JP2015503610A5 - - Google Patents

Download PDF

Info

Publication number
JP2015503610A5
JP2015503610A5 JP2014551715A JP2014551715A JP2015503610A5 JP 2015503610 A5 JP2015503610 A5 JP 2015503610A5 JP 2014551715 A JP2014551715 A JP 2014551715A JP 2014551715 A JP2014551715 A JP 2014551715A JP 2015503610 A5 JP2015503610 A5 JP 2015503610A5
Authority
JP
Japan
Prior art keywords
compound according
pharmaceutical composition
crystalline form
compound
following characteristic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2014551715A
Other languages
English (en)
Japanese (ja)
Other versions
JP2015503610A (ja
JP6058698B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2013/050283 external-priority patent/WO2013105066A1/en
Publication of JP2015503610A publication Critical patent/JP2015503610A/ja
Publication of JP2015503610A5 publication Critical patent/JP2015503610A5/ja
Application granted granted Critical
Publication of JP6058698B2 publication Critical patent/JP6058698B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2014551715A 2012-01-13 2013-01-11 Ip受容体アゴニストの塩 Expired - Fee Related JP6058698B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261586324P 2012-01-13 2012-01-13
US61/586,324 2012-01-13
PCT/IB2013/050283 WO2013105066A1 (en) 2012-01-13 2013-01-11 Salts of an ip receptor agonist

Publications (3)

Publication Number Publication Date
JP2015503610A JP2015503610A (ja) 2015-02-02
JP2015503610A5 true JP2015503610A5 (enExample) 2016-02-25
JP6058698B2 JP6058698B2 (ja) 2017-01-11

Family

ID=47757663

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014551715A Expired - Fee Related JP6058698B2 (ja) 2012-01-13 2013-01-11 Ip受容体アゴニストの塩

Country Status (6)

Country Link
US (1) US9174985B2 (enExample)
EP (1) EP2802584B1 (enExample)
JP (1) JP6058698B2 (enExample)
CN (1) CN104169282B (enExample)
ES (1) ES2561353T3 (enExample)
WO (1) WO2013105066A1 (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101491938B1 (ko) 2010-07-14 2015-02-10 노파르티스 아게 Ip 수용체 효능제 헤테로시클릭 화합물
US10744223B2 (en) 2011-03-25 2020-08-18 Szent Co. Scented material compositions and articles for use with food and beverage
US9801969B2 (en) 2011-03-25 2017-10-31 Szent Bev Co. Scented attachment for containers
US9174985B2 (en) 2012-01-13 2015-11-03 Novartis Ag Salts of 7-(2,3-di-p-tolyl-7,8-dihydropyrido[2,3-b]pyrazin-5(6H)-yl)heptanoic acid as IP receptor agonists
UY34572A (es) 2012-01-13 2013-09-02 Novartis Ag Compuestos heterocíclicos agonistas del receptor ip
US9115129B2 (en) 2012-01-13 2015-08-25 Novartis Ag Substituted pyrido[2,3-B]pyrazines as IP receptor agonists
CN105189500A (zh) * 2013-02-13 2015-12-23 诺华股份有限公司 Ip受体激动剂杂环化合物
UA119247C2 (uk) 2013-09-06 2019-05-27 РОЙВЕНТ САЙЕНСИЗ ҐмбГ Спіроциклічні сполуки як інгібітори триптофангідроксилази
WO2015089137A1 (en) 2013-12-11 2015-06-18 Karos Pharmaceuticals, Inc. Acylguanidines as tryptophan hydroxylase inhibitors
WO2016109501A1 (en) 2014-12-30 2016-07-07 Karos Pharmaceuticals, Inc. Amide compounds as tryptophan hydroxylase inhibitors
US9611201B2 (en) 2015-03-05 2017-04-04 Karos Pharmaceuticals, Inc. Processes for preparing (R)-1-(5-chloro-[1,1′-biphenyl]-2-yl)-2,2,2-trifluoroethanol and 1-(5-chloro-[1,1′-biphenyl]-2-yl)-2,2,2-trifluoroethanone
CN105801578B (zh) * 2016-04-28 2018-06-22 华南理工大学 一种半饱和吡嗪衍生物的合成方法及应用
USD826047S1 (en) 2017-03-29 2018-08-21 Szent Co. Bottle ring
CN110877768B (zh) * 2017-05-05 2022-05-06 圣特公司 一种用于制作香味传递系统的方法
USD950384S1 (en) 2018-05-16 2022-05-03 Szent Co. Bottle
US11097877B2 (en) 2018-05-31 2021-08-24 Szent Co. Scent delivery and preservation systems and methods for beverage containers
WO2020099929A1 (en) 2018-11-14 2020-05-22 Roivant Sciences Gmbh A crystalline spirocyclic compound inhibitor of tryptophan hydroxylase 1 (tph1) for treating diseases or disorders associated with peripheral serotonin
US11018362B2 (en) 2019-05-30 2021-05-25 Lih-Ren Shiue System for generating electricity using oxygen from water
US11312528B2 (en) 2019-10-07 2022-04-26 Szent Co. Scented attachments for beverage cartons

Family Cites Families (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1016489B (it) 1974-03-18 1977-05-30 Isf Spa Inalatore
EP0865302B1 (de) 1995-12-07 2000-05-31 Jago Pharma Ag Inhalator zur mehrfachen dosisweisen abgabe eines pharmakologischen trockenpulvers
UA49878C2 (uk) 1996-02-21 2002-10-15 Шерінг Корпорейшн Пристрій для інгаляції порошку (варіанти)
US6166037A (en) 1997-08-28 2000-12-26 Merck & Co., Inc. Pyrrolidine and piperidine modulators of chemokine receptor activity
DE19834044A1 (de) 1998-07-29 2000-02-03 Bayer Ag Neue substituierte Pyrazolderivate
DE19834047A1 (de) 1998-07-29 2000-02-03 Bayer Ag Substituierte Pyrazolderivate
GB9913083D0 (en) 1999-06-04 1999-08-04 Novartis Ag Organic compounds
EP1632479B1 (en) 1999-05-04 2011-01-12 Schering Corporation Pharmaceutical compositions comprising CCR5 antagonizing piperazine derivatives
IL145742A0 (en) 1999-05-04 2002-07-25 Schering Corp Piperidine derivatives useful as ccr5 antagonists
DE19943639A1 (de) 1999-09-13 2001-03-15 Bayer Ag Dicarbonsäurederivate mit neuartigen pharmazeutischen Eigenschaften
DE19943636A1 (de) 1999-09-13 2001-03-15 Bayer Ag Neuartige Dicarbonsäurederivate mit pharmazeutischen Eigenschaften
DE19943634A1 (de) 1999-09-13 2001-04-12 Bayer Ag Neuartige Dicarbonsäurederivate mit pharmazeutischen Eigenschaften
DE19943635A1 (de) 1999-09-13 2001-03-15 Bayer Ag Neuartige Aminodicarbonsäurederivate mit pharmazeutischen Eigenschaften
AR031176A1 (es) 2000-11-22 2003-09-10 Bayer Ag Nuevos derivados de pirazolpiridina sustituidos con piridina
DE10110749A1 (de) 2001-03-07 2002-09-12 Bayer Ag Substituierte Aminodicarbonsäurederivate
DE10110750A1 (de) 2001-03-07 2002-09-12 Bayer Ag Neuartige Aminodicarbonsäurederivate mit pharmazeutischen Eigenschaften
DE10220570A1 (de) 2002-05-08 2003-11-20 Bayer Ag Carbamat-substituierte Pyrazolopyridine
ES2201907B1 (es) 2002-05-29 2005-06-01 Almirall Prodesfarma, S.A. Nuevos derivados de indolilpiperidina como potentes agentes antihistaminicos y antialergicos.
SE0202483D0 (sv) 2002-08-21 2002-08-21 Astrazeneca Ab Chemical compounds
TW200413372A (en) 2002-09-18 2004-08-01 Ono Pharmaceutical Co Derivatives of triazaspiro [5.5] undecane and medicants using such derivatives as effective ingredient
JP2006096662A (ja) 2002-09-18 2006-04-13 Sumitomo Pharmaceut Co Ltd 新規6−置換ウラシル誘導体及びアレルギー性疾患の治療剤
JP2004107299A (ja) 2002-09-20 2004-04-08 Japan Energy Corp 新規1−置換ウラシル誘導体及びアレルギー性疾患の治療剤
PE20040950A1 (es) 2003-02-14 2005-01-01 Theravance Inc DERIVADOS DE BIFENILO COMO AGONISTAS DE LOS RECEPTORES ADRENERGICOS ß2 Y COMO ANTAGONISTAS DE LOS RECEPTORES MUSCARINICOS
GB2407042B (en) 2003-10-17 2007-10-24 Vectura Ltd Inhaler
GB0410712D0 (en) 2004-05-13 2004-06-16 Novartis Ag Organic compounds
GB0413960D0 (en) 2004-06-22 2004-07-28 Novartis Ag Organic compounds
ES2270715B1 (es) * 2005-07-29 2008-04-01 Laboratorios Almirall S.A. Nuevos derivados de pirazina.
EP2300425A4 (en) * 2008-06-24 2012-03-21 Panmira Pharmaceuticals Llc PROSTAGLANDIN D2 RECEPTOR CYCLOALCANEÝBINDLUCK ANTAGONISTS
TWI368513B (en) * 2009-04-30 2012-07-21 Univ Kaohsiung Medical Synthesis of pulmodil and pulmodil-1, two chlorophenylpiperazine salt derivatives, and rhokinase-dependent inhibition activity on pulmonary artery endothelium dysfunction, medial wall thickness and vascular obstruction thereof
KR101491938B1 (ko) 2010-07-14 2015-02-10 노파르티스 아게 Ip 수용체 효능제 헤테로시클릭 화합물
US9174985B2 (en) 2012-01-13 2015-11-03 Novartis Ag Salts of 7-(2,3-di-p-tolyl-7,8-dihydropyrido[2,3-b]pyrazin-5(6H)-yl)heptanoic acid as IP receptor agonists
WO2013105058A1 (en) 2012-01-13 2013-07-18 Novartis Ag 7,8- dihydropyrido [3, 4 - b] pyrazines as ip receptor agonists for the treatment of pulmonary arterial hypertension (pah) and related disorders
US9115129B2 (en) 2012-01-13 2015-08-25 Novartis Ag Substituted pyrido[2,3-B]pyrazines as IP receptor agonists
WO2013105063A1 (en) 2012-01-13 2013-07-18 Novartis Ag Fused piperidines as ip receptor agonists for the treatment of pulmonary arterial hypertension (pah) and related disorders
WO2013105061A1 (en) 2012-01-13 2013-07-18 Novartis Ag Fused dihydropyrido [2,3 -b] pyrazines as ip receptor agonists for the treatment of pulmonary arterial hypertension (pah) and related disorders
UY34572A (es) 2012-01-13 2013-09-02 Novartis Ag Compuestos heterocíclicos agonistas del receptor ip
CN105189500A (zh) 2013-02-13 2015-12-23 诺华股份有限公司 Ip受体激动剂杂环化合物

Similar Documents

Publication Publication Date Title
JP2015503610A5 (enExample)
JP2014502641A5 (enExample)
JP2015520151A5 (enExample)
JP2020512337A5 (enExample)
JP2017528503A5 (enExample)
JP2019505529A5 (enExample)
JP2016505637A5 (enExample)
JP2016517857A5 (enExample)
JP2014518266A5 (enExample)
JP2016522835A5 (enExample)
FI2744810T4 (fi) Tenofoviirialafenamidihemifumaraatti
JP2017528507A5 (enExample)
JP2015522018A5 (enExample)
JP2012513416A5 (enExample)
JP2013542261A5 (enExample)
JP2018509438A5 (enExample)
JP2016522254A5 (enExample)
JP2010521516A5 (enExample)
HRP20151338T1 (hr) [4-(5-aminometil-2-fluoro-fenil)-piperidin-1-il]-[7-fluoro-1-(2-metoksi-etil)-4trifluorometoksi-1h-indol-3-il]metanon kao inhibitor triptaze mastocita
JP2015500223A5 (enExample)
JP2017526724A5 (enExample)
JP2019520344A5 (enExample)
JP2020505354A5 (enExample)
JP2014509653A5 (enExample)
JP2016510768A5 (enExample)