JP2016513681A5 - - Google Patents

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Publication number
JP2016513681A5
JP2016513681A5 JP2016502333A JP2016502333A JP2016513681A5 JP 2016513681 A5 JP2016513681 A5 JP 2016513681A5 JP 2016502333 A JP2016502333 A JP 2016502333A JP 2016502333 A JP2016502333 A JP 2016502333A JP 2016513681 A5 JP2016513681 A5 JP 2016513681A5
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JP
Japan
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optionally substituted
compound
alkyl
optionally
heteroaryl
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JP2016502333A
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English (en)
Japanese (ja)
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JP2016513681A (ja
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Priority claimed from PCT/US2014/027097 external-priority patent/WO2014152229A2/en
Publication of JP2016513681A publication Critical patent/JP2016513681A/ja
Publication of JP2016513681A5 publication Critical patent/JP2016513681A5/ja
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JP2016502333A 2013-03-14 2014-03-14 ロイコトリエンａ４加水分解酵素の阻害剤 Pending JP2016513681A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361781181P 2013-03-14 2013-03-14
US61/781,181 2013-03-14
PCT/US2014/027097 WO2014152229A2 (en) 2013-03-14 2014-03-14 Inhibitors of leukotriene a4 hydrolase

Publications (2)

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JP2016513681A JP2016513681A (ja) 2016-05-16
JP2016513681A5 true JP2016513681A5 (enExample) 2017-04-13

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ID=51581688

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JP2016502333A Pending JP2016513681A (ja) 2013-03-14 2014-03-14 ロイコトリエンａ４加水分解酵素の阻害剤

Country Status (10)

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US (2) US9856249B2 (enExample)
EP (1) EP2968264A4 (enExample)
JP (1) JP2016513681A (enExample)
KR (1) KR20150127245A (enExample)
AU (2) AU2014240042C1 (enExample)
BR (1) BR112015022226A2 (enExample)
CA (1) CA2906035A1 (enExample)
MX (1) MX2015011677A (enExample)
RU (1) RU2696559C2 (enExample)
WO (1) WO2014152229A2 (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
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DK1976828T3 (en) 2005-12-29 2017-03-06 Celtaxsys Inc DIAMINE DERIVATIVES AS INhibitors of Leukotriene A4 HYDROLASE
CN104144708B (zh) 2011-04-06 2017-07-28 德克萨斯大学系统董事会 基于脂质的纳米粒子
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AU2014249168B2 (en) 2013-03-12 2018-07-12 Celltaxis, Llc Methods of inhibiting leukotriene A4 hydrolase
EP2968264A4 (en) * 2013-03-14 2016-11-02 Celtaxsys Inc INHIBITORS OF LEUCOTRIENE A4 HYDROLASE
WO2014152536A2 (en) 2013-03-14 2014-09-25 Celtaxsys, Inc. Inhibitors of leukotriene a4 hydrolase
JP6534650B2 (ja) 2013-03-14 2019-06-26 セルタクシス，インコーポレイテッド ロイコトリエンａ４加水分解酵素の阻害剤
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TWI691486B (zh) * 2016-01-29 2020-04-21 日商東麗股份有限公司 環狀胺衍生物及其醫藥用途
JP7145154B2 (ja) * 2016-12-09 2022-09-30 セルタクシー、エルエルシー ロイコトリエンａ４ヒドロラーゼの阻害剤
CA3045954A1 (en) 2016-12-09 2018-06-14 Celtaxsys, Inc. Monamine and monoamine derivatives as inhibitors of leukotriene a4 hydrolase
WO2019232306A1 (en) 2018-05-31 2019-12-05 Celtaxsys, Inc. Method of reducing pulmonary exacerbations in respiratory disease patients
KR20230051227A (ko) 2020-08-14 2023-04-17 노파르티스 아게 헤테로아릴 치환된 스피로피페리디닐 유도체 및 이의 제약 용도

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