JP2016536363A - 節足動物を処理するための置換されたベンズアミド - Google Patents

節足動物を処理するための置換されたベンズアミド Download PDF

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Publication number
JP2016536363A
JP2016536363A JP2016551033A JP2016551033A JP2016536363A JP 2016536363 A JP2016536363 A JP 2016536363A JP 2016551033 A JP2016551033 A JP 2016551033A JP 2016551033 A JP2016551033 A JP 2016551033A JP 2016536363 A JP2016536363 A JP 2016536363A
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alkyl
halogen
substituted
spp
formula
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Japanese (ja)
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JP2016536363A5 (enExample
Inventor
ベルナー、ハレンバッハ
ハンス−ゲオルク、シュワルツ
ケルスティン、イルク
ウルリッヒ、ジェルゲン
ヨハネス、ケベルリンク
アンドレアス、トゥルベルク
ニールス、ベーンケ
ミヒャエル、マウエ
ローベルト、フェルテン
トビアス、ハルシュネック
ユリア、ヨハンナ、ハーン
セバスティアン、ホーストマン
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Bayer CropScience AG
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Bayer CropScience AG
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Publication of JP2016536363A publication Critical patent/JP2016536363A/ja
Publication of JP2016536363A5 publication Critical patent/JP2016536363A5/ja
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    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/36Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/561,2-Diazoles; Hydrogenated 1,2-diazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/337Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/08Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyrrole Compounds (AREA)
  • Pyridine Compounds (AREA)
JP2016551033A 2013-11-05 2014-11-05 節足動物を処理するための置換されたベンズアミド Pending JP2016536363A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP13191610.8 2013-11-05
EP13191610 2013-11-05
EP14181149.7 2014-08-15
EP14181149 2014-08-15
PCT/EP2014/073794 WO2015067646A1 (de) 2013-11-05 2014-11-05 Substituierte benzamide zur behandlung von arthropoden

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JP2016536363A true JP2016536363A (ja) 2016-11-24
JP2016536363A5 JP2016536363A5 (enExample) 2018-11-29

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JP2016551034A Pending JP2016536364A (ja) 2013-11-05 2014-11-05 節足動物を防除するための新規化合物
JP2016551033A Pending JP2016536363A (ja) 2013-11-05 2014-11-05 節足動物を処理するための置換されたベンズアミド
JP2019154161A Active JP6840803B2 (ja) 2013-11-05 2019-08-26 節足動物を処理するための置換されたベンズアミド
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US (2) US10150737B2 (enExample)
EP (2) EP3066080B1 (enExample)
JP (4) JP2016536364A (enExample)
KR (2) KR102400756B1 (enExample)
CN (2) CN106103414B (enExample)
AP (1) AP2016009182A0 (enExample)
AU (2) AU2014345593C1 (enExample)
BR (2) BR112016010094B1 (enExample)
CA (2) CA2929390C (enExample)
CL (2) CL2016001080A1 (enExample)
CR (2) CR20160210A (enExample)
CU (1) CU24381B1 (enExample)
DK (2) DK3066080T5 (enExample)
DO (2) DOP2016000103A (enExample)
ES (2) ES2683445T3 (enExample)
HR (2) HRP20181290T1 (enExample)
HU (2) HUE038665T2 (enExample)
IL (2) IL245408B (enExample)
LT (2) LT3066080T (enExample)
MX (2) MX367300B (enExample)
MY (1) MY175845A (enExample)
PE (2) PE20160905A1 (enExample)
PH (2) PH12016500830B1 (enExample)
PL (2) PL3066080T3 (enExample)
PT (2) PT3066080T (enExample)
RU (2) RU2712092C2 (enExample)
SI (2) SI3066079T1 (enExample)
SV (1) SV2016005194A (enExample)
TR (2) TR201808573T4 (enExample)
TW (2) TWI640507B (enExample)
UA (2) UA119972C2 (enExample)
UY (1) UY35819A (enExample)
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Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2016536364A (ja) * 2013-11-05 2016-11-24 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 節足動物を防除するための新規化合物
JP2019529413A (ja) * 2016-09-15 2019-10-17 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ripk2の阻害剤としてのピリジンおよびピラジン化合物
JPWO2018116945A1 (ja) * 2016-12-19 2019-10-24 日本曹達株式会社 ジアリールピラゾール化合物および有害生物防除剤
JP2020500901A (ja) * 2016-12-08 2020-01-16 バイエル・クロップサイエンス・アクチェンゲゼルシャフト フェニルヒドラジン中間体を単離又は精製することなく5−(1−フェニル−1h−ピラゾール−4−イル)−ニコチンアミド誘導体及び類似化合物を製造する方法
JP2020532563A (ja) * 2017-09-06 2020-11-12 バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Animal Health Gmbh 動物寄生虫(animal parasites)の防除および予防のための局所投与製剤
JP2023512012A (ja) * 2020-01-29 2023-03-23 バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング 非ヒト生物の寄生虫を防除するための医薬組成物
WO2023112988A1 (ja) * 2021-12-16 2023-06-22 住友化学株式会社 有害節足動物の防除方法

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PE20160654A1 (es) 2013-11-22 2016-07-15 Pharmakea Inc Compuestos de inhibidor de autotaxina
AR104398A1 (es) * 2015-04-30 2017-07-19 Bayer Animal Health Gmbh Combinaciones antiparasíticas
EP3302490B1 (en) 2015-05-27 2022-04-13 Sabre Therapeutics LLC Autotaxin inhibitors and uses thereof
WO2016204270A1 (ja) * 2015-06-18 2016-12-22 日本曹達株式会社 ジアリールアゾール化合物および有害生物防除剤
MX2018001707A (es) * 2015-08-13 2018-06-06 Bayer Cropscience Ag Novedosos compuestos para controlar artropodos.
BR112018005888A2 (pt) * 2015-09-25 2018-10-16 Syngenta Participations Ag derivados heterocíclicos ativos em termos pesticidas com substituintes contendo enxofre.
JP6802805B2 (ja) * 2015-11-30 2020-12-23 北興化学工業株式会社 1,2,3−トリアゾール誘導体および当該誘導体を有効成分とする殺虫・殺ダニ剤
JP6943857B2 (ja) 2015-12-22 2021-10-06 シンジェンタ パーティシペーションズ アーゲー 有害生物防除活性ピラゾール誘導体
US10874104B2 (en) 2016-02-18 2020-12-29 Syngenta Participations Ag Pesticidally active pryazole derivatives
WO2017188078A1 (ja) * 2016-04-28 2017-11-02 住友化学株式会社 複素環化合物
JP6931695B2 (ja) * 2016-04-29 2021-09-08 エフジーエイチ バイオテック,インコーポレーテッド 疾患の治療のための二置換ピラゾール化合物
AU2017323521B9 (en) 2016-09-07 2022-02-17 Fgh Biotech, Inc. Di-substituted pyrazole compounds for the treatment of diseases
KR101773442B1 (ko) 2017-02-15 2017-08-31 김순일 흡혈성 절지동물 기피제 조성물
WO2018185191A1 (en) 2017-04-05 2018-10-11 Syngenta Participations Ag Pesticidally active pyrazole derivatives
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AR112673A1 (es) 2017-08-11 2019-11-27 Syngenta Participations Ag Derivados de pirazol activos como plaguicidas
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EP3665166A1 (en) 2017-08-11 2020-06-17 Syngenta Participations AG Pesticidally active pyrazole derivatives
US11459318B2 (en) 2017-10-06 2022-10-04 Syngenta Participations Ag Pesticidally active pyrrole derivatives
EP3692038A1 (en) 2017-10-06 2020-08-12 Syngenta Participations AG Pesticidally active pyrrole derivatives
BR112020022763A2 (pt) * 2018-05-24 2021-02-02 Bayer Aktiengesellschaft processo para a produção de n-arilpirazóis halogenados
EP3802496A1 (de) * 2018-05-24 2021-04-14 Bayer Aktiengesellschaft Verfahren zur herstellung von substituierten n-arylpyrazolen
MX2020013827A (es) 2018-06-22 2021-03-25 Bayer Ag Proceso de preparacion de compuestos triciclicos.
EP3586630A1 (en) 2018-06-28 2020-01-01 Bayer AG Active compound combinations having insecticidal/acaricidal properties
EP3590927A1 (en) 2018-07-05 2020-01-08 Bayer Animal Health GmbH Novel compounds for controlling arthropods
AU2019387370A1 (en) 2018-11-30 2021-06-10 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
KR102809629B1 (ko) 2018-12-18 2025-05-20 디스커버리 퍼체이서 코퍼레이션 증가된 접촉 효능을 갖는 벡터 및 해충 방제를 위한 살충 제제
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