JP2017513808A5 - - Google Patents

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JP2017513808A5
JP2017513808A5 JP2016549758A JP2016549758A JP2017513808A5 JP 2017513808 A5 JP2017513808 A5 JP 2017513808A5 JP 2016549758 A JP2016549758 A JP 2016549758A JP 2016549758 A JP2016549758 A JP 2016549758A JP 2017513808 A5 JP2017513808 A5 JP 2017513808A5
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JP
Japan
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methyl
triazolo
pyrimidin
piperidine
carbonyl
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JP2016549758A
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Japanese (ja)
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JP6626449B2 (ja
JP2017513808A (ja
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Priority claimed from PCT/US2015/027102 external-priority patent/WO2015164508A1/en
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Publication of JP2017513808A5 publication Critical patent/JP2017513808A5/ja
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JP2016549758A 2014-04-23 2015-04-22 ＰＤＥ２阻害剤としての置換［１，２，４］トリアゾロ［１，５−ａ］ピリミジン−７−イル化合物 Active JP6626449B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461983387P 2014-04-23 2014-04-23
US61/983,387 2014-04-23
PCT/US2015/027102 WO2015164508A1 (en) 2014-04-23 2015-04-22 Substituted [1,2,4] triazolo [1,5-a] pyrimidin-7-yl compounds as pde2 inhibitors

Publications (3)

Publication Number Publication Date
JP2017513808A JP2017513808A (ja) 2017-06-01
JP2017513808A5 true JP2017513808A5 (https=) 2018-05-24
JP6626449B2 JP6626449B2 (ja) 2019-12-25

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ID=53055118

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JP2016549758A Active JP6626449B2 (ja) 2014-04-23 2015-04-22 ＰＤＥ２阻害剤としての置換［１，２，４］トリアゾロ［１，５−ａ］ピリミジン−７−イル化合物

Country Status (23)

Country Link
US (5) US9932345B2 (https=)
EP (2) EP3597649B8 (https=)
JP (1) JP6626449B2 (https=)
KR (1) KR102471058B1 (https=)
CN (2) CN106459062A (https=)
AU (2) AU2015249753B2 (https=)
BR (1) BR112016024713B1 (https=)
CA (1) CA2938294C (https=)
DK (2) DK3134413T3 (https=)
ES (2) ES2902806T3 (https=)
HR (1) HRP20212035T1 (https=)
HU (1) HUE057317T2 (https=)
IL (2) IL248292A (https=)
MA (1) MA50375A (https=)
MX (1) MX358004B (https=)
NZ (1) NZ725161A (https=)
PL (1) PL3597649T3 (https=)
PT (1) PT3597649T (https=)
RU (1) RU2659070C9 (https=)
SG (1) SG11201606216UA (https=)
SI (1) SI3597649T1 (https=)
TW (1) TWI664181B (https=)
WO (1) WO2015164508A1 (https=)

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DK3134413T3 (da) 2014-04-23 2019-10-14 Dart Neuroscience Cayman Ltd Substituerede [1,2,4]triazolo[1,5-a]pyrimidin-7-yl-forbindelser som pde2-inhibitorer
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AU2017222964B2 (en) 2016-02-25 2020-01-02 Asceneuron S. A. Glycosidase inhibitors
KR20180132629A (ko) 2016-02-25 2018-12-12 아셰뉴론 에스아 글리코시다제 저해제
US11261183B2 (en) 2016-02-25 2022-03-01 Asceneuron Sa Sulfoximine glycosidase inhibitors
CA3014572C (en) 2016-02-25 2023-10-03 Asceneuron S.A. Acid addition salts of piperazine derivatives
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US20190359609A1 (en) * 2016-12-16 2019-11-28 Janssen Pharmaceutica Nv Bicyclic oga inhibitor compounds
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US11213525B2 (en) 2017-08-24 2022-01-04 Asceneuron Sa Linear glycosidase inhibitors
WO2020039029A1 (en) 2018-08-22 2020-02-27 Asceneuron S. A. Spiro compounds as glycosidase inhibitors
WO2020039027A1 (en) 2018-08-22 2020-02-27 Asceneuron S. A. Pyrrolidine glycosidase inhibitors
WO2020039028A1 (en) 2018-08-22 2020-02-27 Asceneuron S. A. Tetrahydro-benzoazepine glycosidase inhibitors
JP7407171B2 (ja) 2018-08-22 2023-12-28 エースニューロン・ソシエテ・アノニム グリコシダーゼ阻害剤として有用なピペラジン誘導体のコハク酸付加塩及びフマル酸付加塩
EP3969639B1 (en) 2019-05-13 2025-03-12 Ecolab Usa Inc. 1,2,4-triazolo[1,5-a] pyrimidine derivative as copper corrosion inhibitor
TWI907472B (zh) 2020-08-05 2025-12-11 匈牙利商羅特格登公司 具藥理活性之經雜環取代的吡唑并〔１，５－ａ〕嘧啶衍生物

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