JP2015503560A5 - - Google Patents

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Publication number
JP2015503560A5
JP2015503560A5 JP2014550335A JP2014550335A JP2015503560A5 JP 2015503560 A5 JP2015503560 A5 JP 2015503560A5 JP 2014550335 A JP2014550335 A JP 2014550335A JP 2014550335 A JP2014550335 A JP 2014550335A JP 2015503560 A5 JP2015503560 A5 JP 2015503560A5
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JP
Japan
Prior art keywords
composition
solid dispersion
hcv
solid
polymer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2014550335A
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English (en)
Japanese (ja)
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JP2015503560A (ja
JP5781706B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2012/070349 external-priority patent/WO2013101550A1/en
Publication of JP2015503560A publication Critical patent/JP2015503560A/ja
Publication of JP2015503560A5 publication Critical patent/JP2015503560A5/ja
Application granted granted Critical
Publication of JP5781706B2 publication Critical patent/JP5781706B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2014550335A 2011-12-29 2012-12-18 Hcv阻害剤を含む固体組成物 Expired - Fee Related JP5781706B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161581146P 2011-12-29 2011-12-29
US61/581,146 2011-12-29
US201261645696P 2012-05-11 2012-05-11
US61/645,696 2012-05-11
PCT/US2012/070349 WO2013101550A1 (en) 2011-12-29 2012-12-18 Solid compositions comprising an hcv inhibitor

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015140513A Division JP2015227352A (ja) 2011-12-29 2015-07-14 Hcv阻害剤を含む固体組成物

Publications (3)

Publication Number Publication Date
JP2015503560A JP2015503560A (ja) 2015-02-02
JP2015503560A5 true JP2015503560A5 (enExample) 2015-03-12
JP5781706B2 JP5781706B2 (ja) 2015-09-24

Family

ID=47470243

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2014550335A Expired - Fee Related JP5781706B2 (ja) 2011-12-29 2012-12-18 Hcv阻害剤を含む固体組成物
JP2015140513A Pending JP2015227352A (ja) 2011-12-29 2015-07-14 Hcv阻害剤を含む固体組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2015140513A Pending JP2015227352A (ja) 2011-12-29 2015-07-14 Hcv阻害剤を含む固体組成物

Country Status (9)

Country Link
US (1) US20130172239A1 (enExample)
EP (2) EP2797586A1 (enExample)
JP (2) JP5781706B2 (enExample)
CN (1) CN104010631B (enExample)
CA (1) CA2857339C (enExample)
DE (1) DE212012000197U1 (enExample)
HK (1) HK1201186A1 (enExample)
MX (1) MX2014008008A (enExample)
WO (1) WO2013101550A1 (enExample)

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US8969588B2 (en) * 2012-06-05 2015-03-03 Gilead Pharmasset Llc Solid forms of an antiviral compound
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TW201446286A (zh) * 2013-01-31 2014-12-16 Gilead Pharmasset Llc 抗病毒化合物之固態分散調製劑
CN105228593B (zh) * 2013-03-15 2018-08-28 勃林格殷格翰国际有限公司 呈无定形状态的hcv抑制剂的固体口服剂型
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US20150023913A1 (en) 2013-07-02 2015-01-22 Bristol-Myers Squibb Company Hepatitis C Virus Inhibitors
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JP2016529293A (ja) * 2013-08-27 2016-09-23 ギリアド ファーマセット エルエルシー 2つの抗ウイルス化合物の組合せ製剤
US20160346198A1 (en) * 2014-02-05 2016-12-01 Merck Sharp & Dohme Corp. Novel disintegration systems for pharmaceutical dosage forms
EP3102210A4 (en) * 2014-02-05 2017-10-11 Merck Sharp & Dohme Corp. Pharmaceutical composition of selective hcv ns3/4a inhibitors
CA2937942A1 (en) * 2014-02-05 2015-08-13 Merck Sharp & Dohme Corp. Fixed-dose combinations of antiviral compounds
CA2943574A1 (en) * 2014-04-03 2015-10-08 Sandoz Ag Solid composition comprising amorphous sofosbuvir
TWI721947B (zh) 2014-06-11 2021-03-21 美商基利法瑪席特有限責任公司 抗病毒化合物的固態形式
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WO2016075588A1 (en) * 2014-11-11 2016-05-19 Sun Pharmaceutical Industries Limited Stable amorphous daclatasvir dihydrochloride
WO2016128453A1 (en) * 2015-02-13 2016-08-18 Sandoz Ag Pharmaceutical compositions comprising ledipasvir and sofosbuvir
WO2016145269A1 (en) 2015-03-12 2016-09-15 Teva Pharmaceuticals International Gmbh Solid state forms ledipasvir and processes for preparation of ledipasvir
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US20180228828A1 (en) * 2015-08-04 2018-08-16 Merck Sharp & Dohme Corp. Fixed-dose combinations of antiviral compounds
WO2017023714A1 (en) * 2015-08-04 2017-02-09 Merck Sharp & Dohme Corp. Fixed-dose combinations of antiviral compounds
US20180221282A1 (en) * 2015-08-04 2018-08-09 Merck Sharp & Dohme Corp. Methods for making pharmaceutical solid dosage forms of spray-dried dispersions
US20180228827A1 (en) * 2015-08-04 2018-08-16 Merck Sharp & Dohme Corp. Fixed-dose combinations of antiviral compounds
WO2017023631A1 (en) 2015-08-06 2017-02-09 Bristol-Myers Squibb Company Hepatitis c virus inhibitors
US20180271890A1 (en) * 2015-10-07 2018-09-27 Sandoz Ag Solid Pharmaceutical Composition Comprising Amorphous Sofosbuvir
WO2017072714A1 (en) 2015-10-30 2017-05-04 Lupin Limited Stable ledipasvir premix and process of preparation thereof
JOP20170127A1 (ar) * 2016-06-02 2017-12-02 Gilead Pharmasset Llc صيغة مشتركة مكونة من ثلاث مركبات مضادة للفيروسات
BR112019002729A2 (pt) 2016-08-12 2019-05-14 Sandoz Ag composição farmacêutica sólida e processo para preparar uma composição farmacêutica sólida
WO2018078536A1 (en) 2016-10-26 2018-05-03 Lupin Limited Stable solid dispersion of sofosbuvir and process for preparation thereof
CN106727516A (zh) * 2017-01-10 2017-05-31 山东省立医院 一种治疗丙型肝炎的药物组合物
WO2019134971A1 (en) * 2018-01-04 2019-07-11 Sandoz Ag Encapsulated particles comprising a pharmaceutically active ingredient
US11378965B2 (en) 2018-11-15 2022-07-05 Toyota Research Institute, Inc. Systems and methods for controlling a vehicle based on determined complexity of contextual environment
CN113209087B (zh) * 2020-02-05 2023-11-07 歌礼药业(浙江)有限公司 一种抑制冠状病毒的药物组合物及其用途
CN116887866A (zh) 2020-12-03 2023-10-13 巴特尔纪念研究院 聚合物纳米颗粒和dna纳米结构组合物及用于非病毒递送的方法
JP2024516108A (ja) 2021-04-07 2024-04-12 バテル・メモリアル・インスティテュート 非ウイルス性担体を同定および使用するための迅速な設計、構築、試験、および学習技術
NL2028762B1 (en) * 2021-07-16 2023-01-23 Seranovo Holding B V Micelle-generating formulations for enhanced bioavailability
KR102842201B1 (ko) * 2023-09-19 2025-08-06 한국해양과학기술원 Lng 추진 선박용 이산화탄소 액화 시스템 및 방법
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AU2005253957B2 (en) * 2004-06-08 2011-08-25 Janssen Pharmaceutica Nv Pharmaceutical compositions
WO2007109604A2 (en) * 2006-03-20 2007-09-27 Vertex Pharmaceuticals Incorporated Pharmaceutical compositions
US7964580B2 (en) * 2007-03-30 2011-06-21 Pharmasset, Inc. Nucleoside phosphoramidate prodrugs
PE20091041A1 (es) * 2007-10-19 2009-08-22 Abbott Gmbh & Co Kg Producto de dispersion solida que contiene un compuesto a base de n-aril urea
US20110207660A1 (en) * 2008-08-07 2011-08-25 Schering Corporation Pharmaceutical formulations of an hcv protease inhibitor in a solid molecular dispersion
MX340792B (es) * 2009-02-27 2016-07-25 Ortho-Mcneil-Janssen Pharmaceuticals Inc * Sal amorfa de un inhibidor macrociclico de virus de hepatitis c.
RS56654B8 (sr) * 2009-05-13 2021-06-30 Gilead Pharmasset Llc Antiviralna jedinjenja
US8937150B2 (en) * 2009-06-11 2015-01-20 Abbvie Inc. Anti-viral compounds
EA020031B1 (ru) * 2009-06-11 2014-08-29 Эббви Бахамаз Лтд. Противовирусные соединения
US8415374B2 (en) * 2009-10-12 2013-04-09 Bristol-Myers Squibb Company Combinations of hepatitis C virus inhibitors
NZ605440A (en) * 2010-06-10 2014-05-30 Abbvie Bahamas Ltd Solid compositions comprising an hcv inhibitor
TW201446286A (zh) * 2013-01-31 2014-12-16 Gilead Pharmasset Llc 抗病毒化合物之固態分散調製劑

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