JP2017526706A5 - - Google Patents
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- JP2017526706A5 JP2017526706A5 JP2017513199A JP2017513199A JP2017526706A5 JP 2017526706 A5 JP2017526706 A5 JP 2017526706A5 JP 2017513199 A JP2017513199 A JP 2017513199A JP 2017513199 A JP2017513199 A JP 2017513199A JP 2017526706 A5 JP2017526706 A5 JP 2017526706A5
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- lymphoma
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462048759P | 2014-09-10 | 2014-09-10 | |
| US62/048,759 | 2014-09-10 | ||
| US201562146794P | 2015-04-13 | 2015-04-13 | |
| US62/146,794 | 2015-04-13 | ||
| PCT/US2015/049213 WO2016040498A1 (en) | 2014-09-10 | 2015-09-09 | Isoxazole carboxamide compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2017526706A JP2017526706A (ja) | 2017-09-14 |
| JP2017526706A5 true JP2017526706A5 (enExample) | 2018-10-18 |
Family
ID=55459522
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017513199A Pending JP2017526706A (ja) | 2014-09-10 | 2015-09-09 | イソオキサゾールカルボキサミド化合物 |
Country Status (6)
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|---|---|
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| JP (1) | JP2017526706A (enExample) |
| AU (1) | AU2015315167A1 (enExample) |
| CA (1) | CA2960274A1 (enExample) |
| WO (1) | WO2016040498A1 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2016040515A1 (en) * | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Substituted piperidine compounds |
| JP2017527576A (ja) | 2014-09-10 | 2017-09-21 | エピザイム，インコーポレイティド | 置換シクロヘキシルアミン化合物 |
| WO2016040511A1 (en) | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Isoxazole carboxamides as irreversible smyd inhibitors |
| KR102496364B1 (ko) | 2014-09-10 | 2023-02-06 | 에피자임, 인코포레이티드 | Ｓｍｙｄ 억제제 |
| JP6763380B2 (ja) | 2015-06-17 | 2020-09-30 | 住友化学株式会社 | 有害節足動物防除剤 |
| MA53645A (fr) * | 2018-09-21 | 2021-12-29 | Novartis Ag | Composés d'isoxazole carboxamide et leurs utilisations |
| CN109879868B (zh) * | 2019-03-07 | 2022-04-22 | 南通大学 | 含2-芳基噁唑结构的吡唑酰胺类化合物的制备和应用 |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3065225A (en) * | 1960-02-05 | 1962-11-20 | Hoffmann La Roche | N', n4-di-isoxazolylcarbonyl-sulfanilamide derivatives |
| DE19930075A1 (de) * | 1999-06-30 | 2001-01-04 | Bayer Ag | Neue Amino- und Amidosulfonamide als antivirale Mittel |
| GB0017518D0 (en) * | 2000-07-17 | 2000-08-30 | Merck Sharp & Dohme | Therapeutic agents |
| US7259157B2 (en) * | 2001-04-03 | 2007-08-21 | Merck & Co., Inc. | N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists |
| CA2449249A1 (en) * | 2001-06-12 | 2002-12-19 | Merck & Co., Inc. | Nr2b receptor antagonists for the treatment or prevention of migraines |
| DE10306250A1 (de) * | 2003-02-14 | 2004-09-09 | Aventis Pharma Deutschland Gmbh | Substituierte N-Arylheterozyklen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| WO2005004810A2 (en) * | 2003-07-02 | 2005-01-20 | Merck & Co., Inc. | Arylsulfonamide derivatives |
| US7709645B2 (en) * | 2004-07-27 | 2010-05-04 | Sgx Pharmaceuticals, Inc. | Pyrrolo-pyridine kinase modulators |
| WO2006067446A1 (en) * | 2004-12-22 | 2006-06-29 | Astrazeneca Ab | Pyridine carboxamide derivatives for use as anticancer agents |
| US7291743B2 (en) * | 2005-03-29 | 2007-11-06 | Geneblue Corporation | Isoxazole derivatives and methods of treating nitric oxide mediated diseases |
| NL2000284C2 (nl) * | 2005-11-04 | 2007-09-28 | Pfizer Ltd | Pyrazine-derivaten. |
| WO2008040149A1 (en) * | 2006-09-05 | 2008-04-10 | Dexian Dou | Composition and method for treating immune-mediated skin disorders |
| BRPI0810202A2 (pt) * | 2007-05-03 | 2014-10-21 | Pfizer Ltd | Derivados de piridina |
| WO2008137834A2 (en) | 2007-05-04 | 2008-11-13 | Osi Pharmaceuticals, Inc. | Crystal structure of smyd3 protein |
| CA2786438C (en) * | 2010-01-29 | 2015-10-13 | Hanmi Science Co., Ltd. | Thieno[3,2-d]pyrimidine derivatives having inhibitory activity on protein kinases |
| WO2013043826A1 (en) * | 2011-09-21 | 2013-03-28 | Abbvie Inc. | Tricyclic compounds useful as protein kinase inhibitors |
| WO2014100157A1 (en) * | 2012-12-18 | 2014-06-26 | Alcyone Lifesciences, Inc. | Systems and methods for reducing or preventing backflow in a delivery system |
| AU2014237312B2 (en) * | 2013-03-15 | 2019-03-28 | Shifa Biomedical Corporation | Anti-proprotein convertase subtilisin kexin type 9 (anti-PCSK9) compounds and methods of using the same in the treatment and/or prevention of cardiovascular diseases |
| WO2016040511A1 (en) | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Isoxazole carboxamides as irreversible smyd inhibitors |
| US20170253601A1 (en) * | 2014-09-10 | 2017-09-07 | Epizyme, Inc. | Substituted Pyrrolidine Compounds |
| KR102496364B1 (ko) | 2014-09-10 | 2023-02-06 | 에피자임, 인코포레이티드 | Ｓｍｙｄ 억제제 |
| WO2016040508A1 (en) | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Substituted pyrrolidine carboxamide compounds |
| JP2017527576A (ja) | 2014-09-10 | 2017-09-21 | エピザイム，インコーポレイティド | 置換シクロヘキシルアミン化合物 |
| WO2016040515A1 (en) | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Substituted piperidine compounds |
-
2015
- 2015-09-09 US US15/510,593 patent/US10428029B2/en active Active
- 2015-09-09 WO PCT/US2015/049213 patent/WO2016040498A1/en not_active Ceased
- 2015-09-09 CA CA2960274A patent/CA2960274A1/en not_active Abandoned
- 2015-09-09 AU AU2015315167A patent/AU2015315167A1/en not_active Abandoned
- 2015-09-09 JP JP2017513199A patent/JP2017526706A/ja active Pending
- 2015-09-09 EP EP15839331.4A patent/EP3193603A4/en not_active Withdrawn
-
2019
- 2019-09-30 US US16/588,209 patent/US20200148650A1/en not_active Abandoned
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