JP2017527576A5 - - Google Patents
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- JP2017527576A5 JP2017527576A5 JP2017513205A JP2017513205A JP2017527576A5 JP 2017527576 A5 JP2017527576 A5 JP 2017527576A5 JP 2017513205 A JP2017513205 A JP 2017513205A JP 2017513205 A JP2017513205 A JP 2017513205A JP 2017527576 A5 JP2017527576 A5 JP 2017527576A5
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- Prior art keywords
- cancer
- tumor
- cell
- lymphoma
- carcinoma
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462048756P | 2014-09-10 | 2014-09-10 | |
| US62/048,756 | 2014-09-10 | ||
| PCT/US2015/049217 WO2016040502A1 (en) | 2014-09-10 | 2015-09-09 | Substituted cyclohexylamine compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2017527576A JP2017527576A (ja) | 2017-09-21 |
| JP2017527576A5 true JP2017527576A5 (enExample) | 2018-10-18 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017513205A Pending JP2017527576A (ja) | 2014-09-10 | 2015-09-09 | 置換シクロヘキシルアミン化合物 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US10106510B2 (enExample) |
| EP (1) | EP3190891B1 (enExample) |
| JP (1) | JP2017527576A (enExample) |
| AU (1) | AU2015315171A1 (enExample) |
| CA (1) | CA2960271A1 (enExample) |
| WO (1) | WO2016040502A1 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2017002985A (es) | 2014-09-10 | 2017-11-17 | Epizyme Inc | Inhibidores de smyd. |
| CA2960274A1 (en) | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Isoxazole carboxamide compounds |
| JP2017528464A (ja) | 2014-09-10 | 2017-09-28 | エピザイム，インコーポレイティド | 置換ピペリジン化合物 |
| WO2016040511A1 (en) * | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Isoxazole carboxamides as irreversible smyd inhibitors |
| CN121311462A (zh) * | 2023-04-19 | 2026-01-09 | 爱尔康公司 | N-取代的c6环基甲酰胺化合物及其用途 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20060089398A1 (en) * | 2003-03-19 | 2006-04-27 | Gang Liu | Isoxazole carboxamide derivatives as ghrelin receptor modulators |
| GB0317484D0 (en) * | 2003-07-25 | 2003-08-27 | Pfizer Ltd | Nicotinamide derivatives useful as pde4 inhibitors |
| WO2008065500A2 (en) * | 2006-11-30 | 2008-06-05 | Pfizer Products Inc. | Heteroaryl amides as type i glycine transport inhibitors |
| US20090062286A1 (en) * | 2007-05-04 | 2009-03-05 | Kenneth William Foreman | Crystal Structure of SMYD3 Protein |
| RU2509077C2 (ru) | 2008-05-27 | 2014-03-10 | Астразенека Аб | Феноксипиридиниламидные производные и их применение в лечении pde4-опосредованных болезненных состояний |
| KR20110036797A (ko) * | 2008-07-25 | 2011-04-11 | 하. 룬트벡 아크티에 셀스카브 | 아다만틸 디아미드 유도체 및 이의 용도 |
| JP6135391B2 (ja) | 2013-08-16 | 2017-05-31 | ソニー株式会社 | 撮像装置、画像処理装置、および画像処理方法、並びにプログラム |
| MX2017002985A (es) | 2014-09-10 | 2017-11-17 | Epizyme Inc | Inhibidores de smyd. |
| US20170253601A1 (en) | 2014-09-10 | 2017-09-07 | Epizyme, Inc. | Substituted Pyrrolidine Compounds |
| CA2960274A1 (en) | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Isoxazole carboxamide compounds |
| JP2017528461A (ja) | 2014-09-10 | 2017-09-28 | エピザイム インコーポレイテッド | 置換ピロリジンカルボキサミド化合物 |
| JP2017528464A (ja) | 2014-09-10 | 2017-09-28 | エピザイム，インコーポレイティド | 置換ピペリジン化合物 |
| WO2016040511A1 (en) | 2014-09-10 | 2016-03-17 | Epizyme, Inc. | Isoxazole carboxamides as irreversible smyd inhibitors |
-
2015
- 2015-09-09 WO PCT/US2015/049217 patent/WO2016040502A1/en not_active Ceased
- 2015-09-09 AU AU2015315171A patent/AU2015315171A1/en not_active Abandoned
- 2015-09-09 US US15/510,605 patent/US10106510B2/en active Active
- 2015-09-09 JP JP2017513205A patent/JP2017527576A/ja active Pending
- 2015-09-09 CA CA2960271A patent/CA2960271A1/en not_active Abandoned
- 2015-09-09 EP EP15839333.0A patent/EP3190891B1/en active Active
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