen Inc Pharmaceutical formulations of HIF hydroxylase inhibitor
PL3277270T3 (pl) * 2015-04-01 2022-02-14 Akebia Therapeutics, Inc. Kompozycje i sposoby leczenia niedokrwistości
WO2019042485A1 (en) 2017-08-30 2019-03-07 Zentiva, K.S. FORMS IN THE STRONG STATE OF ROXADUSTAT
JP7144510B2 (ja) * 2017-09-04 2022-09-29 サンド・アクチエンゲゼルシヤフト 経口投与可能なhifプロリルヒドロキシラーゼ阻害剤の共結晶
CN110664814A (zh) * 2019-10-24 2020-01-10 上海长海医院 Fg-4592在制备治疗炎性肠病药物中的用途
CN110934833B (zh) * 2019-12-17 2022-08-19 河北长天药业有限公司 一种复方氨酚那敏颗粒
EP4121009A4 (en) * 2020-03-17 2024-04-17 Zydus Lifesciences Limited Formulation comprising hif prolyl hydroxylase inhibitors
US20220280482A1 (en) * 2021-03-06 2022-09-08 Mind Medicine, Inc. Formulations of psilocin that have enhanced stability
CN116832005A (zh) * 2022-03-23 2023-10-03 石药集团中奇制药技术(石家庄)有限公司 一种罗沙司他胶囊
CN114796280B (zh) * 2022-06-15 2024-06-25 河北长天药业有限公司 一种复方氨酚那敏颗粒及其制备工艺
EP4321155A1 (en) * 2022-08-08 2024-02-14 Sanovel Ilac Sanayi Ve Ticaret A.S. An oral pharmaceutical composition comprising roxadustat
WO2025111214A1 (en) 2023-11-22 2025-05-30 Fibrogen, Inc. [(4-hydroxy-1-methyl-7-phenoxyisoquinoline-3- carbonyl)amino]acetic acid (roxadustat) for the treatment of anemia in subjects with myelodysplastic syndrome (mds)
CN118436652A (zh) * 2024-04-18 2024-08-06 南方医科大学顺德医院(佛山市顺德区第一人民医院) 一种罗沙司他药物制剂及其应用

Family Cites Families (52)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE149486T1 (de) 1993-11-02 1997-03-15 Hoechst Ag Substituierte heterocyclische carbonsäureamide, ihre herstellung und ihre verwendung als arzneimittel
DE19746287A1 (de) 1997-10-20 1999-04-22 Hoechst Marion Roussel De Gmbh Substituierte Isochinolin-2-Carbonsäureamide, ihre Herstellung und ihre Verwendung als Arzneimittel
US8318703B2 (en) 2001-12-06 2012-11-27 Fibrogen, Inc. Methods for improving kidney function
CN102526045A (zh) 2001-12-06 2012-07-04 法布罗根股份有限公司 提高内源性红细胞生成素(epo)的方法
DE10209692A1 (de) 2002-03-06 2003-09-18 Merck Patent Gmbh Isochinolinderivate
US7618940B2 (en) 2002-12-06 2009-11-17 Fibrogen, Inc. Fat regulation
US8124582B2 (en) 2002-12-06 2012-02-28 Fibrogen, Inc. Treatment of diabetes
HRP20050544B1 (hr) 2002-12-16 2017-12-01 Kissei Pharmaceutical Co., Ltd. Čvrsti oblik za oralnu upotrebu
JP4805234B2 (ja) * 2002-12-16 2011-11-02 キッセイ薬品工業株式会社 経口固形医薬
KR100932169B1 (ko) 2003-06-06 2009-12-16 피브로겐, 인크. 질소-함유 헤테로아릴 화합물 및 내인성 적혈구생성소의증가에서의 그들의 사용
US8614204B2 (en) 2003-06-06 2013-12-24 Fibrogen, Inc. Enhanced erythropoiesis and iron metabolism
EP1658074B1 (en) 2003-08-01 2012-11-07 Fibrogen, Inc. Inhibitors of 2-oxoglutarate dioxygenase as gamma globin inducers
CN1929847B (zh) 2004-03-16 2011-01-19 旭化成制药株式会社 含有法舒地尔的制剂及改善其稳定性的方法
CN101166745A (zh) 2005-03-02 2008-04-23 菲布罗根有限公司 噻吩并吡啶化合物和其使用方法
US20060276477A1 (en) 2005-06-06 2006-12-07 Fibrogen, Inc. Treatment method for anemia
ATE470439T1 (de) 2005-06-15 2010-06-15 Fibrogen Inc Verwendung von hif 1alfa modulatoren zur behandlung von krebs
UA97349C2 (uk) * 2005-09-08 2012-02-10 Х. Луннбэк А/С Стійкі тверді склади сертиндолу
CA2626309A1 (en) 2005-10-31 2007-05-10 Kowa Co., Ltd. Pharmaceutical preparation containing pitavastatin with excellent photostability
GB0523810D0 (en) 2005-11-23 2006-01-04 Astrazeneca Ab Pharmaceutical compositions
WO2007090068A2 (en) 2006-01-27 2007-08-09 Fibrogen, Inc. Cyanoisoquinoline compounds that stabilize hypoxia inducible factor (hif)
CA2635841A1 (en) * 2006-02-09 2007-08-16 Teva Pharmaceutical Industries Ltd. Stable pharmaceutical formulations of montelukast sodium
KR20080097446A (ko) 2006-02-16 2008-11-05 피브로겐, 인크. 뇌졸중의 치료를 위한 화합물과 방법
EP2016078B1 (en) 2006-04-04 2016-06-15 Fibrogen, Inc. Pyrrolo- and thiazolo-pyridine compounds as hif modulators
US20100172984A1 (en) * 2006-06-06 2010-07-08 Bijay Kumar Padhi tablet dosage form comprising cetirizine and pseudoephedrine
US7713986B2 (en) 2006-06-15 2010-05-11 Fibrogen, Inc. Compounds and methods for treatment of chemotherapy-induced anemia
US20070293575A1 (en) 2006-06-15 2007-12-20 Fibrogen, Inc. Compounds and methods for treatment of cancer-related anemia
JP5683058B2 (ja) * 2007-04-27 2015-03-11 ニプロ株式会社 経口固形製剤及びその製造方法
EP2209501B1 (en) 2007-10-12 2011-12-14 AstraZeneca AB Zibotentan composition containing mannitol and microcrystalline cellulose
AU2008319229A1 (en) 2007-11-02 2009-05-07 Fibrogen, Inc. Methods for reducing blood pressure
US8269008B2 (en) 2007-12-03 2012-09-18 Fibrogen, Inc. Oxazolopyridine and isoxazolopyridine derivatives for use in the treatment of HIF-mediated conditions
WO2009075824A1 (en) 2007-12-06 2009-06-18 Fibrogen, Inc. Methods for increasing endothelial progentior cells
US20110039879A1 (en) 2007-12-07 2011-02-17 FibroGen ,Inc. Methods for increasing white blood cells
EP2252619B1 (en) 2008-01-11 2013-10-09 Fibrogen, Inc. Isothiazole-pyridine derivatives as modulators of hif (hypoxia inducible factor) activity
US8324405B2 (en) 2008-02-05 2012-12-04 Fibrogen, Inc. Chromene derivatives and use thereof as HIF hydroxylase activity inhibitors
US8217043B2 (en) 2008-08-20 2012-07-10 Fibrogen, Inc. Compounds and methods for their use
EP2341904A1 (en) 2008-08-26 2011-07-13 Fibrogen, Inc. Methods for treatment of multiple sclerosis
CN102272117B (zh) 2008-11-14 2015-06-17 菲布罗根有限公司 作为hif羟化酶抑制剂的苯并噻喃衍生物
US20100144737A1 (en) 2008-12-08 2010-06-10 Fibrogen, Inc. Methods for inhibiting t helper cell differentiation
US20110305758A1 (en) 2009-01-29 2011-12-15 Mitsuhiro Matono Orally disintegrating tablet having inner core
JP2010248106A (ja) * 2009-04-14 2010-11-04 Dainippon Sumitomo Pharma Co Ltd フィルムコーティング錠
JP2012176899A (ja) * 2009-05-19 2012-09-13 Mitsubishi Tanabe Pharma Corp 2−(1−ピペラジニル)−5−メチルベンゼンスルホン酸誘導体を含む注射用水溶液
US20140057941A1 (en) 2011-01-13 2014-02-27 Kin-Hung (Peony) Yu Methods For Increasing Mean Corpuscular Volume
CN103429239A (zh) * 2011-01-13 2013-12-04 菲布罗根有限公司 增加网织红细胞血红蛋白含量的方法
CN103608346B (zh) 2011-02-02 2016-06-15 菲布罗根有限公司 作为缺氧诱导因子(hif)羟化酶抑制剂的萘啶衍生物
CA2842730C (en) 2011-07-22 2018-08-21 Beijing Betta Pharmaceuticals Co., Ltd Polymorphic forms of compounds as prolyl hydroxylase inhibitor, and uses thereof
US20140309256A1 (en) * 2011-11-09 2014-10-16 Fibrogen, Inc. Therapeutic Method
SG11201405574UA (en) 2012-03-09 2014-10-30 Fibrogen Inc 4 -hydroxy- isoquinoline compounds as hif hydroxylase inhibitors
US8883823B2 (en) 2012-07-16 2014-11-11 Fibrogen, Inc. Crystalline forms of a prolyl hydroxylase inhibitor
US9340511B2 (en) 2012-07-16 2016-05-17 Fibrogen, Inc. Process for making isoquinoline compounds
US9115085B2 (en) 2012-07-16 2015-08-25 Fibrogen, Inc. Crystalline forms of a prolyl hydroxylase inhibitor
WO2014116849A1 (en) 2013-01-24 2014-07-31 Fibrogen, Inc. Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid
IL296484B2 (en) 2013-06-06 2025-03-01 Fibrogen Inc Pharmaceutical formulations of HIF hydroxylase inhibitor

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