JP2018516963A5 - - Google Patents

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JP2018516963A5
JP2018516963A5 JP2017564114A JP2017564114A JP2018516963A5 JP 2018516963 A5 JP2018516963 A5 JP 2018516963A5 JP 2017564114 A JP2017564114 A JP 2017564114A JP 2017564114 A JP2017564114 A JP 2017564114A JP 2018516963 A5 JP2018516963 A5 JP 2018516963A5
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alkylene
alkyl
cycloalkyl
compound according
haloalkyl
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JP2017564114A
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JP6838004B2 (ja
JP2018516963A (ja
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Priority claimed from PCT/US2016/036889 external-priority patent/WO2016201225A1/en
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JP2017564114A 2015-06-11 2016-06-10 ＲＯＲγのアゴニストとしての使用及び疾患の治療のためのアリールジヒドロ−２Ｈ−ベンゾ［ｂ］［１，４］オキサジンスルホンアミド及び関連化合物 Expired - Fee Related JP6838004B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201562174094P 2015-06-11 2015-06-11
US62/174,094 2015-06-11
US201562210078P 2015-08-26 2015-08-26
US62/210,078 2015-08-26
PCT/US2016/036889 WO2016201225A1 (en) 2015-06-11 2016-06-10 Aryl dihydro-2h-benzo[b][1,4]oxazine sulfonamide and related compounds for use as agonists of rory and the treatment of disease

Publications (3)

Publication Number Publication Date
JP2018516963A JP2018516963A (ja) 2018-06-28
JP2018516963A5 true JP2018516963A5 (cg-RX-API-DMAC10.html) 2019-06-13
JP6838004B2 JP6838004B2 (ja) 2021-03-03

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JP2017564114A Expired - Fee Related JP6838004B2 (ja) 2015-06-11 2016-06-10 ＲＯＲγのアゴニストとしての使用及び疾患の治療のためのアリールジヒドロ−２Ｈ−ベンゾ［ｂ］［１，４］オキサジンスルホンアミド及び関連化合物

Country Status (11)

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US (2) US10611740B2 (cg-RX-API-DMAC10.html)
EP (1) EP3307738B1 (cg-RX-API-DMAC10.html)
JP (1) JP6838004B2 (cg-RX-API-DMAC10.html)
KR (1) KR20180025894A (cg-RX-API-DMAC10.html)
CN (1) CN107980042B (cg-RX-API-DMAC10.html)
AU (2) AU2016276947A1 (cg-RX-API-DMAC10.html)
CA (1) CA2987289A1 (cg-RX-API-DMAC10.html)
HK (1) HK1253734A1 (cg-RX-API-DMAC10.html)
IL (1) IL255919A (cg-RX-API-DMAC10.html)
MX (1) MX2017016134A (cg-RX-API-DMAC10.html)
WO (1) WO2016201225A1 (cg-RX-API-DMAC10.html)

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HK1253734A1 (zh) 2015-06-11 2019-06-28 The Regents Of The University Of Michigan 用作RORγ激动剂和用於治疗疾病的芳基二氢-2H-苯并[B][1，4]恶嗪磺酰胺和相关化合物
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CN112119065B (zh) * 2018-07-13 2024-01-23 四川科伦博泰生物医药股份有限公司 苯并二氮杂环类化合物、其制备方法及用途
CN110872243B (zh) * 2018-08-31 2023-03-31 四川科伦博泰生物医药股份有限公司 磺酰胺类化合物、其制备方法及用途
CN109568321B (zh) * 2019-01-14 2022-02-22 山东轩竹医药科技有限公司 RORγ调节剂
JP7290356B2 (ja) * 2019-01-23 2023-06-13 アビスコ セラピューティクス カンパニー リミテッド １，２，３，４－テトラヒドロキノキサリン誘導体、その製造方法および使用
CN111499591A (zh) * 2019-01-30 2020-08-07 山东轩竹医药科技有限公司 RORγ调节剂
CN111635373B (zh) * 2019-03-01 2022-07-12 山东轩竹医药科技有限公司 多环磺酰胺类RORγ调节剂
CN114096533B (zh) * 2019-09-10 2024-03-08 四川科伦博泰生物医药股份有限公司 一种三并环类化合物，包含其的药物组合物，其制备方法及其用途
CN115557913A (zh) * 2021-07-02 2023-01-03 广东东阳光药业有限公司 苯并氮杂环类化合物及其在药物中的应用
WO2023016530A1 (zh) * 2021-08-13 2023-02-16 南京明德新药研发有限公司 一类3,4-二氢-2H-苯并[b][1,4]噁嗪类化合物及其制备方法
WO2023016528A1 (zh) * 2021-08-13 2023-02-16 南京明德新药研发有限公司 一类苯并吗啉类化合物及其制备方法和用途
WO2023232870A1 (en) 2022-05-31 2023-12-07 Immunic Ag Rorg/rorgt modulators for the treatment of virus infections like covid-19
CN117865883B (zh) * 2022-12-10 2025-10-24 常州琦诺生物科技有限公司 一种6-溴喹啉的制备方法
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