JP2018524342A5 - - Google Patents

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JP2018524342A5
JP2018524342A5 JP2017568018A JP2017568018A JP2018524342A5 JP 2018524342 A5 JP2018524342 A5 JP 2018524342A5 JP 2017568018 A JP2017568018 A JP 2017568018A JP 2017568018 A JP2017568018 A JP 2017568018A JP 2018524342 A5 JP2018524342 A5 JP 2018524342A5
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JP
Japan
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crystalline form
pain
pharmaceutical composition
ray powder
powder diffraction
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JP2017568018A
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English (en)
Japanese (ja)
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JP6917910B2 (ja
JP2018524342A (ja
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Priority claimed from PCT/US2016/040728 external-priority patent/WO2017004537A1/en
Publication of JP2018524342A publication Critical patent/JP2018524342A/ja
Publication of JP2018524342A5 publication Critical patent/JP2018524342A5/ja
Application granted granted Critical
Publication of JP6917910B2 publication Critical patent/JP6917910B2/ja
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JP2017568018A 2015-07-02 2016-07-01 （４−（（３ｒ，４ｒ）−３−メトキシテトラヒドロ−ピラン−４−イルアミノ）ピペリジン−１−イル）（５−メチル−６−（（（２ｒ，６ｓ）−６−（ｐ−トリル）テトラヒドロ−２ｈ−ピラン−２−イル）メチルアミノ）ピリミジン−４イル）メタノンクエン酸塩 Expired - Fee Related JP6917910B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15175066 2015-07-02
EP15175066.8 2015-07-02
PCT/US2016/040728 WO2017004537A1 (en) 2015-07-02 2016-07-01 (4-((3r,4r)-3-methoxytetrahydro-pyran-4-ylamino)piperidin-1-yl)(5-methyl-6-(((2r,6s)-6-(p-tolyl)tetrahydro-2h-pyran-2-yl)methylamino)pyrimidin-4yl)methanone citrate

Publications (3)

Publication Number Publication Date
JP2018524342A JP2018524342A (ja) 2018-08-30
JP2018524342A5 true JP2018524342A5 (enExample) 2019-08-08
JP6917910B2 JP6917910B2 (ja) 2021-08-11

Family

ID=53502570

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JP2017568018A Expired - Fee Related JP6917910B2 (ja) 2015-07-02 2016-07-01 （４−（（３ｒ，４ｒ）−３−メトキシテトラヒドロ−ピラン−４−イルアミノ）ピペリジン−１−イル）（５−メチル−６−（（（２ｒ，６ｓ）−６−（ｐ−トリル）テトラヒドロ−２ｈ−ピラン−２−イル）メチルアミノ）ピリミジン−４イル）メタノンクエン酸塩

Country Status (13)

Country Link
US (4) US10213428B2 (enExample)
EP (1) EP3317270B1 (enExample)
JP (1) JP6917910B2 (enExample)
CN (1) CN108026087B (enExample)
AU (1) AU2016287584B2 (enExample)
BR (1) BR112017028492B1 (enExample)
CA (1) CA2990460C (enExample)
ES (1) ES2811098T3 (enExample)
IL (1) IL256530A (enExample)
MX (1) MX383744B (enExample)
PL (1) PL3317270T3 (enExample)
PT (1) PT3317270T (enExample)
WO (1) WO2017004537A1 (enExample)

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WO2025228899A1 (en) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Further heterocyclic compounds as sting antagonists and the use thereof as medicament
WO2025228892A1 (en) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Monoaryl and hetaryl substituted indazoles and benzimidazoles as sting antagonists and the use thereof as medicament
WO2025228889A1 (en) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Monoarylic heterocyclic compounds as sting antagonists and the use thereof as medicament
WO2025228902A1 (en) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Heterocyclic acids as sting antagonists and the use thereof as medicament

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JP5786258B2 (ja) 2011-07-15 2015-09-30 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規かつ選択的なｃｃｒ２拮抗薬
JP6229575B2 (ja) 2014-03-31 2017-11-15 京セラドキュメントソリューションズ株式会社 画像処理装置
WO2017004537A1 (en) 2015-07-02 2017-01-05 Centrexion Therapeutics Corporation (4-((3r,4r)-3-methoxytetrahydro-pyran-4-ylamino)piperidin-1-yl)(5-methyl-6-(((2r,6s)-6-(p-tolyl)tetrahydro-2h-pyran-2-yl)methylamino)pyrimidin-4yl)methanone citrate

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