JP2016522195A5 - - Google Patents

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JP2016522195A5
JP2016522195A5 JP2016513374A JP2016513374A JP2016522195A5 JP 2016522195 A5 JP2016522195 A5 JP 2016522195A5 JP 2016513374 A JP2016513374 A JP 2016513374A JP 2016513374 A JP2016513374 A JP 2016513374A JP 2016522195 A5 JP2016522195 A5 JP 2016522195A5
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pain
compound
medicament
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JP2016513374A
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JP2016522195A (ja
JP6309616B2 (ja
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Priority claimed from EP13168165.2A external-priority patent/EP2803668A1/en
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JP2016513374A 2013-05-17 2014-05-16 新規な（シアノ−ジメチル−メチル）−イソオキサゾール及び−［１，３，４］チアジアゾール Active JP6309616B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13168165.2 2013-05-17
EP13168165.2A EP2803668A1 (en) 2013-05-17 2013-05-17 Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles
PCT/EP2014/060033 WO2014184327A1 (en) 2013-05-17 2014-05-16 Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles

Publications (3)

Publication Number Publication Date
JP2016522195A JP2016522195A (ja) 2016-07-28
JP2016522195A5 true JP2016522195A5 (enExample) 2017-06-22
JP6309616B2 JP6309616B2 (ja) 2018-04-11

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JP2016513374A Active JP6309616B2 (ja) 2013-05-17 2014-05-16 新規な（シアノ−ジメチル−メチル）−イソオキサゾール及び−［１，３，４］チアジアゾール

Country Status (24)

Country Link
US (7) US8865744B1 (enExample)
EP (2) EP2803668A1 (enExample)
JP (1) JP6309616B2 (enExample)
KR (1) KR102293386B1 (enExample)
CN (1) CN105229000B (enExample)
AR (1) AR096338A1 (enExample)
AU (1) AU2014267197B2 (enExample)
BR (1) BR112015028235A2 (enExample)
CA (1) CA2912463C (enExample)
CL (1) CL2015003286A1 (enExample)
DK (1) DK2997027T3 (enExample)
EA (1) EA031021B1 (enExample)
ES (1) ES2626396T3 (enExample)
IL (1) IL242309B (enExample)
MX (1) MX350885B (enExample)
NZ (1) NZ713614A (enExample)
PH (1) PH12015502523A1 (enExample)
PL (1) PL2997027T3 (enExample)
PT (1) PT2997027T (enExample)
TW (1) TW201536762A (enExample)
UA (1) UA118031C2 (enExample)
UY (1) UY35571A (enExample)
WO (1) WO2014184327A1 (enExample)
ZA (1) ZA201507957B (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2803668A1 (en) * 2013-05-17 2014-11-19 Boehringer Ingelheim International Gmbh Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles
UA117830C2 (uk) 2013-05-17 2018-10-10 Інсайт Корпорейшн Похідні біпіразолу як інгібітори jak
EP3824906A1 (en) 2016-12-21 2021-05-26 Amgen Inc. Anti-tnf alpha antibody formulations
CA3049389A1 (en) * 2017-01-06 2018-07-12 Clexio Biosciences Ltd. Topical detomidine formulations
BR122023022189A2 (pt) 2018-02-16 2024-02-20 Incyte Corporation Usos de inibidores da via de jak1 para o tratamento de distúrbios relacionados a citocinas
CN112423759A (zh) 2018-03-30 2021-02-26 因赛特公司 使用jak抑制剂治疗化脓性汗腺炎
IL298118B1 (en) 2020-06-02 2025-10-01 Incyte Corp Processes for preparing JAK1 inhibitor
WO2022125670A1 (en) 2020-12-08 2022-06-16 Incyte Corporation Jak1 pathway inhibitors for the treatment of vitiligo
DK4333840T3 (da) 2021-05-03 2025-11-24 Incyte Corp Jak1-vejinhibitorer til behandling af prurigo nodularis

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WO2011109324A1 (en) 2010-03-05 2011-09-09 Boehringer Ingelheim International Gmbh Tetrazole compounds which selectively modulate the cb2 receptor
JP5746764B2 (ja) 2010-07-22 2015-07-08 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を調節する化合物
EP2803668A1 (en) 2013-05-17 2014-11-19 Boehringer Ingelheim International Gmbh Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles

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